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Letters in Drug Design & Discovery

Volume 18, 12 Issues, 2021
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

In the current pandemic scenario, publication process of all articles related to Coronavirus will be expedited, for timely publication of much needed research


Letters in Drug Design & Discovery, Volume 15 - Number 4

Research Article

Synthesis, Anti-Methicillin-resistant S. aureus (MRSA) Evaluation, Quantitative Structure-Activity Relationship and Molecular Modeling Studies of Some Novel Bis-indoles as Prospective MRSA Pyruvate Kinase Inhibitors

, 15(4): 336 - 346

Mardia T. El Sayed*, Nermien M. Sabry, Nehal A. Hamdy, Andrey Voronkov, Ifedayo V. Ogungbe , Konstantin Balakin and Mohamed S. Abdel-Aziz

DOI: 10.2174/1570180815666171213144922

Research Article

Microwave-assisted Synthesis and Antifungal Activity of Novel 1,2,4- Triazole Thioether Derivatives Containing Pyrimidine Moiety

, 15(4): 347 - 352

Meng Xu, Ya-Bo Zhu, Mei Wang, Ikhlas A. Khan, Xing-Hai Liu and Jian-Quan Weng*

DOI: 10.2174/1570180814666170602082440

Research Article

Anti-MRSA (Multidrug Resistant Staphylococcus aureus) Activity of 3-Substituted Coumarins

, 15(4): 353 - 362

Uzma Salar, Khalid Mohammed Khan*, Humaira Muhammad, Muhammed Imran Fakhri, Sanaullah, Shahnaz Perveen and Muhammed Iqbal Choudhary

DOI: 10.2174/1570180814666170619121844

Research Article

Synthesis and Anti-influenza Activity of Novel Thiadiazole, Oxadiazole and Triazole Based Scaffolds

, 15(4): 363 - 374

Samar S. Tawfik, Abdelbasset A. Farahat*, Magda A.-A El-Sayed, Atif S. Tantawy, Ola Bagato and Mohamed A. Ali

DOI: 10.2174/1570180814666170512122832

Research Article

Exploration of Some Thiazolidine-2,4-dione and 2-Oxoindoline Derivatives Incorporating 3,4,5-Trimethoxybenzyl Moiety as Novel Anticancer Agents

, 15(4): 375 - 387

Le Cong Huan, Hai Pham-The, Huong Le-Thi-Thu, Tran Phuong Thao, Do Nguyet Que, Nguyen-Thu Trang, Phan Thi Phuong Dung, Minji Pyo, Sang-Bae Han, Nguyen Thi Thuan* and Nguyen-Hai Nam*

DOI: 10.2174/1570180814666170605122552

Research Article

Design, Synthesis and Biological Evaluation of Some Novel Thiazole-2- Carboxamide Derivatives as Antitumor Agents

, 15(4): 388 - 397

Haibo Wang*, Zhengjiang Cai, Shan Zheng, Huidan Ma, Haiming Lin and Xiaohe Zheng*

DOI: 10.2174/1570180814666170704143015

Research Article

Design, Synthesis, and Screening of Hybrid Benzothiazolyl-Oxadiazoles as Anticonvulsant Agents

, 15(4): 398 - 405

Sheikh Murtuja, Mohammad Shaquiquzzaman and Mohammad Amir*

DOI: 10.2174/1570180814666170526154914

Research Article

Synthesis and Evaluation of the Anticonvulsant Activities of New 5-substitued-[1,2,4]triazolo[4,3-a]quinoxalin-4(5H)-one Derivatives

, 15(4): 406 - 413

Guo-Rui Zhang, Yang Ren, Xiu-Mei Yin* and Zhe-Shan Quan

DOI: 10.2174/1570180814666170619094408

Research Article

Fighting Against Alzheimer's Disease: Synthesis of New Pyrazoline and Benzothiazole Derivatives as New Acetylcholinesterase and MAO Inhibitors

, 15(4): 414 - 427

Gulhan Turan-Zitouni*, Weiam Hussein, Begum Nurpelin Saglik, Merve Baysal and Zafer Asim Kaplancikli

DOI: 10.2174/1570180814666170704144917

Research Article

Synthesis and Urease Inhibitory Activity of Some 5-Aminomethylene Barbituric/Thiobarbituric Acid Derivatives

, 15(4): 428 - 436

Mehdi Asadi, Mohammad Mahdavi, Shabnam Mahernia, Zahra Rezaei, Maliheh Safavi, Mina Saeedi and Massoud Amanlou*

DOI: 10.2174/1570180814666170727142928

Research Article

Design, Synthesis and Pharmacological Evaluation of Some Novel Tetrahydrocarbazoles as Potential COX-2 Inhibitors

, 15(4): 437 - 449

Padmavathi Sakinala, Rupesh Chikhale and Madhukar Tajne*

DOI: 10.2174/1570180814666170602084037


K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 1.05

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