Contents

Letters in Drug Design & Discovery, Volume 11 - Number 9

Modeling the Active Conformation of Human µ Opioid Receptor

, 11(9): 1053 - 1061

Agnieszka A. Kaczor, Damian Bartuzi and Dariusz Matosiuk


DOI: 10.2174/1570180811666140322001506





Synthesis and In vitro Evaluation of Thiadiazole Derivatives as AChE, Bu- ChE and LOX Inhibitors

, 11(9): 1062 - 1069

Mehlika Dilek Altintop, Ahmet Ozdemir, Usama Abu Mohsen, Halide Edip Temel, Gulsen Akal n Ciftci and Zafer Asim Kaplancikli


DOI: 10.2174/1570180811666140529004517





Synthesis and Studies on Anticonvulsant and Antibacterial Activities of 1- Alkyl-4-(4H-1,2,4-triazol-4-yl)piperidine Derivatives

, 11(9): 1070 - 1078

Yan-Ping Yuan, Shi-Ben Wang, Guo-Hua Gong and Zhe-Shan Quan


DOI: 10.2174/1570180811666140623204022





Design, Synthesis and Antitumor Activities of Bis-arylureas and Bis-arylamides Based on1H-benzo[d]imidazole Moiety as Novel BRafV600E/VEGFR2 Dual inhibitors

, 11(9): 1079 - 1089

Weimin Yang, Yadong Chen, Yanmin Zhang, Sanzhi Tang, Hongli Chen, Weifang Tang and Tao Lu


DOI: 10.2174/1570180811666140724184806





To Preliminarily Evaluate The Anticancer Activiy of 1,2-di(quinazolin-4- yl)diselane Against MDA-MB-435 Cells in vitro

, 11(9): 1090 - 1095

Yinjiu Huang, Hong Xie, Gang Liu, Xiaomei Hu, Lin Su, Jianguo Hu, Qiyi Wang and Yibo Ding


DOI: 10.2174/1570180811666140617212723





Evaluation of Alkylating and Intercalating Properties of Mannich Bases for Cytotoxic Activity

, 11(9): 1096 - 1106

Huseyin Istanbullu, Yalcin Erzurumlu, Petek Ballar Kirmizibayrak and Ercin Erciyas


DOI: 10.2174/1570180811666140529005029





Synthesis and Antifungal Activity of 1,3,4-Thiadiazole Derivatives Containing Pyridine Group

, 11(9): 1107 - 1111

Lin-Jiong Zhang, Ming-Yan Yang, Zhao-Hui Sun, Cheng-Xia Tan, Jian-Quan Weng, Hong-Ke Wu and Xing-Hai Liu


DOI: 10.2174/1570180811666140610212731





Pharmacokinetic Modeling of Caco-2 Cell Permeability Using Genetic Programming (GP) Method

, 11(9): 1112 - 1118

Renu Vyas, Purva Goel, M. Karthikeyan, S.S. Tambe and B.D. Kulkarni


DOI: 10.2174/1570180811666140610213438





Synthesis and Bioactivities of Novel 1,3,4-oxadiazole Derivatives Containing Pyridine Moiety

, 11(9): 1119 - 1123

Guo-Xiang Sun, Yan-Xia Shi, Zhao-Hui Sun, Ming-Yan Yang, Hong-Ke Wu, Jian-Quan Weng, Cheng-Xia Tan, Xing-Hai Liu, Bao-Ju Li and Yong-Gang Zhang


DOI: 10.2174/1570180811666140522002929





Solvent-Free Synthesis and Insecticidal Activities of C6-Esterified Coumarins

, 11(9): 1124 - 1132

Ying Xie, Zheng-Lin Lei and Yan-Ping Luo


DOI: 10.2174/1570180811666140603003043





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