Contents

Letters in Drug Design & Discovery, Volume 13 - Number 10

Research Article

β-Galactosidase – Excipients Interaction by Docking Simulation Studies

, 13(10): 993 - 998

Larissa L. Rodrigues, Alexandre C. Bertoli, Ihosvany Camps, Marcello G. Trevisan and Jerusa S. Garcia


DOI: 10.2174/1570180813666160628075149



Research Article

Analysis of the Applicability and Use of Lipinski`s Rule for Central Nervous System Drugs

, 13(10): 999 - 1006

Thais B. Fernandes, Mariana C. F. Segretti, Michelle C. Polli and Roberto Parise-Filho


DOI: 10.2174/1570180813666160622092839



Research Article

Principles of an Adenovirus-Based Assay for Candidate Compounds with Broad Spectrum of Anti-Neoplastic Activities

, 13(10): 1007 - 1011

Mikhail V. Shepelev, Elena V. Korobko and Igor V. Korobko


DOI: 10.2174/1570180813666160422162612



Research Article

Structure-based Virtual Screening to Get New Scaffold Inhibitors of the Ser/Thr Protein Kinase PknB from Mycobacterium tuberculosis

, 13(10): 1012 - 1018

Antonio Coluccia, Giuseppe La Regina, Nathalie Barilone, María-Natalia Lisa, Andrea Brancale, Gwenaëlle André-Leroux, Pedro M. Alzari and Romano Silvestri


DOI: 10.2174/1570180813666160801162204



Research Article

Synthesis and Antiviral Activity of 2-aryl-4H-chromen-4-one Derivatives Against Chikungunya Virus

, 13(10): 1019 - 1024

Vishnu N. Badavath, Surender S. Jadav, Boris Pastorino, Xavier de Lamballerie, Barij N. Sinha and Venkatesan Jayaprakash


DOI: 10.2174/1570180813666160711163349



Research Article

Novel Dual Inhibitors of Secretory Phospholipase A2 and Sphingomyelin Synthase: Design, Synthesis and Evaluation

, 13(10): 1025 - 1032

Haojun Gong, Lu Zhou, Deyong Ye, Xing Gao, Yali Li, Xiangyu Qi and Yong Chu


DOI: 10.2174/1570180813666160805155116



Research Article

Binding Free Energy-Based Footprint Pharmacophore Model to Enhance Virtual Screening and Drug Discovery: A Case on Glycosidases as Anti-influenza Drug Targets

, 13(10): 1033 - 1046

Ndumiso N. Mhlongo and Mahmoud E. S. Soliman


DOI: 10.2174/1570180813666160714162534



Research Article

Exploring the QSAR Analysis of imidazole-4, 5- and pyrazine-2,3- Dicarboxamides Derivatives Using Online Available Resources

, 13(10): 1047 - 1054

Arpit K. Gupta, Ravi Raushan, Jagadish Singh and Partha P. Roy


DOI: 10.2174/1570180813666160714144725



Research Article

Topomer CoMFA 3D-QSAR and Docking Studies of Pyrimidine Inhibitors of Pneumocystis Carinii Dihydrofolate Reductase

, 13(10): 1055 - 1062

Jianbo Tong, Pei Zhan, Tuanli Yao, Lanbing Ma and Min Bai


DOI: 10.2174/1570180813666160324154549



Research Article

Synthesis and Antimicrobial Evaluation of Aminoguanidine and 3-amino- 1,2,4-triazole Derivatives as Potential Antibacterial Agents

, 13(10): 1063 - 1075

Tian-Yi Zhang, Chao Li, Ya-Ru Li, Xiao-Zhen Li, Liang-Peng Sun, Chang-Ji Zheng and Hu-Ri Piao


DOI: 10.2174/1570180813666160819151239



Research Article

Microwave Assisted Synthesis and Antimicrobial Activity Evaluation of New Heterofunctionalized Norfloxacine Derivatives

, 13(10): 1076 - 1090

Meltem Mentese, Serpil Demirci, Serap B. Ozdemir, Ahmet Demirbas, Serdar Ulker and Neslihan Demirbas


DOI: 10.2174/1570180813666160712222922



Research Article

Facile Synthesis and Nitric Oxide Inhibitory Activity of Aurones, Rugaurone A, Gramflavonoid A and Their Derivatives

, 13(10): 1091 - 1098

Kongara Damodar, Jin-Kyung Kim and Jong-Gab Jun


DOI: 10.2174/1570180813666160824124224



Research Article

Preparation of Edible Zein Hybrid Particles and Its Controlled Release Behaviors

, 13(10): 1099 - 1103

Siyao Lv, Jie Liu, Fei Pei, Yufeng He and Rong-Min Wang


DOI: 10.2174/1570180813666160720122349



Acknowledgement



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