Contents

Letters in Drug Design & Discovery, Volume 14 - Number 2

Research Article

In Vitro and In Vivo Investigations into the Carbene Gold Chloride and Thioglucoside Anticancer Drug Candidates NHC-AuCl and NHC-AuSR

, 14(2): 125 - 134

Wolfgang Walther, Oyinlola Dada, Cillian O’Beirne, Ingo Ott, Goar Sánchez-Sanz, Claudia Schmidt, Carsta Werner, Xiangming Zhu and Matthias Tacke


DOI: 10.2174/1570180813666160826100158



Research Article

Estrogen Catechols Detection as Biomarkers in Schistosomiasis Induced Cancer and Infertility

, 14(2): 135 - 138

Monica C. Botelho, Helena Alves and Joachim Richter


DOI: 10.2174/1570180813666160720165057



Research Article

Zinc Tetrafluoroborate Catalyzed Synthesis, Molecular Docking and Cytotoxicity of Pyrrolidinyl Aminophosphonates

, 14(2): 139 - 150

Sarva Santhisudha, Kandula Madhu Kumar Reddy, Yellapu Nanda Kumar, Ethiraj Selvarajan, Vaithiyalingam Mohanasrinivasan, Sandip Kumar Nayak and Cirandur Suresh Reddy


DOI: 10.2174/1570180813666160722123045



Research Article

Synthesis and Cytotoxicity of Amino-Pyrazole Derivatives with Preliminary SAR

, 14(2): 151 - 158

Chunqi Hu, Jianfeng Shen and Wenting Du


DOI: 10.2174/1570180813666160930162522



Research Article

Synthesis of Some New 1(2H)-Phthalazinone Derivatives and Evaluation of Their Acetylcholinesterase and Butyrylcholinesterase Inhibitory Activities

, 14(2): 159 - 166

Burcu Kılıç, Hayrettin Ozan Gülcan, Mertcan Yalçın, Fatma Aksakal, Anatoli Dimoglo, Mustafa Fethi Şahin and Deniz Songül Doğruer


DOI: 10.2174/1570180813666160819124611



Research Article

Discovery of 6-benzamide Containing 4-phenylquinazoline Derivatives as Novel PI3Kδ Inhibitors

, 14(2): 167 - 174

Minhang Xin, Yuan-Yuan Hei, Hao Zhang, Xiao-Xiao Xie, Shuai Mao, Sai-Jie Zuo and San-Qi Zhang


DOI: 10.2174/1570180813666160720160523



Research Article

Identification of Thiazoloquin(az)olin(on)es Derivatives as CD38 Inhibitors Through 3D-QSAR and Molecular Docking Simulations

, 14(2): 175 - 185

Xiaodong Gao and Yujie Ren


DOI: 10.2174/1570180813666160919121104



Research Article

Synthesis of New Benzofuran-Pyrazole Hybrids as Potential Antibiofilm Agents

, 14(2): 186 - 194

Gejjalagere S. Lingaraju, Somashekaraiah Rakesh, Koravangala S.V. Kumar, Kanchepalli P. Rao, Marikunte Y. Sreenivasa and Maralinganadoddi P. Sadashiva


DOI: 10.2174/1570180813666160923170414



Research Article

Synthesis and Herbicidal Activity of Some Novel Pyrazole Derivatives

, 14(2): 195 - 200

Hai-Qin He, Xing-Hai Lie, Jian-Quan Weng and Cheng-Xia Tan


DOI: 10.2174/1570180813666160805150148



Research Article

Synthesis and Antioxidant Evaluation of Some Novel Benzimidazole Derivatives Containing a Triazole Nucleus

, 14(2): 201 - 208

Fatih Yılmaz, Emre Menteşe and Nimet Baltaş


DOI: 10.2174/1570180813666160609082633



Research Article

Synthesis and Evaluation of Morpholinoethyl Ester Conjugate of N-acetylcysteine in Ovalbumin-induced Airway Hyperresponsiveness in Sprague Dawley Rats

, 14(2): 209 - 215

Neha V. Bhilare and Suneela S. Dhaneshwar


DOI: 10.2174/1570180813666160804152912



Research Article

Biologically Potent Pyrazoline Derivatives from Versatile (2)-1-(4- Chlorophenyl)-3-[4-(propan-2-yl)phenyl]prop-2-en-1-one

, 14(2): 216 - 227

Vinutha V. Salian, Badiadka Narayana, Balladka K. Sarojini, Enumadisetty S. Sindhupriya, Leelavathi N. Madhu and Shama Rao


DOI: 10.2174/1570180813666160519151723



Research Article

Design, Synthesis and Bioactivity of Phenoxy Carboxylate(amide) Derivatives Containing 4,6-Dimethoxypyrimidine

, 14(2): 228 - 232

Zhiqiang Huang, Chenpeng Feng, Jun Tong, Qiang Bian and Yu Zhao


DOI: 10.2174/1570180813666160818153617



Research Article

The Synthesis of (Iodobenzyl)oxybenzaldehydes, Useful Intermediates for Biologically Active Targets

, 14(2): 233 - 239

Hedvig Bölcskei, Andrea Német-Hanzelik, István Greiner, Zsófia Dubrovay, Viktor Háda and György Keglevich


DOI: 10.2174/1570180813666160804142245



Review Article

Anti-inflammatory Potential of Alkaloids as a Promising Therapeutic Modality

, 14(2): 240 - 249

Marya and Haroon Khan


DOI: 10.2174/1570180813666160712224752




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