Contents

Letters in Drug Design & Discovery, Volume 14 - Number 4

Biography

Meet Our Editorial Board Member

, 14(4): 373

Romano Silvestri


DOI: 10.2174/157018081404170223193954




Research Article

Quinoline Derivatives as Novel Depigmenting and Antioxidant Agents

, 14(4): 374 - 379

Rebeca Mol Lima, Kauana Cristina de Souza, Jordana de Abreu Lazzarini, Isabela O. Souza, Adilson David da Silva and Nadia Rezende Barbosa Raposo


DOI: 10.2174/1570180813666160930164926




Research Article

Synthesis and Antioxidant Activity of Indole Derivatives Containing 4-Substituted Piperazine Moieties

, 14(4): 380 - 386

Tunca Gul Altuntas, Nilüfer Yılmaz, Tulay Coban and Sureyya Olgen


DOI: 10.2174/1570180813666161020165623




Research Article

In Silico Modeling for the Design of 2-substitted Benzimidazole Derivatives, and Prediction of Activity as Procaspase-3 Activators and Apoptosis Inducer

, 14(4): 387 - 397

Prajakta U. Kulkarni, Manjunath D. Ghate and Vivek K. Vyas


DOI: 10.2174/1570180813666160826114120




Research Article

Synthesis, Antiproliferative, and Antiangiogenic Activities of Benzochromene and Benzoquinoline Derivatives on Prostate Cancer in vitro

, 14(4): 398 - 413

Gricelda Mata, Juan Rodrigues, Neira Gamboa, Katiuska Charris, Gricela Lobo, Melina Monasterios, Milagros Avendano, Michael Lein, Klaus Jung, Claudia Abramjuk, Bianca Nitzsche, Michael Hopfner and Jaime Charris


DOI: 10.2174/1570180814666161118163844




Research Article

3D-QSAR and Molecular Docking Studies of Pyrazole Derivatives as Inhibitors of Enoyl Acyl Carrier Protein Reductase from Mycobacterium tuberculosis

, 14(4): 414 - 433

Sheshagiri R. Dixit, Shrinivas D. Joshi, V. H. Kulkarni and Tejraj M. Aminabhavi


DOI: 10.2174/1570180814666161107155459




Research Article

Synthesis, Molecular Docking and Pharmacological Study of Pyrimidothiadiazinones and its bis-derivatives

, 14(4): 434 - 443

Sobhi M. Gomha, Ikhlass M. Abbas, Mohamed A. A. Elneairy, Mahmoud M. Elaasser and Bazada K. A. Mabrouk


DOI: 10.2174/1570180813666160815125409




Research Article

Structure-Based Hybridization, Conventional and Microwave Irradiated Synthesis, Biological Evaluation and Molecular Docking Studies of New Compounds Derived from Thiomorpholin

, 14(4): 444 - 463

Serpil Demirci, Fatma Aksakal, Nesrin Colak, Serdar Ulker, Ahmet Demirbas and Neslihan Demirbas


DOI: 10.2174/1570180813666161024165613




Research Article

Improved Anti-inflammatory Activity and Potential Cytoprotective Properties of Tolfenamic Acid, Naproxen and Indomethacin Derivatives

, 14(4): 464 - 475

Panagiotis Theodosis-Nobelos, Theodora C. Politou, Chrysoula Athanasekou and Eleni A. Rekka


DOI: 10.2174/1570180813666160831143112




Research Article

Chronobiotic Hormone Melatonin: Comparative in vitro Release Studies from Matrix Tablets and Liposomal Formulations

, 14(4): 476 - 480

Androniki Zampakola, Angeliki Siamidi, Natassa Pippa, Costas Demetzos and Marilena Vlachou


DOI: 10.2174/1570180813666161006162246




Research Article

Caffeic Acid Phenethyl Ester Restores Adipocyte Gene Profile Expression Following Lipopolysaccharide Treatment

, 14(4): 481 - 487

Ignazio Barbagallo, Giovanni Li Volti, Valeria Sorrenti, Claudia Di Giacomo, Rosaria Acquaviva, Marco Raffaele, Fabio Galvano and Luca Vanella


DOI: 10.2174/1570180813666160901124707




Research Article

Pharmacokinetic Evaluation of Callistemon viminalis Derived Natural Compounds as Targeted Inhibitors Against δ -Opioid Receptor and Farnesyl Transferase

, 14(4): 488 - 499

Kamal Ahmad, Abdul Roouf Bhat and Fareeda Athar


DOI: 10.2174/1570180814666161214114322




Research Article

Sequential Therapy For Helicobacter pylori in Elderly Patients: Effectiveness, Safety and Predictors of Success

, 14(4): 500 - 505

Giuseppe Losurdo, Andrea Iannone, Floriana Giorgio, Michele Barone, Mariabeatrice Principi, Enzo Ierardi and Alfredo Di Leo


DOI: 10.2174/1570180813666160922113541




Webmaster Contact: info@benthamscience.org
Copyright © 2018 Bentham Science