Contents

Letters in Drug Design & Discovery, Volume 14 - Number 12

Biography

Meet Our Editorial Board Member

, 14(12): 1347

Enrico Garattini


DOI: 10.2174/157018081412171031113907




Research Article

QSAR Modeling of Aminopeptidase N/CD13 (APN) Inhibitory Activity of some Leucine Ureido Derivatives by GA-MLR and SW-MLR Methods

, 14(12): 1348 - 1357

Naser Faraji, Tannaz Zebardast, Afshin Zarghi and Zahra Hajimahdi


DOI: 10.2174/1570180814666170529084557





Research Article

A Study on Identification of Nutraceutical Value of New Imidazolone Schiff Base Analogues

, 14(12): 1358 - 1370

Subbulakshmi N. Karanth, Badiadka Narayana, Balladka K. Sarojini, Saleemulla Khan and Shashidhara S. Kenkere


DOI: 10.2174/1570180814666170412120555





Research Article

An Improved Preparation of (R)-3-Aminobutanol, a Key Intermediate for the Synthesis of Dolutegravir Sodium

, 14(12): 1371 - 1375

Y. Srinivasa Rao, B. Hari Babu, I. Aminual, D. Nageshwar and P.V.V. Satyanarayana


DOI: 10.2174/1570180814666170602083756





Research Article

Design and Synthesis of Amino Acid Tethered Thiazolones to Screen for Hepatitis C NS5B Polymerase Inhibitors

, 14(12): 1376 - 1381

Yili Ding, Kenneth L. Smith and Chamakura V.N.S. Varaprasad


DOI: 10.2174/1570180814666170505121156





Research Article

Design, Synthesis and Antiproliferative Activities Evaluation of Thiazolopyrimidines Derivatives through Biginelli Reaction

, 14(12): 1382 - 1390

Pengju Zhu, Huansheng Fu and Hao Fang


DOI: 10.2174/1570180814666170512123132





Research Article

CETP Inhibitory Activity of Chlorobenzyl Benzamides: QPLD Docking, Pharmacophore Mapping and Synthesis

, 14(12): 1391 - 1400

Reema Abu Khalaf, Hamada Abd El-Aziz, Dima Sabbah, Ghadeer Albadawi and Ghassan Abu Sheikha


DOI: 10.2174/1570180814666170412122304





Research Article

Preparation and Characterization of Mixed Polymeric Micelles as a Versatile Strategy for Meloxicam Oral Administration

, 14(12): 1401 - 1408

Claudia Amaral, Mariana Magalhaes, Celia Cabral, Francisco Veiga and Ana Figueiras


DOI: 10.2174/1570180814666170505120728





Research Article

The Impact of 5-Substituted Uracil Derivatives on Immortalized Embryo Lung Cells

, 14(12): 1409 - 1414

Natalia N. Kabal'nova, Stanislav A. Grabovskiy, Nadezhda M. Andriayshina, Vladislav I. Egorov, Lenar R. Valiullin, Alexey A. Nabatov, Ivan S. Raginov and Yurii I. Murinov


DOI: 10.2174/1570180814666170502171640





Research Article

A SAR Study: Evaluation of Bromo Derivatives of 8-Substituted Quinolines as Novel Anticancer Agents

, 14(12): 1415 - 1424

Salih Okten, Osman Cakmak, Saban Tekin and Tugba Kul Koprulu


DOI: 10.2174/1570180814666170504150050





Research Article

Synthesis and Anti-Oxidant Evaluation of Some Novel Sulfa Drugs

, 14(12): 1425 - 1432

Moustafa A. Gouda and Belal H.M. Hussein


DOI: 10.2174/1570180814666170607144811





Research Article

Spices Chemoconstituents as Persuasive Inhibitor of S. typhimurium Virulent Protein L-asparaginase

, 14(12): 1433 - 1454

Archana Vimal and Awanish Kumar


DOI: 10.2174/1570180814666170602080822





Research Article

In Silico Prioritization, Synthesis and In Vitro Evaluation of Tembamide Analogs for Anti-HIV Activity

, 14(12): 1455 - 1464

Shiv Gupta, Sanjay Kumar, Nisha Jariwala, Deepali Bhadane, Kamlesh Kumar Bhutani, Smita Kulkarni and Inder Pal Singh


DOI: 10.2174/1570180814666170419115526





Review Article

Neurokinin-1 Receptor Antagonists in Lung Cancer Therapy

, 14(12): 1465 - 1476

Miguel Munoz, Marisa Rosso and Rafael Covenas


DOI: 10.2174/1570180814666170327163854





Acknowledgement

Acknowledgements to Reviewers

, 14(12): 1477


DOI: 10.2174/157018081412171031150240




Webmaster Contact: info@benthamscience.org
Copyright © 2018 Bentham Science