Contents

Letters in Drug Design & Discovery, Volume 12 - Number 7



Anticancer Evaluation of 3,4,5,4'-trans-tetramethoxystilbene (DMU-212) and Its Analogs Against an Extensive Panel of Human Tumor Cell Lines

, 12(7): 521 - 528

Nikhil Reddy Madadi and Peter Anthony Crooks


DOI: 10.2174/1570180812999150324163710



6-Bromo-2,3-Dioxoindolin Phenylacetamide Derivatives: Synthesis, Potent CDC25B, PTP1B Inhibitors and Anticancer Activity

, 12(7): 529 - 536

Shui-Lian Zhao, Zhou Peng, Xing-Hua Zhen, Yan Han, Hai-Ying Jiang, You-Le Qu and Li-Ping Guan


DOI: 10.2174/1570180812666141219003209



3D-QSAR Study of Flavone Derivatives as Inhibitors of HeLa Cervix Adenocarcinoma Cell Lines

, 12(7): 537 - 544

Yeonjoong Yong, Yearam Jung, Eunil Cho, Hyeonji Kim, Jin Sil Yoo, Dongsoo Koh, Hi Jae Cho, Somi Kim Cho and Yoongho Lim


DOI: 10.2174/1570180812666141205235800



Proteins as Alternate Targets of Enediynes

, 12(7): 545 - 557

Hussam M. Bdour, Snigdha Roy and Amit Basak


DOI: 10.2174/1570180812666150213224756



Identification of Potential Mps1 Inhibitors Through Multiple Pharmacophore- based Virtual Screening and Molecular Docking

, 12(7): 558 - 573

Xiaoli Li, Lu Zhou, Yahui Tian and Suwen Zhou


DOI: 10.2174/1570180812999150210142710



Design, Synthesis and Biological Evaluation of Lapatinib Derivatives as HER1/HER2 Inhibitors

, 12(7): 574 - 584

Aifeng Lyu, Lei Fang, Shaohua Gou and Xia Liu


DOI: 10.2174/1570180812999150206111626



Synthesis and Preliminary Evaluation of Novel Bone-targeting NSAIDs Prodrugs based on Glutamic Acid Oligopeptides

, 12(7): 585 - 590

Yi Zhao, Dongsheng He, Lifang Ma and Li Guo


DOI: 10.2174/1570180812999150217171229



Syntheses of Ethyl Pyruvate’s Bioisosteres Inhibiting Inducible Nitric Oxide Production in Lipopolysaccharide-induced BV2 Cells

, 12(7): 591 - 596

Ju-Young Park, Byung-Wook Kim, Soon-Jung Kwon, Dong-Kug Choi, Ja-Kyeong Lee and Sung-Hwa Yoon


DOI: 10.2174/1570180812999150225112225



Synthesis and In vitro Evaluation of Dibenzoazepine Triazole Derivatives: A Novel Class of Antileishmanial Agents

, 12(7): 597 - 606

Maria Aqeel Khan, Aliyan Saleem, Nida Ghouri, Abdul Hameed, M. Iqbal Choudhary and Fatima Z. Basha


DOI: 10.2174/1570180812999150225111959



Synthesis and In Vitro Evaluation of Furan-Based Chalcone Derivatives as Antimicrobial Agents

, 12(7): 607 - 611

Ahmet Ozdemir, Mehlika Dilek Altıntop, Zerrin Canturk and Zafer Asim Kaplancikli


DOI: 10.2174/1570180812999150202112352




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