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Letters in Drug Design & Discovery

Volume 18, 12 Issues, 2021
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

In the current pandemic scenario, publication process of all articles related to Coronavirus will be expedited, for timely publication of much needed research


Letters in Drug Design & Discovery, Volume 13 - Number 10

Research Article

β-Galactosidase – Excipients Interaction by Docking Simulation Studies

, 13(10): 993 - 998

Larissa L. Rodrigues, Alexandre C. Bertoli, Ihosvany Camps, Marcello G. Trevisan and Jerusa S. Garcia

DOI: 10.2174/1570180813666160628075149

Research Article

Analysis of the Applicability and Use of Lipinski`s Rule for Central Nervous System Drugs

, 13(10): 999 - 1006

Thais B. Fernandes, Mariana C. F. Segretti, Michelle C. Polli and Roberto Parise-Filho

DOI: 10.2174/1570180813666160622092839

Research Article

Principles of an Adenovirus-Based Assay for Candidate Compounds with Broad Spectrum of Anti-Neoplastic Activities

, 13(10): 1007 - 1011

Mikhail V. Shepelev, Elena V. Korobko and Igor V. Korobko

DOI: 10.2174/1570180813666160422162612

Research Article

Structure-based Virtual Screening to Get New Scaffold Inhibitors of the Ser/Thr Protein Kinase PknB from Mycobacterium tuberculosis

, 13(10): 1012 - 1018

Antonio Coluccia, Giuseppe La Regina, Nathalie Barilone, María-Natalia Lisa, Andrea Brancale, Gwenaëlle André-Leroux, Pedro M. Alzari and Romano Silvestri

DOI: 10.2174/1570180813666160801162204

Research Article

Synthesis and Antiviral Activity of 2-aryl-4H-chromen-4-one Derivatives Against Chikungunya Virus

, 13(10): 1019 - 1024

Vishnu N. Badavath, Surender S. Jadav, Boris Pastorino, Xavier de Lamballerie, Barij N. Sinha and Venkatesan Jayaprakash

DOI: 10.2174/1570180813666160711163349

Research Article

Novel Dual Inhibitors of Secretory Phospholipase A2 and Sphingomyelin Synthase: Design, Synthesis and Evaluation

, 13(10): 1025 - 1032

Haojun Gong, Lu Zhou, Deyong Ye, Xing Gao, Yali Li, Xiangyu Qi and Yong Chu

DOI: 10.2174/1570180813666160805155116

Research Article

Binding Free Energy-Based Footprint Pharmacophore Model to Enhance Virtual Screening and Drug Discovery: A Case on Glycosidases as Anti-influenza Drug Targets

, 13(10): 1033 - 1046

Ndumiso N. Mhlongo and Mahmoud E. S. Soliman

DOI: 10.2174/1570180813666160714162534

Research Article

Exploring the QSAR Analysis of imidazole-4, 5- and pyrazine-2,3- Dicarboxamides Derivatives Using Online Available Resources

, 13(10): 1047 - 1054

Arpit K. Gupta, Ravi Raushan, Jagadish Singh and Partha P. Roy

DOI: 10.2174/1570180813666160714144725

Research Article

Topomer CoMFA 3D-QSAR and Docking Studies of Pyrimidine Inhibitors of Pneumocystis Carinii Dihydrofolate Reductase

, 13(10): 1055 - 1062

Jianbo Tong, Pei Zhan, Tuanli Yao, Lanbing Ma and Min Bai

DOI: 10.2174/1570180813666160324154549

Research Article

Synthesis and Antimicrobial Evaluation of Aminoguanidine and 3-amino- 1,2,4-triazole Derivatives as Potential Antibacterial Agents

, 13(10): 1063 - 1075

Tian-Yi Zhang, Chao Li, Ya-Ru Li, Xiao-Zhen Li, Liang-Peng Sun, Chang-Ji Zheng and Hu-Ri Piao

DOI: 10.2174/1570180813666160819151239

Research Article

Microwave Assisted Synthesis and Antimicrobial Activity Evaluation of New Heterofunctionalized Norfloxacine Derivatives

, 13(10): 1076 - 1090

Meltem Mentese, Serpil Demirci, Serap B. Ozdemir, Ahmet Demirbas, Serdar Ulker and Neslihan Demirbas

DOI: 10.2174/1570180813666160712222922

Research Article

Facile Synthesis and Nitric Oxide Inhibitory Activity of Aurones, Rugaurone A, Gramflavonoid A and Their Derivatives

, 13(10): 1091 - 1098

Kongara Damodar, Jin-Kyung Kim and Jong-Gab Jun

DOI: 10.2174/1570180813666160824124224

Research Article

Preparation of Edible Zein Hybrid Particles and Its Controlled Release Behaviors

, 13(10): 1099 - 1103

Siyao Lv, Jie Liu, Fei Pei, Yufeng He and Rong-Min Wang

DOI: 10.2174/1570180813666160720122349


K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 1.05

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