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Letters in Drug Design & Discovery

Volume 18, 12 Issues, 2021
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

In the current pandemic scenario, publication process of all articles related to Coronavirus will be expedited, for timely publication of much needed research


Letters in Drug Design & Discovery, Volume 12 - Number 6

First Efficient Two-Step/One-Pot Zirconium (IV)isopropoxide–Mediated Reductive Amination of Carbonyl Compounds

, 12(6): 448 - 456

Cyril Pieri and Jean Michel Brunel

DOI: 10.2174/1570180812666141215215120

FeCl3/Ultrasound Mediated Reaction of 2-aminothiophenol with Aldehydes in Water: Synthesis of 2-substituted Benzothiazoles of Pharmacological Interest

, 12(6): 457 - 465

Ponasanapalli Tirumala Venkata Ankayya Srinivas, Sallagundla Bhavani, Dandela Rambabu, Mandava Venkata Basaveswara Rao, Ravikumar Kapavarapu and Manojit Pal

DOI: 10.2174/1570180812666141216211045

Synthesis of Six Phenylalanine Derivatives and their Cell Toxicity Effect on Human Colon Cancer Cell Line HT-29

, 12(6): 466 - 470

Qianyi Zhao, Ting Xu, Menghua Li, Ying Yang, Haopeng Hu, Shupei Wang, Wenjuan Yan, Ran Chen, Chunyan Zhang and Cunshuan Xu

DOI: 10.2174/1570180812666141206001604

Synthesis and Antitumor Activity of New Pyrimidine and Caffeine Derivatives

, 12(6): 471 - 478

Ameen Ali Abu-Hashem and Hoda Abdel Raouf Hussein

DOI: 10.2174/1570180812666150429234237

De Novo Design of High Potent DPP-IV Inhibitors Based on the Scaffold of Cyanopyrrolidine

, 12(6): 479 - 487

Yu-Lei Jiang, Hao-Liang Yuan, Wei-Wei Zhang, Hai-Chun Liu, Yan-Min Zhang, Xiao Xiong, Jin-Xing Xu, Shuai Lu, Tao Lu and Ya-Dong Chen

DOI: 10.2174/1570180812666141201223016

Biological Evaluation of Halogenated Thioureas as Cholinesterases Inhibitors Against Alzheimer’s Disease & Molecular Modeling Studies

, 12(6): 488 - 494

Jamshed Iqbal, Sumera Zaib, Aamer Saeed and Muhammad Muddassar

DOI: 10.2174/1570180812666141201222247

Novel Fatty Acid Analogues as Human Fatty Acid Synthase Thioesterase Domain Inhibitors: Synthesis and their Cytotoxicity Screening

, 12(6): 495 - 499

Selvaraj Jubie, Pawan Kumar Yadhav, Moola Joghee Nanjan Chandrasekar, Jeyapal Gomathi Priya, Chaitanya MVNL and Palanisamy Dhanabal

DOI: 10.2174/1570180812666141216210751

Synthesis and Anti-tubercular Activity of 6-(4-Chloro/Methyl-phenyl)-4- Arylidene-4,5-dihydropyridazin-3(2H)-one Derivatives Against Mycobacterium tuberculosis

, 12(6): 500 - 504

Mohammad Asif and Anita Singh

DOI: 10.2174/157018081206150507130832

Synthesis, Characterization and Microbial Activity of new Aryl esters of 1,1'-bis(4-hydroxyphenyl)cyclohexane

, 12(6): 505 - 511

Chirag Bhupendra Patel, Bhavin Babu Dhaduk and Parsotam Hari Parsania

DOI: 10.2174/1570180812666141224211602

Preparation and Characterization of CS/(β-CD)/PAA Composite Hydrogels for Controlled Drug Delivery

, 12(6): 512 - 517

Jie Ren, Xiaoci Yang, Mengqi Yao, Jinfen Gu, Xiaohua Tang and W u Yang

DOI: 10.2174/1570180812666150224231250


K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 1.05


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