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Letters in Drug Design & Discovery

Volume 18, 12 Issues, 2021
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

In the current pandemic scenario, publication process of all articles related to Coronavirus will be expedited, for timely publication of much needed research


Letters in Drug Design & Discovery, Volume 12 - Number 4

The Synthesis of Risedronic Acid and Alendronate Applying Phosphorus Oxychloride and Phosphorous Acid in Methanesulfonic Acid

, 12(4): 253 - 258

Alajos Grun, Rita Kovacs, Sandor Garadnay, Istvan Greiner and Gyorgy Keglevich

DOI: 10.2174/1570180811666141010220427

Controlled Release from Solid Pharmaceutical Formulations of two Nalkanoyl- 4-methoxybicyclo[4.2.0]octa-1,3,5-trien-7-ethanamines with Melatoninergic Activity

, 12(4): 259 - 262

Marilena Vlachou, Vasiliki Ioannidou, Maria Vertzoni, Andrew Tsotinis, Pandelis A. Afroudakis and David Sugden

DOI: 10.2174/1570180811666141024005226

Synthesis, Antimicrobial and Pharmacological Evaluation of Thioureaderivatives of 4H-1,2,4-triazole

, 12(4): 263 - 276

Anna Bielenica, Ewa Kedzierska, Sylwia Fidecka, Hanna Maluszynska, Barbara Miroslaw, Anna E. Koziol, Joanna Stefanska, Silvia Madeddu, Gabriele Giliberti, Giuseppina Sanna and Marta Struga

DOI: 10.2174/1570180811666141001010044

First Discovery of Tylophora Alkaloids as HIV Inhibitors

, 12(4): 277 - 283

Ziwen Wang, Mingxiao Wang, Lei Wang, Xue Yao, Yue Li, Juan Tan, Wentao Qiao, Yunqi Geng, Yuxiu Liu and Qingmin Wang

DOI: 10.2174/1570180811666141009235124

Docking Study of Novel Pyrrolidine Derivatives as Potential Dipeptidyl Peptidase-IV (DPP-IV) Inhibitors

, 12(4): 284 - 291

Sant Kumar Verma, Shashi Kant Sharma and Suresh Thareja

DOI: 10.2174/1570180811666141016000752

Identification of Pyrazole Derivative as an Antiviral Agent Against Chikungunya Through HTVS

, 12(4): 292 - 301

Surender Singh Jadav, Barij Nayan Sinha, Boris Pastorino, Xavier de Lamballerie, Rolf Hilgenfeld and Venkatesan Jayaprakash

DOI: 10.2174/1570180811666141001005402

Computer-aided Identification of Novel DprE1 Inhibitors as Potential Anti-TB Lead Compounds: A Hybrid Virtual-screening and Molecular Dynamics Approach

, 12(4): 302 - 313

Yushir Maharaj, Soumendranath Bhakat and Mahmoud E. S. Soliman

DOI: 10.2174/1570180811666141001005536

Synthesis and Biological Activity of Acylthiourea Derivatives Contain 1,2,3-thiadiazole and 1,3,4-thiadiazole

, 12(4): 314 - 318

Ming-Yan Yang, Wen Zhao, Zhao-Hui Sun, Cheng-Xia Tan, Jian-Quan Weng and Xing-Hai Liu

DOI: 10.2174/1570180811666141010000435

Role of Curcumin in Modulating Plasma PON1 Arylesterase Activity and Susceptibility to LDL Oxidation in Oxidatively Challenged Wistar Rats

, 12(4): 319 - 323

Prabhakar Singh and Syed Ibrahim Rizvi

DOI: 10.2174/1570180811666141016000539

The Novel Derivatives of 3-(iminomethyl)-2H-chromen-2-one with Thiourea and Piperazine Structural Motive: Rationale, Synthesis, Antimicrobial and Anti-TB Evaluation

, 12(4): 324 - 341

Harshad P. Lakum, Dhruvin R. Shah and Kishor H. Chikhalia

DOI: 10.2174/1570180811666141009234835


K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 1.05


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