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Contents

Letters in Drug Design & Discovery, Volume 14 - Number 12


Research Article

QSAR Modeling of Aminopeptidase N/CD13 (APN) Inhibitory Activity of some Leucine Ureido Derivatives by GA-MLR and SW-MLR Methods

, 14(12): 1348 - 1357

Naser Faraji, Tannaz Zebardast, Afshin Zarghi* and Zahra Hajimahdi*


DOI: 10.2174/1570180814666170529084557



Research Article

A Study on Identification of Nutraceutical Value of New Imidazolone Schiff Base Analogues

, 14(12): 1358 - 1370

Subbulakshmi N. Karanth, Badiadka Narayana*, Balladka K. Sarojini, Saleemulla Khan and Shashidhara S. Kenkere


DOI: 10.2174/1570180814666170412120555



Research Article

An Improved Preparation of (R)-3-Aminobutanol, a Key Intermediate for the Synthesis of Dolutegravir Sodium

, 14(12): 1371 - 1375

Y. Srinivasa Rao, B. Hari Babu*, I. Aminual, D. Nageshwar and P.V.V. Satyanarayana


DOI: 10.2174/1570180814666170602083756



Research Article

Design and Synthesis of Amino Acid Tethered Thiazolones to Screen for Hepatitis C NS5B Polymerase Inhibitors

, 14(12): 1376 - 1381

Yili Ding*, Kenneth L. Smith and Chamakura V.N.S. Varaprasad


DOI: 10.2174/1570180814666170505121156



Research Article

Design, Synthesis and Antiproliferative Activities Evaluation of Thiazolopyrimidines Derivatives through Biginelli Reaction

, 14(12): 1382 - 1390

Pengju Zhu, Huansheng Fu and Hao Fang*


DOI: 10.2174/1570180814666170512123132



Research Article

CETP Inhibitory Activity of Chlorobenzyl Benzamides: QPLD Docking, Pharmacophore Mapping and Synthesis

, 14(12): 1391 - 1400

Reema Abu Khalaf*, Hamada Abd El-Aziz, Dima Sabbah, Ghadeer Albadawi and Ghassan Abu Sheikha


DOI: 10.2174/1570180814666170412122304



Research Article

Preparation and Characterization of Mixed Polymeric Micelles as a Versatile Strategy for Meloxicam Oral Administration

, 14(12): 1401 - 1408

Claudia Amaral, Mariana Magalhaes, Celia Cabral, Francisco Veiga and Ana Figueiras*


DOI: 10.2174/1570180814666170505120728



Research Article


Research Article

A SAR Study: Evaluation of Bromo Derivatives of 8-Substituted Quinolines as Novel Anticancer Agents

, 14(12): 1415 - 1424

Salih Okten*, Osman Cakmak, Saban Tekin and Tugba Kul Koprulu


DOI: 10.2174/1570180814666170504150050



Research Article

Synthesis and Anti-Oxidant Evaluation of Some Novel Sulfa Drugs

, 14(12): 1425 - 1432

Moustafa A. Gouda* and Belal H.M. Hussein


DOI: 10.2174/1570180814666170607144811



Research Article

Spices Chemoconstituents as Persuasive Inhibitor of S. typhimurium Virulent Protein L-asparaginase

, 14(12): 1433 - 1454

Archana Vimal and Awanish Kumar*


DOI: 10.2174/1570180814666170602080822



Research Article

In Silico Prioritization, Synthesis and In Vitro Evaluation of Tembamide Analogs for Anti-HIV Activity

, 14(12): 1455 - 1464

Shiv Gupta, Sanjay Kumar, Nisha Jariwala, Deepali Bhadane, Kamlesh Kumar Bhutani, Smita Kulkarni* and Inder Pal Singh*


DOI: 10.2174/1570180814666170419115526



Review Article

Neurokinin-1 Receptor Antagonists in Lung Cancer Therapy

, 14(12): 1465 - 1476

Miguel Munoz*, Marisa Rosso and Rafael Covenas


DOI: 10.2174/1570180814666170327163854





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