Contents

Letters in Drug Design & Discovery, Volume 12 - Number 5

Meet the Editorial Board Member

, 12(5): 343

Mihail Lucian Pascu


DOI: 10.2174/157018081205150324101302




Discovery of Novel HDAC Inhibitors by Structure-based Optimization of Cinnamic Hydroxamic Scaffold

, 12(5): 344 - 350

Chengqing Ning, Wenyuan Huang, Wen Wu, Cheng Lu, Yujun He, Lei Yao, Lifei Liu, Xiaohe Zhen, Xiaoyu Liu and Niefang Yu


DOI: 10.2174/1570180811666141024004832





Development of Structure Activity Correlation Model on Azetidin-2-ones as Tubulin Polymerization Inhibitors

, 12(5): 351 - 365

Vijay Kumar Patel, Kavibhushan Singh Chouhan, Avineesh Singh, Deepak Kumar Jain, Ravichandran Veerasamy, Pradeep Kumar. Singour, Rajesh Singh Pawar and Harish Rajak


DOI: 10.2174/1570180811666141010000110





Synthesis and Anticancer Activity of 7,8-dihydroxy-4-arylcoumarins

, 12(5): 366 - 373

Jianrui Wu, Ting Peng, Fang Chen, Yixin Leng, Linjiang Tong, Mengyuan Li, Rong Qu, Hua Xie, Jian Ding and Wenhu Duan


DOI: 10.2174/1570180812666141111235026





Hybrid Pharmacophore Design and Synthesis of Naphthalimide– Benzimidazole Conjugates as Potential Anticancer Agents

, 12(5): 374 - 384

Ahmed Kamal, Pogula Praveen Kumar, Mohammed Naseer Ahmed Khan, Bobburi Naga Sheshadri and Naga Sheshadri


DOI: 10.2174/1570180811666140915221955





Promising Anticancer Drug Candidates Based on the 7-methoxychromone Scaffold: Synthesis and Evaluation of Antiproliferative Activity

, 12(5): 385 - 392

Hoang Le Tuan Anh, Nguyen Thi Cuc, Pham Hai Yen, Nguyen Xuan Nhiem, Bui Huu Tai, Do Thi Thao, Nguyen Hoai Nam, Chau Van Minh, Phan Van Kiem and Young Ho Kim


DOI: 10.2174/1570180812666141111235539





Design, Synthesis and Biological Evaluation of Novel Fluorinated Heterocyclic Hybrid Molecules Based on Triazole & Quinoxaline Scaffolds Lead to Highly Potent Antimalarials and Antibacterials

, 12(5): 393 - 407

Adimulam Chandra Shekhar, Boddupally Pedda Venkat Lingaiah, Pamulaparthy Shanthan Rao, Banda Narsaiah, Aparna Devi Allanki and Puran Singh Sijwali


DOI: 10.2174/1570180812666141111235301





Synthesis of Derivatives of Artesunate α-Aminophosphonate and Their Antimicrobial Activities

, 12(5): 408 - 416

Sheng He, Xilin Ouyang, Xiaochao Huang, Weisong Hu, Weilong Dai, Xiaoyan Tian, Yingming Pan, Shiwen Huang and Hengshan Wang


DOI: 10.2174/1570180812666141125004502





Synthesis and Preliminary Biological Evaluation of New Heterocyclic Carboxamide Models

, 12(5): 417 - 429

Kamal Sweidan, Jorn Engelmann, Walid Abu Rayyan, Dima Sabbah, Musa Abu Zarga, Dima Sabbah, Tariq Al-Qirim, Yusuf Al-Hiari, Ghassan Abu Sheikha and Ghassan Shattat


DOI: 10.2174/1570180812666141201222527





Synthesis and Analysis of Anticonvulsant Activities of New 4-[2-(4- alkoxybenzylamino)ethyl]-2H-1,2,4-triazol-3(4H)-one Derivatives

, 12(5): 430 - 438

Qing-Kun Shen, Shi-Ben Wang, Guo-Hua Gong, Xiu-Mei Yin and Zhe-Shan Quan


DOI: 10.2174/1570180812666141111235746





Nematicidal Activity of Sprio and Bridged Heterocyclic Neonicotinoid Analogues against Meloidogyne incognita

, 12(5): 439 - 445

Minming Zou, Xue Tian, Nanyang Chen and Xusheng Shao


DOI: 10.2174/1570180812666141125003823





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