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Letters in Drug Design & Discovery

Volume 17, 12 Issues, 2020
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

In the current pandemic scenario, publication process of all articles related to Coronavirus will be expedited, for timely publication of much needed research

Contents

Letters in Drug Design & Discovery, Volume 13 - Number 1



Evaluation of Serine Protease Inhibitors as Potent FVIIa-sTF Inhibitors in the Blood Coagulation Cascade

, 13(1): 3 - 23

Andrea Roxanne J. Anas and Ken-ichi Harada


DOI: 10.2174/1570180812666150608230214



Development of Energy-based Pharmacophore Model and Stepwise Virtual Screening of LRRK2 Inhibitors Through Molecular Dynamics and Mechanics

, 13(1): 24 - 32

Sagar S. Bhayye, Kunal Roy and Achintya Saha


DOI: 10.2174/1570180812666150611185331



Studies on the IC50 of Trisubstituted Thiazoles as Cdc7 Kinase Inhibitors

, 13(1): 33 - 42

Huazhen Yang, Xun Liu, Zhiling Ye, Fucheng Song, Lianhua Cui, Zhuang Yu, Hongzong Si and Honglin Zhai


DOI: 10.2174/1570180812999150713144215



Molecular Simulation of HDAC1/3 Inhibitor: Insights into the Structural Basis of Selectivity

, 13(1): 43 - 46

Lei Zhang and Lihui Zhang


DOI: 10.2174/1570180812666150630183816



Recent Developments in the Synthesis and Applications of Anticancer Amonafide Derivatives. A Mini Review

, 13(1): 47 - 63

Gary Gellerman


DOI: 10.2174/1570180812666150529205049



A Series of 2,4(1H,3H)-Quinazolinedione Derivatives: Synthesis and Biological Evaluation as Potential Anticancer Agents

, 13(1): 64 - 76

Hulya Akgun, Demet Us Yilmaz, Rengul Cetin Atalay and Damla Gozen


DOI: 10.2174/1570180812666150529204909



Synthesis, Biological Evaluation and Molecular Docking Studies of 4Hbenzo[ h]chromenes, 7H-benzo[h]chromeno[2,3-d]pyrimidines as Antitumor Agents

, 13(1): 77 - 88

Ahmed H. Halawa, Ahmed M. Fouda, Al-Anood M. Al-Dies and Ahmed M. El-Agrody


DOI: 10.2174/1570180812666150611185830



Design, Synthesis and Biological Evaluation of 4-(Imidazolylmethyl)-2- Aryl-Quinoline Derivatives as Aromatase Inhibitors and Anti-breast Cancer Agents

, 13(1): 89 - 97

Razieh Ghodsi, Ebrahim Azizi, Maria Grazia Ferlin, Vincenzo Pezzi and Afshin Zarghi


DOI: 10.2174/1570180812666150611185605



Novel Aminopeptidase N Inhibitors with Improved Antitumor Activities

, 13(1): 98 - 106

Qiang Wang, Qiao Shi and Lu Huang


DOI: 10.2174/1570180812666150611190608



Biological Properties of Heterocyclic Pyridinylimines and Pyridinylhydrazones

, 13(1): 107 - 114

Francislene J. Martins, Rebeca Mol Lima, Juliana Alves dos Santos, Patricia de Almeida Machado, Elaine Soares Coimbra, Adilson David da Silva and Nádia Rezende Barbosa Raposo


DOI: 10.2174/1570180812666141216205601




Editor-in-Chief

K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
Biography
View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 1.05

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