Contents

Letters in Drug Design & Discovery, Volume 14 - Number 5


Research Article

The Decisive Role of Mutual Arrangement of Hydroxy and Methoxy Groups in (3(4)-hydroxy-4(3)-methoxyphenyl)-4,7-dimethyl-3,4,4a,5,8,8ahexahydro- 2H-chromene-4,8-diols in their Biological Activity

, 14(5): 508 - 514

Alla Pavlova, Oksana Patrusheva, Irina Il`ina, Konstantin Volcho, Tat`yana Tolstikova and Nariman Salakhutdinov


DOI: 10.2174/1570180813666161102142642



Research Article

Possible Binding Mode Analysis of Pyrazolo-triazole Hybrids as Potential Anticancer Agents through Validated Molecular Docking and 3D-QSAR Modeling Approaches

, 14(5): 515 - 527

Siekh Abdul Amin, Nilanjan Adhikari, Ram K. Agrawal, Tarun Jha and Shovanlal Gayen


DOI: 10.2174/1570180813666160916153017



Research Article

Synthesis of Novel 4-(Dimethylaminoalkyl)piperazine-1-carbodithioa t e Derivatives as Cholinesterase Inhibitors

, 14(5): 528 - 539

Ulviye Acar Cevik, Serkan Levent, Begum Nurpelin Saglık, Yusuf Ozkay and Zafer Asım Kaplancıklı


DOI: 10.2174/1570180813666160923105636



Research Article

Synthesis, Docking and Antidiabetic Activity of Some Newer Benzamide Derivatives as Potential Glucokinase Activators

, 14(5): 540 - 553

Rohit Singh, Viney Lather, Deepti Pandita, Vikramjeet Judge, Karthikeyan N. Arumugam and Ajmer Singh Grewal


DOI: 10.2174/1570180813666160819125342



Research Article

Cytotoxic, Apoptotic and DNA Synthesis Inhibitory Effects of Some Thiazole Derivatives

, 14(5): 554 - 566

Gulsen Akalın Ciftci, Mehlika Dilek Altıntop, Halide Edip Temel, Ahmet Ozdemir and Zafer Asım Kaplancıklı


DOI: 10.2174/1570180813666160907170553



Research Article

Synthesis of Phosphorylated Derivatives of 2', 3'-O-Isopropylidene Adenosine and their In Ovo Antiviral Activity

, 14(5): 567 - 572

Syed Rasheed, Chamarthi Naga Raju, Golla Madhava, Chennamsetty Subramanyam, Shaik Thaslim Basha, Avilala Janardhan and Golla Narasimha


DOI: 10.2174/1570180813666161020112309



Research Article

Synthesis of Mannich Bases by Two Different Methods and Evaluation of their Acetylcholine Esterase and Carbonic Anhydrase Inhibitory Activities

, 14(5): 573 - 580

Halise I. Gul, Alkan Demirtas, Gokbay Ucar, Parham Taslimi and İlhami Gulcin


DOI: 10.2174/1570180814666161128120612



Research Article

Computational Analysis of Pyridopyrimidine-based Polo Like Kinase 2 (PLK2) Inhibitors: Examining the Structural Basis for Anticancer Activity

, 14(5): 581 - 596

Anand Balupuri, Pavithra K. Balasubramanian and Seung Joo Cho


DOI: 10.2174/1570180813666160831113237



Research Article

In Vivo Antimalarial and In Vitro Antileishmanial Activity of 4- Aminoquinoline Derivatives Hybridized to Isoniazid or Sulfa or Hydrazine Groups

, 14(5): 597 - 604

Roberta R. Soares, Luciana M. R. Antinarelli, Isabela de O. Souza, Isabela de O. Souza, Fernanda V. Lopes, Kézia K. G. Scopel, Elaine S. Coimbra, Adilson D. da Silva and Clarice Abramo


DOI: 10.2174/1570180813666160927113743



Research Article

Vitamin B12 Controlled Release with Crosslinked Poly (Acrylic Acid) and Poly (Methacrylic Acid) Based on Chitosan and Starch as pH Sensitive Hydrogels

, 14(5): 605 - 612

Massomeh Ghorbanloo and Somaieh Tarasi


DOI: 10.2174/1570180814666161118150532



Research Article

Quorum Sensing Inhibitor Activities of Celecoxib Derivatives in Pseudomonas aeruginosa

, 14(5): 613 - 618

Seyhan Ulusoy, Sevil Senkardes, Inci Coskun, Gulgun Bosgelmez-Tınaz, Laurent Soulere, Yves Queneau and S. Guniz Kucukguzel


DOI: 10.2174/1570180814666161121120719



Review Article

NF-κB Inhibitors in Head and Neck Cancer

, 14(5): 619 - 633

Siddavaram Nagini, Kranthi Kiran Kishore Tanagala and Indranil Chattopadhyay


DOI: 10.2174/1570180813666160926095002




Webmaster Contact: info@benthamscience.org
Copyright © 2018 Bentham Science