Contents

Letters in Drug Design & Discovery, Volume 15 - Number 4

Biography

Meet Our Editorial Board Member

, 15(4): 335

James David Adams


DOI: 10.2174/157018081504180312110402




Research Article

Synthesis, Anti-Methicillin-resistant S. aureus (MRSA) Evaluation, Quantitative Structure-Activity Relationship and Molecular Modeling Studies of Some Novel Bis-indoles as Prospective MRSA Pyruvate Kinase Inhibitors

, 15(4): 336 - 346

Mardia T. El Sayed*, Nermien M. Sabry, Nehal A. Hamdy, Andrey Voronkov, Ifedayo V. Ogungbe , Konstantin Balakin and Mohamed S. Abdel-Aziz


DOI: 10.2174/1570180815666171213144922





Research Article

Microwave-assisted Synthesis and Antifungal Activity of Novel 1,2,4- Triazole Thioether Derivatives Containing Pyrimidine Moiety

, 15(4): 347 - 352

Meng Xu, Ya-Bo Zhu, Mei Wang, Ikhlas A. Khan, Xing-Hai Liu and Jian-Quan Weng*


DOI: 10.2174/1570180814666170602082440





Research Article

Anti-MRSA (Multidrug Resistant Staphylococcus aureus) Activity of 3-Substituted Coumarins

, 15(4): 353 - 362

Uzma Salar, Khalid Mohammed Khan*, Humaira Muhammad, Muhammed Imran Fakhri, Sanaullah, Shahnaz Perveen and Muhammed Iqbal Choudhary


DOI: 10.2174/1570180814666170619121844





Research Article

Synthesis and Anti-influenza Activity of Novel Thiadiazole, Oxadiazole and Triazole Based Scaffolds

, 15(4): 363 - 374

Samar S. Tawfik, Abdelbasset A. Farahat*, Magda A.-A El-Sayed, Atif S. Tantawy, Ola Bagato and Mohamed A. Ali


DOI: 10.2174/1570180814666170512122832





Research Article

Exploration of Some Thiazolidine-2,4-dione and 2-Oxoindoline Derivatives Incorporating 3,4,5-Trimethoxybenzyl Moiety as Novel Anticancer Agents

, 15(4): 375 - 387

Le Cong Huan, Hai Pham-The, Huong Le-Thi-Thu, Tran Phuong Thao, Do Nguyet Que, Nguyen-Thu Trang, Phan Thi Phuong Dung, Minji Pyo, Sang-Bae Han, Nguyen Thi Thuan* and Nguyen-Hai Nam*


DOI: 10.2174/1570180814666170605122552





Research Article

Design, Synthesis and Biological Evaluation of Some Novel Thiazole-2- Carboxamide Derivatives as Antitumor Agents

, 15(4): 388 - 397

Haibo Wang*, Zhengjiang Cai, Shan Zheng, Huidan Ma, Haiming Lin and Xiaohe Zheng*


DOI: 10.2174/1570180814666170704143015





Research Article

Design, Synthesis, and Screening of Hybrid Benzothiazolyl-Oxadiazoles as Anticonvulsant Agents

, 15(4): 398 - 405

Sheikh Murtuja, Mohammad Shaquiquzzaman and Mohammad Amir*


DOI: 10.2174/1570180814666170526154914





Research Article

Synthesis and Evaluation of the Anticonvulsant Activities of New 5-substitued-[1,2,4]triazolo[4,3-a]quinoxalin-4(5H)-one Derivatives

, 15(4): 406 - 413

Guo-Rui Zhang, Yang Ren, Xiu-Mei Yin* and Zhe-Shan Quan


DOI: 10.2174/1570180814666170619094408





Research Article

Fighting Against Alzheimer's Disease: Synthesis of New Pyrazoline and Benzothiazole Derivatives as New Acetylcholinesterase and MAO Inhibitors

, 15(4): 414 - 427

Gulhan Turan-Zitouni*, Weiam Hussein, Begum Nurpelin Saglik, Merve Baysal and Zafer Asim Kaplancikli


DOI: 10.2174/1570180814666170704144917





Research Article

Synthesis and Urease Inhibitory Activity of Some 5-Aminomethylene Barbituric/Thiobarbituric Acid Derivatives

, 15(4): 428 - 436

Mehdi Asadi, Mohammad Mahdavi, Shabnam Mahernia, Zahra Rezaei, Maliheh Safavi, Mina Saeedi and Massoud Amanlou*


DOI: 10.2174/1570180814666170727142928





Research Article

Design, Synthesis and Pharmacological Evaluation of Some Novel Tetrahydrocarbazoles as Potential COX-2 Inhibitors

, 15(4): 437 - 449

Padmavathi Sakinala, Rupesh Chikhale and Madhukar Tajne*


DOI: 10.2174/1570180814666170602084037





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