Contents

Letters in Drug Design & Discovery, Volume 12 - Number 1

Editorial

Editorial

, 12(1): 1

Atta-ur-Rahman


DOI: 10.2174/157018081201141030111644




Identification of Novel GSK1070916 Analogs as Potential Aurora B Inhibitors: Insights from Molecular Dynamics and MM/GBSA Based Rescoring

, 12(1): 2 - 13

Faraz Shaikh, Soumendranath Bhakat, Abhishek Thakur, Ashish Radadiya, Mahmoud E. S. Soliman and Anamik Shah


DOI: 10.2174/1570180811666140725184953





Design, Synthesis and Antimycobacterial Activity of Some New Azaheterocycles: Phenanthroline with p-halo-benzoyl Skeleton. Part V

, 12(1): 14 - 19

Ramona Danac, Teofil Daniloaia, Vasilichia Antoci, Violeta Vasilache and Ionel I. Mangalagiu


DOI: 10.2174/1570180811666140819223501





Design, Synthesis and Cytotoxic Evaluation of Novel Imatinib Amide Derivatives that Target Abl Kinase

, 12(1): 20 - 28

Ri-Sheng Yao, Qiu-Xiang Guan, Xiao-Qin Lu and Ban-Feng Ruan


DOI: 10.2174/1570180811666140812231519





Design, Synthesis and Antitubercular Evaluation of New 2-amino-5-(4- (benzyloxy)benzyl)thiophene-3-carboxylic Acid Derivatives. Part 3

, 12(1): 29 - 37

Xiaoyun Lu, Jian Tang, Qidong You, Baojie Wan and Scott G. Franzblau


DOI: 10.2174/1570180811666140812231321





Design, Synthesis and Biological Evaluation of Benzimidazole-pyridine- Piperidine Hybrids as a New Class of Potent Antimicrobial Agents

, 12(1): 38 - 45

Kothapally. Beulah, Akula Ravi Kumara, Boddupally Peda Venkat Lingaiah, Pamulaparthy Shanthan Rao, Banda Narsaiah, Aaramadaka Sunil Kumar Reddy and Upadhyayula Surya Narayana Murty


DOI: 10.2174/1570180811666140725185713





Structure Based Functional Annotation of Putative Conserved Proteins from Treponema pallidum: Search for a Potential Drug Target

, 12(1): 46 - 59

Avni Sinha, Faizan Ahmad and Md. Imtaiyaz Hassan


DOI: 10.2174/1570180811666140806005822





Theoretical Modelling of Potential Chk1 Inhibitors

, 12(1): 60 - 65

Pedro M.M. Araujo, Luis Pinto da Silva and Joaquim C.G. Esteves da Silva


DOI: 10.2174/1570180811666140725190051





A Screening Method for Potential Anti-pancreatic Cancer Candidate Compounds Based on Hsp90-Cdc37 Interaction Model in vitro

, 12(1): 66 - 71

Hai Zhang, Sen Sun, Qingshan Chen, Guoqing Zhang, Zhenqing Zhang, Duxin Sun and Wenpeng Zhang


DOI: 10.2174/1570180811666140725185235





Synthesis and Evaluation of Transdermal Permeation, Pharmacological Activity of Bornyl NSAID Esters

, 12(1): 72 - 77

Jiufeng Lin, Kefeng Ni, Yang Zhang, Dongzhi Wei and Yuhong Ren


DOI: 10.2174/1570180811666140627004820





Efficient Synthesis of Benzidronate Applying of Phosphorus Trichloride and Phosphorous Acid

, 12(1): 78 - 84

Alajos Grun, Rita Kovacs, David Illes Nagy, Sandor Garadnay, Istvan Greiner and Gyorgy Keglevich


DOI: 10.2174/1570180811666141001004732





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