Letters in Drug Design & Discovery, Volume 14 - Number 5


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, 14(5): 507

Gyorgy Keglevich

DOI: 10.2174/157018081405170406182644

Research Article

The Decisive Role of Mutual Arrangement of Hydroxy and Methoxy Groups in (3(4)-hydroxy-4(3)-methoxyphenyl)-4,7-dimethyl-3,4,4a,5,8,8ahexahydro- 2H-chromene-4,8-diols in their Biological Activity

, 14(5): 508 - 514

Alla Pavlova, Oksana Patrusheva, Irina Il`ina, Konstantin Volcho, Tat`yana Tolstikova and Nariman Salakhutdinov

DOI: 10.2174/1570180813666161102142642

Research Article

Possible Binding Mode Analysis of Pyrazolo-triazole Hybrids as Potential Anticancer Agents through Validated Molecular Docking and 3D-QSAR Modeling Approaches

, 14(5): 515 - 527

Siekh Abdul Amin, Nilanjan Adhikari, Ram K. Agrawal, Tarun Jha and Shovanlal Gayen

DOI: 10.2174/1570180813666160916153017

Research Article

Synthesis of Novel 4-(Dimethylaminoalkyl)piperazine-1-carbodithioa t e Derivatives as Cholinesterase Inhibitors

, 14(5): 528 - 539

Ulviye Acar Cevik, Serkan Levent, Begum Nurpelin Saglık, Yusuf Ozkay and Zafer Asım Kaplancıklı

DOI: 10.2174/1570180813666160923105636

Research Article

Synthesis, Docking and Antidiabetic Activity of Some Newer Benzamide Derivatives as Potential Glucokinase Activators

, 14(5): 540 - 553

Rohit Singh, Viney Lather, Deepti Pandita, Vikramjeet Judge, Karthikeyan N. Arumugam and Ajmer Singh Grewal

DOI: 10.2174/1570180813666160819125342

Research Article

Cytotoxic, Apoptotic and DNA Synthesis Inhibitory Effects of Some Thiazole Derivatives

, 14(5): 554 - 566

Gulsen Akalın Ciftci, Mehlika Dilek Altıntop, Halide Edip Temel, Ahmet Ozdemir and Zafer Asım Kaplancıklı

DOI: 10.2174/1570180813666160907170553

Research Article

Synthesis of Phosphorylated Derivatives of 2', 3'-O-Isopropylidene Adenosine and their In Ovo Antiviral Activity

, 14(5): 567 - 572

Syed Rasheed, Chamarthi Naga Raju, Golla Madhava, Chennamsetty Subramanyam, Shaik Thaslim Basha, Avilala Janardhan and Golla Narasimha

DOI: 10.2174/1570180813666161020112309

Research Article

Synthesis of Mannich Bases by Two Different Methods and Evaluation of their Acetylcholine Esterase and Carbonic Anhydrase Inhibitory Activities

, 14(5): 573 - 580

Halise I. Gul, Alkan Demirtas, Gokbay Ucar, Parham Taslimi and İlhami Gulcin

DOI: 10.2174/1570180814666161128120612

Research Article

Computational Analysis of Pyridopyrimidine-based Polo Like Kinase 2 (PLK2) Inhibitors: Examining the Structural Basis for Anticancer Activity

, 14(5): 581 - 596

Anand Balupuri, Pavithra K. Balasubramanian and Seung Joo Cho

DOI: 10.2174/1570180813666160831113237

Research Article

In Vivo Antimalarial and In Vitro Antileishmanial Activity of 4- Aminoquinoline Derivatives Hybridized to Isoniazid or Sulfa or Hydrazine Groups

, 14(5): 597 - 604

Roberta R. Soares, Luciana M. R. Antinarelli, Isabela de O. Souza, Isabela de O. Souza, Fernanda V. Lopes, Kézia K. G. Scopel, Elaine S. Coimbra, Adilson D. da Silva and Clarice Abramo

DOI: 10.2174/1570180813666160927113743

Research Article

Vitamin B12 Controlled Release with Crosslinked Poly (Acrylic Acid) and Poly (Methacrylic Acid) Based on Chitosan and Starch as pH Sensitive Hydrogels

, 14(5): 605 - 612

Massomeh Ghorbanloo and Somaieh Tarasi

DOI: 10.2174/1570180814666161118150532

Research Article

Quorum Sensing Inhibitor Activities of Celecoxib Derivatives in Pseudomonas aeruginosa

, 14(5): 613 - 618

Seyhan Ulusoy, Sevil Senkardes, Inci Coskun, Gulgun Bosgelmez-Tınaz, Laurent Soulere, Yves Queneau and S. Guniz Kucukguzel

DOI: 10.2174/1570180814666161121120719

Review Article

NF-κB Inhibitors in Head and Neck Cancer

, 14(5): 619 - 633

Siddavaram Nagini, Kranthi Kiran Kishore Tanagala and Indranil Chattopadhyay

DOI: 10.2174/1570180813666160926095002

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