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Letters in Drug Design & Discovery

Volume 18, 12 Issues, 2021
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

In the current pandemic scenario, publication process of all articles related to Coronavirus will be expedited, for timely publication of much needed research


Letters in Drug Design & Discovery, Volume 14 - Number 1

Research Article

Proteochemometrics for the Prediction of Binding to the MHC Proteins

, 14(1): 2 - 9

Ventsislav Yordanov, Ivan Dimitrov and Irini Doytchinova

DOI: 10.2174/1570180813666160630122341

Research Article

Quantitative Structure-Activity Relationship and Docking Studies on a Series of Oxadiazole and Triazole Substituted Naphthyridines as HIV-1 Integrase Inhibitors

, 14(1): 10 - 27

Basheerulla Shaik, Vijay Agrawal, Satya P. Gupta and Urvana Menon

DOI: 10.2174/1570180813666160610090525

Research Article

Relationships Between the Structural Properties of Flavonoids and their Inhibitory Activities Against Matrix Metallopeptidase 9

, 14(1): 28 - 35

Soon Young Shin, Hyeryoung Jung, Yearam Jung, Beom Soo Kim, Young Han Lee and Yoongho Lim

DOI: 10.2174/1570180813666160919161434

Research Article

3D-QSAR Modeling and Molecular Docking Study on Small Molecule Stat3 Inhibitors, Src Homology 2 Domain Binders

, 14(1): 36 - 49

Jing Li Wang, Li Ping Cheng, Yang Ping Quan, Zhen Wang, Fan Hong Wu and Wei Deng

DOI: 10.2174/1570180813666160801152618

Research Article

Synthesis and Biological Activity of Quinoxalone Derivatives as BRD4 Bromodomain Inhibitors

, 14(1): 50 - 57

Bin Xu, Lei-Lei Zhao, Yi-Fei Yang, Jian Zhang, Ling-Yun Yang, Bing Zhang, Li Han, Hui-Bin Zhang and Jin-Pei Zhou

DOI: 10.2174/1570180813666160715160857

Research Article

1,2,3-Triazole-Isoxazole Based Acetylcholinesterase Inhibitors: Synthesis, Biological Evaluation and Docking Study

, 14(1): 58 - 65

Zahra Najafi, Mohammad Mahdavi, Mina Saeedi, Reyhaneh Sabourian, Mahnaz Khanavi, Maliheh Safavi, Maliheh Barazandeh Tehrani, Abbas Shafiee, Alireza Foroumadi and Tahmineh Akbarzadeh

DOI: 10.2174/1570180813666160628085515

Research Article

Computational Identification of Inhibitors Against DPP-IV for Checking Type-2 Diabetes

, 14(1): 66 - 73

Sarvesh Kumar Gupta, Kamal Kumar Chaudhary, Utkarsh Raj and Nidhi Mishra

DOI: 10.2174/1570180813666160720121718

Research Article

Combined 3D-QSAR, Pharmacophore and Docking Studies on Benzenesulfonamide Derivatives as Potent 12-Lipoxygenase Inhibitors

, 14(1): 74 - 82

Chunhong An, Mao Shu, Xiaoli Zai, Beina Zhang, Jing Li, Zichao Chang, Yong Hu and Zhihua Lin

DOI: 10.2174/1570180813666160930100456

Research Article

QSAR and Molecular Docking Studies on a Series of Cinnamic Acid Analogues as Epidermal Growth Factor Receptor (EGFR) Inhibitors

, 14(1): 83 - 95

Basheerulla Shaik, Omar Deeb, Vijay K. Agrawal and Satya P. Gupta

DOI: 10.2174/1570180813999160721160833

Research Article

Synthesis and Biological Evaluation of a Novel Apogossypolone Derivative

, 14(1): 96 - 101

Yonghua Zhan, Xu Cao, Yingchao Li, Xueli Chen and Xiaofeng Huang

DOI: 10.2174/1570180813666160722115855

Research Article

Novel Artemisinin-Derived Dimers: Synthesis and Evaluation of Anti-cancer Activities

, 14(1): 102 - 111

Vu Tuan Kien, Le Huy Binh, Phan Hai Phong, Doan Thi Hien, Nguyen Thi Thuy My, Nguyen Hai Nam, Do Thi Thao, Michael Baltas and Tran Khac Vua

DOI: 10.2174/1570180813666160810155354

Research Article

Molecular Mechanisms and Potential Treatment Targets for Ovarian Cancer by Analyzing Transcriptional Regulatory Network

, 14(1): 112 - 118

Fei Wu, Xinrui Liu, Yujie Sui, Tianmin Xu and Manhua Cui

DOI: 10.2174/1570180813666160920122412

Research Article

Antileishmanial Activity of Labdane Diterpenes Isolated from Alpinia nigra Seeds

, 14(1): 119 - 124

Sudipta Ghosh, Rajesh Kumar Singh, Vikash Kumar Dubey and Latha Rangan

DOI: 10.2174/1570180813666160725100300


K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 1.05

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