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Letters in Drug Design & Discovery

Volume 17, 12 Issues, 2020
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

In the current pandemic scenario, publication process of all articles related to Coronavirus will be expedited, for timely publication of much needed research

Contents

Letters in Drug Design & Discovery, Volume 15 - Number 4


Research Article

Synthesis, Anti-Methicillin-resistant S. aureus (MRSA) Evaluation, Quantitative Structure-Activity Relationship and Molecular Modeling Studies of Some Novel Bis-indoles as Prospective MRSA Pyruvate Kinase Inhibitors

, 15(4): 336 - 346

Mardia T. El Sayed*, Nermien M. Sabry, Nehal A. Hamdy, Andrey Voronkov, Ifedayo V. Ogungbe , Konstantin Balakin and Mohamed S. Abdel-Aziz


DOI: 10.2174/1570180815666171213144922



Research Article

Microwave-assisted Synthesis and Antifungal Activity of Novel 1,2,4- Triazole Thioether Derivatives Containing Pyrimidine Moiety

, 15(4): 347 - 352

Meng Xu, Ya-Bo Zhu, Mei Wang, Ikhlas A. Khan, Xing-Hai Liu and Jian-Quan Weng*


DOI: 10.2174/1570180814666170602082440



Research Article

Anti-MRSA (Multidrug Resistant Staphylococcus aureus) Activity of 3-Substituted Coumarins

, 15(4): 353 - 362

Uzma Salar, Khalid Mohammed Khan*, Humaira Muhammad, Muhammed Imran Fakhri, Sanaullah, Shahnaz Perveen and Muhammed Iqbal Choudhary


DOI: 10.2174/1570180814666170619121844



Research Article

Synthesis and Anti-influenza Activity of Novel Thiadiazole, Oxadiazole and Triazole Based Scaffolds

, 15(4): 363 - 374

Samar S. Tawfik, Abdelbasset A. Farahat*, Magda A.-A El-Sayed, Atif S. Tantawy, Ola Bagato and Mohamed A. Ali


DOI: 10.2174/1570180814666170512122832



Research Article

Exploration of Some Thiazolidine-2,4-dione and 2-Oxoindoline Derivatives Incorporating 3,4,5-Trimethoxybenzyl Moiety as Novel Anticancer Agents

, 15(4): 375 - 387

Le Cong Huan, Hai Pham-The, Huong Le-Thi-Thu, Tran Phuong Thao, Do Nguyet Que, Nguyen-Thu Trang, Phan Thi Phuong Dung, Minji Pyo, Sang-Bae Han, Nguyen Thi Thuan* and Nguyen-Hai Nam*


DOI: 10.2174/1570180814666170605122552



Research Article

Design, Synthesis and Biological Evaluation of Some Novel Thiazole-2- Carboxamide Derivatives as Antitumor Agents

, 15(4): 388 - 397

Haibo Wang*, Zhengjiang Cai, Shan Zheng, Huidan Ma, Haiming Lin and Xiaohe Zheng*


DOI: 10.2174/1570180814666170704143015



Research Article

Design, Synthesis, and Screening of Hybrid Benzothiazolyl-Oxadiazoles as Anticonvulsant Agents

, 15(4): 398 - 405

Sheikh Murtuja, Mohammad Shaquiquzzaman and Mohammad Amir*


DOI: 10.2174/1570180814666170526154914



Research Article

Synthesis and Evaluation of the Anticonvulsant Activities of New 5-substitued-[1,2,4]triazolo[4,3-a]quinoxalin-4(5H)-one Derivatives

, 15(4): 406 - 413

Guo-Rui Zhang, Yang Ren, Xiu-Mei Yin* and Zhe-Shan Quan


DOI: 10.2174/1570180814666170619094408



Research Article

Fighting Against Alzheimer's Disease: Synthesis of New Pyrazoline and Benzothiazole Derivatives as New Acetylcholinesterase and MAO Inhibitors

, 15(4): 414 - 427

Gulhan Turan-Zitouni*, Weiam Hussein, Begum Nurpelin Saglik, Merve Baysal and Zafer Asim Kaplancikli


DOI: 10.2174/1570180814666170704144917



Research Article

Synthesis and Urease Inhibitory Activity of Some 5-Aminomethylene Barbituric/Thiobarbituric Acid Derivatives

, 15(4): 428 - 436

Mehdi Asadi, Mohammad Mahdavi, Shabnam Mahernia, Zahra Rezaei, Maliheh Safavi, Mina Saeedi and Massoud Amanlou*


DOI: 10.2174/1570180814666170727142928



Research Article

Design, Synthesis and Pharmacological Evaluation of Some Novel Tetrahydrocarbazoles as Potential COX-2 Inhibitors

, 15(4): 437 - 449

Padmavathi Sakinala, Rupesh Chikhale and Madhukar Tajne*


DOI: 10.2174/1570180814666170602084037




Editor-in-Chief

K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
Biography
View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 1.05

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