Contents

Letters in Drug Design & Discovery, Volume 14 - Number 3

Biography

Meet Our Editor

, 14(3): 251

George Perry


DOI: 10.2174/157018081403170126205345




Research Article

Design, Synthesis and Evaluation of Novel Derivatives of Orotic Acid Amide as Potent Glucokinase Activators

, 14(3): 252 - 261

Leilei Zhang, Shengquan Hu, Lei Lei, Yuliang Zhang, Lijing Zhang, Hongrui Song, Zhufang Shen and Zhiqiang Feng


DOI: 10.2174/1570180813666161013150056





Research Article

Design, Synthesis and Insecticidal Activity of Diamides with Oxydibenzene or Diphenylamine Subunits

, 14(3): 262 - 269

Ye Liu, Xinfei Chen, Xiaoyong Xu, Jiagao Cheng, Xusheng Shao and Zhong Li


DOI: 10.2174/1570180813666161028113852





Research Article

3D-QSAR, Molecular Docking and Molecular Dynamics Studies of 2,4- Diarylaminopyrimidine Analogues (DAAP Analogues) as Potent ALK Inhibitors

, 14(3): 270 - 286

Fulong Wu, Qianqian Lv, Zhonghua Wang, Dandan Li, Peng Peng, Yan Yin, Siheng Cui and Fanhong Wu


DOI: 10.2174/1570180813666160930162831





Research Article

Pentoxifylline Alleviates Proteinuria in Fructose Model of Metabolic Syndrome

, 14(3): 287 - 292

Hany M. El-Bassossy, Basma G. Eid and Ahmed Azhar


DOI: 10.2174/1570180813666160920115514





Research Article

Design, Synthesis and Biological Evaluation of Novel Tetrahydroquinoline Based Propanehydrazides as Antitubercular Agents

, 14(3): 293 - 300

Subhash Chander, Penta Ashok, Bidart de Macedo Maira, Paul Cos, Davie Cappoen and Sankaranarayanan Murugesan


DOI: 10.2174/1570180813666160622094013





Research Article

Field Based 3D-QSAR Model of KATP Channel Activation by 4, 6 Di-substituted Benzopyran Derivatives

, 14(3): 301 - 305

Yaseen Gigani, Swati Gupta, Andrew Lynn and Kamlesh Asotra


DOI: 10.2174/1570180813666160810150801





Research Article

3D-QSAR Studies of Novel Cytotoxic Bufadienolides via CoMFA and CoMSIA Approaches

, 14(3): 306 - 313

Hui Lin, Shengrong Li, Shiyao Li, Kangjia Liu, Yushui Han, Jialiang Guo, Longxin Lin, Yiqun Chang, Gaokeng Xiao, Weimin Chen and Pinghua Sun


DOI: 10.2174/1570180813666160906150621





Research Article

Design, Synthesis and Antidepressant and Anticonvulsant Effect of 1-Alkoxy-1H-Benzo[d]-1,2,3-Triazole Derivatives

, 14(3): 314 - 322

Yu Sun, Qing-Hao Jin, Yan Han, Di Yu, Qiu-Ping Dai and Zhou-Jun Zheng


DOI: 10.2174/1570180813666160826113018





Research Article

Synthesis and Nematocidal Activity of Novel Pyrazole Carboxamide Derivatives Against Meloidogyne incognita

, 14(3): 323 - 329

Wen Zhao, Zhong-Hua Shen, Jia-Hua Xing, Tian-Ming Xu, Wei-Li Peng and Xing-Hai Liu


DOI: 10.2174/1570180813666160930164327





Research Article

Structural Studies of Aminopeptidase P from Plasmodium falciparum: A Novel Target Against Malaria

, 14(3): 330 - 338

Polaboina Snigdha, Pachineella Lakshmana Rao, Nagu Prakash Prabhu and Insaf Ahmed Qureshi


DOI: 10.2174/1570180813666160725113524





Research Article

Anti-biofilm and Antibacterial Effects of Novel Metal-coordinated Sulfamethoxazole Against Escherichia coli

, 14(3): 339 - 344

Caren Rigon Mizdal, Sílvio Terra Stefanello, Pauline Cordenonsi Bonez, Vanessa Albertina Agertt, Vanessa da Costa Flores, Grazielle Guidolin Rossi, Fallon dos Santos Siqueira, Lenice de Lourenco Marques and Marli Matiko Anraku de Campos


DOI: 10.2174/1570180813666160930101653





Research Article

Molecular Docking, Molecular Dynamics, and In Silico Prediction of the Toxic Potential of Primaquine Thiazolidinone Derivatives

, 14(3): 345 - 353

Erika Murce and Andre Silva Pimentel


DOI: 10.2174/1570180813666160804170730





Review Article

Novel Second Generation HIV Integrase Inhibitor-DOLUTEGRAVIR: An Emerging Weapon Against HIV

, 14(3): 354 - 371

Vivek Jain, Diksha Gupta, Ashutosh Pareek and Yashumati Ratan


DOI: 10.2174/1570180813666160909121751





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