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Letters in Drug Design & Discovery

Volume 18, 12 Issues, 2021
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

In the current pandemic scenario, publication process of all articles related to Coronavirus will be expedited, for timely publication of much needed research


Letters in Drug Design & Discovery, Volume 14 - Number 2

Research Article

In Vitro and In Vivo Investigations into the Carbene Gold Chloride and Thioglucoside Anticancer Drug Candidates NHC-AuCl and NHC-AuSR

, 14(2): 125 - 134

Wolfgang Walther, Oyinlola Dada, Cillian O’Beirne, Ingo Ott, Goar Sánchez-Sanz, Claudia Schmidt, Carsta Werner, Xiangming Zhu and Matthias Tacke

DOI: 10.2174/1570180813666160826100158

Research Article

Estrogen Catechols Detection as Biomarkers in Schistosomiasis Induced Cancer and Infertility

, 14(2): 135 - 138

Monica C. Botelho, Helena Alves and Joachim Richter

DOI: 10.2174/1570180813666160720165057

Research Article

Zinc Tetrafluoroborate Catalyzed Synthesis, Molecular Docking and Cytotoxicity of Pyrrolidinyl Aminophosphonates

, 14(2): 139 - 150

Sarva Santhisudha, Kandula Madhu Kumar Reddy, Yellapu Nanda Kumar, Ethiraj Selvarajan, Vaithiyalingam Mohanasrinivasan, Sandip Kumar Nayak and Cirandur Suresh Reddy

DOI: 10.2174/1570180813666160722123045

Research Article

Synthesis and Cytotoxicity of Amino-Pyrazole Derivatives with Preliminary SAR

, 14(2): 151 - 158

Chunqi Hu, Jianfeng Shen and Wenting Du

DOI: 10.2174/1570180813666160930162522

Research Article

Synthesis of Some New 1(2H)-Phthalazinone Derivatives and Evaluation of Their Acetylcholinesterase and Butyrylcholinesterase Inhibitory Activities

, 14(2): 159 - 166

Burcu Kılıç, Hayrettin Ozan Gülcan, Mertcan Yalçın, Fatma Aksakal, Anatoli Dimoglo, Mustafa Fethi Şahin and Deniz Songül Doğruer

DOI: 10.2174/1570180813666160819124611

Research Article

Discovery of 6-benzamide Containing 4-phenylquinazoline Derivatives as Novel PI3Kδ Inhibitors

, 14(2): 167 - 174

Minhang Xin, Yuan-Yuan Hei, Hao Zhang, Xiao-Xiao Xie, Shuai Mao, Sai-Jie Zuo and San-Qi Zhang

DOI: 10.2174/1570180813666160720160523

Research Article

Identification of Thiazoloquin(az)olin(on)es Derivatives as CD38 Inhibitors Through 3D-QSAR and Molecular Docking Simulations

, 14(2): 175 - 185

Xiaodong Gao and Yujie Ren

DOI: 10.2174/1570180813666160919121104

Research Article

Synthesis of New Benzofuran-Pyrazole Hybrids as Potential Antibiofilm Agents

, 14(2): 186 - 194

Gejjalagere S. Lingaraju, Somashekaraiah Rakesh, Koravangala S.V. Kumar, Kanchepalli P. Rao, Marikunte Y. Sreenivasa and Maralinganadoddi P. Sadashiva

DOI: 10.2174/1570180813666160923170414

Research Article

Synthesis and Herbicidal Activity of Some Novel Pyrazole Derivatives

, 14(2): 195 - 200

Hai-Qin He, Xing-Hai Lie, Jian-Quan Weng and Cheng-Xia Tan

DOI: 10.2174/1570180813666160805150148

Research Article

Synthesis and Antioxidant Evaluation of Some Novel Benzimidazole Derivatives Containing a Triazole Nucleus

, 14(2): 201 - 208

Fatih Yılmaz, Emre Menteşe and Nimet Baltaş

DOI: 10.2174/1570180813666160609082633

Research Article

Synthesis and Evaluation of Morpholinoethyl Ester Conjugate of N-acetylcysteine in Ovalbumin-induced Airway Hyperresponsiveness in Sprague Dawley Rats

, 14(2): 209 - 215

Neha V. Bhilare and Suneela S. Dhaneshwar

DOI: 10.2174/1570180813666160804152912

Research Article

Biologically Potent Pyrazoline Derivatives from Versatile (2)-1-(4- Chlorophenyl)-3-[4-(propan-2-yl)phenyl]prop-2-en-1-one

, 14(2): 216 - 227

Vinutha V. Salian, Badiadka Narayana, Balladka K. Sarojini, Enumadisetty S. Sindhupriya, Leelavathi N. Madhu and Shama Rao

DOI: 10.2174/1570180813666160519151723

Research Article

Design, Synthesis and Bioactivity of Phenoxy Carboxylate(amide) Derivatives Containing 4,6-Dimethoxypyrimidine

, 14(2): 228 - 232

Zhiqiang Huang, Chenpeng Feng, Jun Tong, Qiang Bian and Yu Zhao

DOI: 10.2174/1570180813666160818153617

Research Article

The Synthesis of (Iodobenzyl)oxybenzaldehydes, Useful Intermediates for Biologically Active Targets

, 14(2): 233 - 239

Hedvig Bölcskei, Andrea Német-Hanzelik, István Greiner, Zsófia Dubrovay, Viktor Háda and György Keglevich

DOI: 10.2174/1570180813666160804142245

Review Article

Anti-inflammatory Potential of Alkaloids as a Promising Therapeutic Modality

, 14(2): 240 - 249

Marya and Haroon Khan

DOI: 10.2174/1570180813666160712224752


K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 1.05


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