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Letters in Drug Design & Discovery

Volume 18, 12 Issues, 2021
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

In the current pandemic scenario, publication process of all articles related to Coronavirus will be expedited, for timely publication of much needed research


Letters in Drug Design & Discovery, Volume 14 - Number 9

Research Article

Docking-based 3D-QSAR Studies of Phosphodiesterase 9A Inhibitors

, 14(9): 986 - 998

Changji Tan, Yinuo Wu, Yongxian Shao, Haibin Luo, Xuehua Zheng* and Laiyou Wang*

DOI: 10.2174/1570180814666170110124314

Research Article

Quantitative Structure Activity Relationship (QSAR) of Methylated Polyphenol Derivatives as Permeability Glycoprotein (P-gp) Inhibitors: A Comparison of Different Training and Test Set Selection Methods

, 14(9): 999 - 1007

Paria Ghaemian and Ali Shayanfar*

DOI: 10.2174/1570180814666170126150447

Research Article

Synthesis and Anticancer Studies of Novel N-benzyl Pyridazino ne Derivatives

, 14(9): 1008 - 1013

Mohamed Elagawany, Mohamed A. Ibrahim, Tarek S. Ibrahim, Amany M.M. AL-Mahmoudy, Alaa Moawad, Mohammed M. Ghoneim, Mohamed M. Radwan and Siva S. Panda*

DOI: 10.2174/1570180814666170223111312

Research Article

Synthesis and Antimicrobial Activities of Hybrid Heterocyclic Molecules Based on 1-(4-Fluorophenyl)piperazine Skeleton

, 14(9): 1014 - 1034

Serap Basoglu Ozdemir, Neslihan Demirbas*, Yıldız Uygun Cebeci, Hacer Bayrak, Arif Mermer, Sule Ceylan and Ahmet Demirbas

DOI: 10.2174/1570180814666170113145023

Research Article

Synthesis, Molecular Docking Studies and Biological Evaluation o f 3-Iminoaurones as Acetylcholinesterase and Butyrylcholinesterase Inhibitors

, 14(9): 1035 - 1041

Ehsan Ullah Mughal*, Amina Sadiq, Bilal Ahmad Khan, Muhammad Naveed Zafar, Ishtiaq Ahmed and Muhammad Zubair

DOI: 10.2174/1570180814666170106123959

Research Article

Antimicrobial and Cytotoxicity Activities of 2-(aryl)-3-(benzo[d][1,3] dioxol-5-yl)thiazolidin-4-ones

, 14(9): 1042 - 1047

Silvana P. Souza, Hellen G. Masteloto, Daniel S. da Silva, Juliana H. Azambuja, Elizandra Braganhol, Juliana S. Ribeiro, Rafael G. Lund and Wilson Cunico*

DOI: 10.2174/1570180814666170106143418

Research Article

Multiplication of Mycobacterium tuberculosis in Peripheral Blood of Mice and Effect of Anti-tubercular Drugs on Bacteremia

, 14(9): 1048 - 1052

Richa Dwivedi, Shubhra Singh, Priyanka Trivedi and Vinita Chaturvedi*

DOI: 10.2174/1570180814666170223171215

Research Article

Antiproliferative Activity of Olive Oil Phenolics against Human Melan oma Cells

, 14(9): 1053 - 1059

A. L.M. Batista de Carvalho, F. Caselli, V. Rodrigues, F. Paiva-Martins and M.P. M. Marques*

DOI: 10.2174/1570180814666170110145658

Research Article

Combination of Irbesartan with Amlodipine Enhances Nitrate/Nitrite Generation by Angiotensin II-exposed Endothelial Cells

, 14(9): 1060 - 1064

Yuji Ishibashi, Takanori Matsui, Nobutaka Nakamura and Sho-ichi Yamagishi*

DOI: 10.2174/1570180814666170102154739

Research Article

Design, Synthesis and Evaluation of Dual-targeting Prodrug Co-modified by Organic Amine and L-ascorbic Acid for CNS Delivery

, 14(9): 1065 - 1072

Shubing Qiu, Yi Zhao, Sha Liu, Xiaocen Li, Li Guo, Li Hai* and Yong Wu*

DOI: 10.2174/1570180814666161230161152

Research Article

Design, Synthesis, Characterization, Molecular Docking, ADME Properties and In Vivo Antipsychotic Activity of Aripiprazole Related Drugs Candidates

, 14(9): 1073 - 1085

Selvarasu Sekar, Srinivasan Pazhamalai, Ganesan Ariharasivakumar and Mannathusamy Gopalakrishnan*

DOI: 10.2174/1570180814666161207143742

Review Article

A Brief Overview on Chemistry and Biology of Benzoxepine

, 14(9): 1086 - 1098

Naveen Kuntala, Jhonsee R. Telu, Jaya S. Anireddy and Sarbani Pal*

DOI: 10.2174/1570180814666161227125227

Review Article

Homology Modeling in Drug Discovery-an Update on the Last Decade

, 14(9): 1099 - 1111

Geraldene Munsamy and Mahmoud E. S. Soliman*

DOI: 10.2174/1570180814666170110122027


K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 1.05


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