Contents

Letters in Drug Design & Discovery, Volume 14 - Number 9


Research Article

Docking-based 3D-QSAR Studies of Phosphodiesterase 9A Inhibitors

, 14(9): 986 - 998

Changji Tan, Yinuo Wu, Yongxian Shao, Haibin Luo, Xuehua Zheng and Laiyou Wang


DOI: 10.2174/1570180814666170110124314



Research Article

Quantitative Structure Activity Relationship (QSAR) of Methylated Polyphenol Derivatives as Permeability Glycoprotein (P-gp) Inhibitors: A Comparison of Different Training and Test Set Selection Methods

, 14(9): 999 - 1007

Paria Ghaemian and Ali Shayanfar


DOI: 10.2174/1570180814666170126150447



Research Article

Synthesis and Anticancer Studies of Novel N-benzyl Pyridazino ne Derivatives

, 14(9): 1008 - 1013

Mohamed Elagawany, Mohamed A. Ibrahim, Tarek S. Ibrahim, Amany M.M. AL-Mahmoudy, Alaa Moawad, Mohammed M. Ghoneim, Mohamed M. Radwan and Siva S. Panda


DOI: 10.2174/1570180814666170223111312



Research Article

Synthesis and Antimicrobial Activities of Hybrid Heterocyclic Molecules Based on 1-(4-Fluorophenyl)piperazine Skeleton

, 14(9): 1014 - 1034

Serap Basoglu Ozdemir, Neslihan Demirbas, Yıldız Uygun Cebeci, Hacer Bayrak, Arif Mermer, Sule Ceylan and Ahmet Demirbas


DOI: 10.2174/1570180814666170113145023



Research Article

Synthesis, Molecular Docking Studies and Biological Evaluation o f 3-Iminoaurones as Acetylcholinesterase and Butyrylcholinesterase Inhibitors

, 14(9): 1035 - 1041

Ehsan Ullah Mughal, Amina Sadiq, Bilal Ahmad Khan, Muhammad Naveed Zafar, Ishtiaq Ahmed and Muhammad Zubair


DOI: 10.2174/1570180814666170106123959



Research Article

Antimicrobial and Cytotoxicity Activities of 2-(aryl)-3-(benzo[d][1,3] dioxol-5-yl)thiazolidin-4-ones

, 14(9): 1042 - 1047

Silvana P. Souza, Hellen G. Masteloto, Daniel S. da Silva, Juliana H. Azambuja, Elizandra Braganhol, Juliana S. Ribeiro, Rafael G. Lund and Wilson Cunico


DOI: 10.2174/1570180814666170106143418



Research Article

Multiplication of Mycobacterium tuberculosis in Peripheral Blood of Mice and Effect of Anti-tubercular Drugs on Bacteremia

, 14(9): 1048 - 1052

Richa Dwivedi, Shubhra Singh, Priyanka Trivedi and Vinita Chaturvedi


DOI: 10.2174/1570180814666170223171215



Research Article

Antiproliferative Activity of Olive Oil Phenolics against Human Melan oma Cells

, 14(9): 1053 - 1059

A. L.M. Batista de Carvalho, F. Caselli, V. Rodrigues, F. Paiva-Martins and M.P. M. Marques


DOI: 10.2174/1570180814666170110145658



Research Article

Combination of Irbesartan with Amlodipine Enhances Nitrate/Nitrite Generation by Angiotensin II-exposed Endothelial Cells

, 14(9): 1060 - 1064

Yuji Ishibashi, Takanori Matsui, Nobutaka Nakamura and Sho-ichi Yamagishi


DOI: 10.2174/1570180814666170102154739



Research Article

Design, Synthesis and Evaluation of Dual-targeting Prodrug Co-modified by Organic Amine and L-ascorbic Acid for CNS Delivery

, 14(9): 1065 - 1072

Shubing Qiu, Yi Zhao, Sha Liu, Xiaocen Li, Li Guo, Li Hai and Yong Wu


DOI: 10.2174/1570180814666161230161152



Research Article

Design, Synthesis, Characterization, Molecular Docking, ADME Properties and In Vivo Antipsychotic Activity of Aripiprazole Related Drugs Candidates

, 14(9): 1073 - 1085

Selvarasu Sekar, Srinivasan Pazhamalai, Ganesan Ariharasivakumar and Mannathusamy Gopalakrishnan


DOI: 10.2174/1570180814666161207143742



Review Article

A Brief Overview on Chemistry and Biology of Benzoxepine

, 14(9): 1086 - 1098

Naveen Kuntala, Jhonsee R. Telu, Jaya S. Anireddy and Sarbani Pal


DOI: 10.2174/1570180814666161227125227



Review Article

Homology Modeling in Drug Discovery-an Update on the Last Decade

, 14(9): 1099 - 1111

Geraldene Munsamy and Mahmoud E. S. Soliman


DOI: 10.2174/1570180814666170110122027




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