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Letters in Drug Design & Discovery

Volume 18, 12 Issues, 2021
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

In the current pandemic scenario, publication process of all articles related to Coronavirus will be expedited, for timely publication of much needed research


Letters in Drug Design & Discovery, Volume 14 - Number 11

Research Article

2D, 3D, G-QSAR and Docking Studies of Thiazolyl-pyrazoline Analogues as Potent (Epidermal Growth Factor Receptor-tyrosine Kinase) EGFR-TK Inhibitors

, 14(11): 1228 - 1238

Ghodgaonkar Sunayana, Bhandari Shashikant and Waghulde Sandeep

DOI: 10.2174/1570180814666170518171236

Research Article

Synthesis, Docking and Evaluation of Phenylacetic Acid and Trifluoro-methylphenyl Substituted Benzamide Derivatives as Potential PPARδ Agonists

, 14(11): 1239 - 1251

Ajmer Singh Grewal, Viney Lather, Deepti Pandita and Garima Bhayana

DOI: 10.2174/1570180814666170327164443

Research Article

Molecular Docking Studies of Novel Thiosemicarbazone-based Indoles as Potential PI3Kα Inhibitors

, 14(11): 1252 - 1258

Dima A. Sabbah and Kamal Sweidan

DOI: 10.2174/1570180814666170619112647

Research Article

Synthesis and Structure-activity Relationships of Chalcone Derivatives as Inhibitors of Ovarian Cancer Cell Growth

, 14(11): 1259 - 1266

Zachary D. Tucker, Francis J. Barrios and Amanda J. Krzysiak

DOI: 10.2174/1570180814666170505120258

Research Article

Molecular Docking and In Silico ADMET Study Reveals Flavonoids as a Potential Inhibitor of Aromatase

, 14(11): 1267 - 1276

Umang Shah, Samir Patel, Mehul Patel and Jagat Upadhayay

DOI: 10.2174/1570180814666170327161908

Research Article

Molecular Simulation and Activity Studies of Oxametacin as an HDAC Inhibitor

, 14(11): 1277 - 1282

Fanbo Jing, Lei Zhang, Yepeng Luan and Jiang Bian

DOI: 10.2174/1570180814666170505123930

Research Article

Molecular Docking Simulations as a Prominent Tool to Envisage the Preformulation Perspectives of Oral Hypoglycaemic Agents with β-cyclodextrin

, 14(11): 1283 - 1290

Sant K. Verma and Akhlesh K. Jain

DOI: 10.2174/1570180814666170420125907

Research Article

Computational Studies of N-substituted Quinolinonyl Diketo Acid Derivatives as HIV Integrase Strand Transfer Inhibitors using 3D-QSAR, Pharmacophore Modeling and Molecular Docking

, 14(11): 1291 - 1302

Yuming Luo, Yujie Ren and Xiaodong Gao

DOI: 10.2174/1570180814666170605120017

Research Article

The Antiviral Effects of Harmine Against BoHV-1 Infection In Vitro

, 14(11): 1303 - 1307

Xinyi Jiang, Jie Zou, Yuncheng Zhuang, Weifeng Yuan, Liqian Zhu and Guoqiang Zhu

DOI: 10.2174/1570180814666170425155554

Research Article

New Cyclohexylamine-dithiocarbamate Derivatives as Potential Anti-microbial Agents

, 14(11): 1308 - 1315

Leyla Yurttas, Betul Kaya , Meral Yilmaz Cankilic and Serkan Levent

DOI: 10.2174/1570180814666170412121402

Research Article

Synthesis and Antimicrobial Activity of Some Novel Substituted 3-(Thiophen-2-yl)pyrazole-based Heterocycles

, 14(11): 1316 - 1323

Bakr F. Abdel-Wahab, Abdelbasset A. Farahat, Ghada E. A. Awad and Gamal A. El-Hiti

DOI: 10.2174/1570180814666170327162447

Research Article

Novel Thiazole Carboxylic Acid Derivatives Possessing a “Zinc Binding Feature” as Potential Human Glyoxalase-I Inhibitors

, 14(11): 1324 - 1334

DOI: 10.2174/1570180814666170306120954

Research Article

Synthesis and Antiproliferative Activity of 3-aza Steroids as 5α-reductase Inhibitors

, 14(11): 1335 - 1346

Milanpreet Kaur, Richa Dhingra, T. R. Bhardwaj and Neelima Dhingra

DOI: 10.2174/1570180814666170505122503


K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 1.05


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