Letters in Drug Design & Discovery
Volume 18, 12 Issues, 2021
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access
Contents
Letters in Drug Design & Discovery, Volume 12 - Number 10
Novel Derivatives of Benfluron and Dimefluron Synthesis and Anticancer activity
, 12(10): 787 - 801Lenka Sucha, Marek Kolenic, Jiri Kratochvil, Milan Pour, Milan Nobilis, Eva Cermakova, Martina Rezacova and Pavel Tomsik
DOI: 10.2174/1570180812666150529204508
Novel Derivatives of Benfluron and Dimefluron Synthesis and Anticancer activity
Synthesis, Cytoprotective and Anti-Tumor Activities of Isatin Schiff Bases
, 12(10): 802 - 805Gang Chen, Mei Meng, Yu Zhang, Xiaojiang Hao, Ye Wang and Shuzhen Mu
DOI: 10.2174/1570180812666150514234029
Synthesis, Cytoprotective and Anti-Tumor Activities of Isatin Schiff Bases
Synthesis and Cytotoxicities of 2-[4-hydroxy-(3,5-bis-aminomethyl)- benzylidene]-indan-1-ones
, 12(10): 806 - 812Mehtap Tugrak, Halise Inci Gul and Hiroshi Sakagami
DOI: 10.2174/1570180812666150430002002
Synthesis and Cytotoxicities of 2-[4-hydroxy-(3,5-bis-aminomethyl)- benzylidene]-indan-1-ones
Synthesis, Anti-tumor Activity and Odd–even Effect of Simple Isatin Derivatives
, 12(10): 813 - 818Gang Chen, Xiaojiang Hao, Ye Wang and Shuzhen Mu
DOI: 10.2174/157018081210151012120940
Synthesis, Anti-tumor Activity and Odd–even Effect of Simple Isatin Derivatives
Discovery of New Inhibitors of Urease Enzyme: A Study Using STD-NMR Spectroscopy
, 12(10): 819 - 827Jalaluddin A. J. Awllia, Ayesha Sara, Atia-tul- Wahab, Maryam AL-Ghamdi, Saima Rasheed, Etimad Huwait and M. Iqbal Choudhary
DOI: 10.2174/1570180812666150520001629
Discovery of New Inhibitors of Urease Enzyme: A Study Using STD-NMR Spectroscopy
Syntheses and Activity of Carbohydrate-Containing Chitinase Inhibitors
, 12(10): 828 - 832Gangliang Huang, Xinya Mei, Xin Chen and Xiaomei Wang
DOI: 10.2174/1570180812666150514234246
Syntheses and Activity of Carbohydrate-Containing Chitinase Inhibitors
Effect of Acute Administration of 8-(Trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-amine Hydrochloride (TC-2153) on Biogenic Amines Metabolism in Mouse Brain
, 12(10): 833 - 836Elizabeth A. Kulikova, Ekaterina Y. Bazhenova, Nina K. Popova, Tatyana M. Khomenko, Konstantin P. Volcho, Nariman F. Salakhutdinov and Alexander V. Kulikov
DOI: 10.2174/1570180812666150522221634
Effect of Acute Administration of 8-(Trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-amine Hydrochloride (TC-2153) on Biogenic Amines Metabolism in Mouse Brain
3D-QSAR and Molecular Docking Studies of Flavonoid Derivatives as Potent Acetylcholinesterase Inhibitors
, 12(10): 837 - 843An Zhou, Zeyu Wu, Ailing Hui, Bin Wang, Xianchun Duan, Haixiang Wang and Jian Pan
DOI: 10.2174/1570180812666150514233543
3D-QSAR and Molecular Docking Studies of Flavonoid Derivatives as Potent Acetylcholinesterase Inhibitors
An Insight into Patents of Fluoroquinolone Derivatives
, 12(10): 844 - 855Prabodh Chander Sharma, Mona Piplani and Harish Rajak
DOI: 10.2174/1570180812666150429234635
An Insight into Patents of Fluoroquinolone Derivatives
Computational Docking Studies of Novel Heterocyclic Carboxamides as Potential PI3Kα Inhibitors
, 12(10): 856 - 863Kamal Sweidan, Dima A. Sabbah, Jorn Engelmann, Heba Abdel-Halim and Ghassan Abu Sheikha
DOI: 10.2174/1570180812666150529205248
Computational Docking Studies of Novel Heterocyclic Carboxamides as Potential PI3Kα Inhibitors
Synthesis and Biological Evaluation of 2´-Hydroxy-4´,6´-Diprenyloxychal-Cone Derivatives as Potent CDC25B and PTP1B Inhibitors
, 12(10): 864 - 871Dong-Hai Zhao, JIan Zhang, Lei Zhang, Da-Peng Li, Zhou Peng and Li-Ping Guan
DOI: 10.2174/1570180812666150723002629
Synthesis and Biological Evaluation of 2´-Hydroxy-4´,6´-Diprenyloxychal-Cone Derivatives as Potent CDC25B and PTP1B Inhibitors
Editor-in-Chief
K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
Biography
University of Hradec Kralove
Hradec Kralove
Biography
Biography of K. Kuca
Kamil Kuca is working for several academic institutes (University of Hradec Kralove, Czech Republic; University Hospital Hradec Kralove, Czech republic; Florida International University, USA; Yangtze University, China; etc.). He is recently rector of the University of Hradec Kralove. He was also technology scout focused on biomedicine in the past. His research interests are toxicology, pharmacology, drug design, technology transfer, pharmacoeconomy, chemical and biological terrorism, etc. He was/is principal investigator on numerous national and international projects (EU, NATO, GACR, IGA MZ, MSMT etc.). He has published more than 350 IF research papers. He is working with several companies as a scientific consultant. He has lots of cooperators throughout the world (e.g. Korea, Croatia, United Arab Emirates, USA, France, Turkey, China, Singapore, Sweden, and Brazil). His Hindex is 36, number of citation in WoS is over 3000.
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Journal History
Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
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