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Letters in Drug Design & Discovery

Volume 17, 12 Issues, 2020
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

In the current pandemic scenario, publication process of all articles related to Coronavirus will be expedited, for timely publication of much needed research

Contents

Letters in Drug Design & Discovery, Volume 11 - Number 8

Synthesis and Antitubercular Activities in Vitro of New p-Aminosalicylic Ester Imines

, 11(8): 953 - 959

Michael J. Hearn, Daniel J. Smaltz and Michael H. Cynamon


DOI: 10.2174/1570180811666140516233652



Synthesis and Antimicrobial Activities of (4,5,6,7-Tetrahydro-1H-indazol- 2(3H)-yl)thiazole Derivatives

, 11(8): 960 - 967

Krzysztof Z. Laczkowski, Konrad Misiura, Anna Biernasiuk and Anna Malm


DOI: 10.2174/1570180811666140516233913



Synthesis and Antimycobacterial Activity of Highly Functionalised Pyrrolothiazole Derivatives

, 11(8): 968 - 974

Abdulrahman I. Almansour, Venu Sanjeevi Lakshmipathi, Elumalai Manogaran, Mohamed Ashraf Ali, Farzana Beevi, Tan Soo Choon, Ang Chee Wei, Raju Suresh Kumar and Mohammad Asad


DOI: 10.2174/1570180811666140506204239



Synthesis and Biological Activity of Novel 1-((benzofuran-2-yl)methyl)-1Htriazole Derivatives

, 11(8): 975 - 984

Yi-Min Shi, Li-Juan Yang, Wen Chen, Cheng-Jun Sun, Xiao-Liang Xu, Shu-Ya Zhou, Hong- Bin Zhang and Xiao-Dong Yang


DOI: 10.2174/1570180811666140423214501



Synthesis, Biological Evaluation and the Rationalisation of the Inhibitory Activity of a Range of Sulfonate Derivatives of Estrone (E1) in the Design of Reversible Inhibitors of Estrone Sulfatase (ES)

, 11(8): 985 - 992

Mohsen Akbarzadeh, Timothy Cartledge and Sabbir Ahmed


DOI: 10.2174/1570180811666140226235116



Synthesis and Evaluation of 4-arylmethyl Curcumin Analgues as Potent Hsp90 Inhibitors

, 11(8): 993 - 999

Yang Liu, Min Ye, Qundan Wu, Lixian Wu and Jianhua Xu


DOI: 10.2174/1570180811666140512221037



Synthesis and Biochemical Evaluation of a Range of 4-(n-alkanesulfonate) benzyl Imidazole-Based Compounds as Inhibitors of Rat Testicular 17α-hydroxylase/17,20-lyase (P45017α) in the Treatment of Hormone- Dependent Prostate Cancer

, 11(8): 1000 - 1009

Pallav S. Shah, Imran Shahid, Wai-Yee Lee, Caroline P. Owen and Sabbir Ahmed


DOI: 10.2174/1570180811666131230235538



Library of Synthetic Compounds Based on Pyrazole Unit: Design and Screening Against Breast and Colorectal Cancer

, 11(8): 1010 - 1016

Farid Abrigach, Mohamed Khoutoul, Noureddine Benchat, Smaail Radi, Nihed Draoui, Olivier Feron, Olivier Riant and Rachid Touzani


DOI: 10.2174/1570180811666140512220842



Quantitative Structure-Retention Relationships Studies of Selected Groups of Compounds Characterized by Different Pharmacological Activity Using Multiple Linear Regression Procedure

, 11(8): 1017 - 1039

Jolanta Stasiak, Marcin Koba and Tomasz Baczek


DOI: 10.2174/1570180811666140506204742



Synthesis and Anticonvulsant Activity of N-(trans)- 3-phenylprop-2-en-1-yl (Cinnamyl) Derivatives of Aminoalkanols

, 11(8): 1040 - 1052

Agnieszka Gunia-Krzyzak, Anna M. Waszkielewicz, Karolina Sloczynska, Magda Borczuch- Kostanska, Marek Cegla, Grzegorz Satala, Andrzej J. Bojarski and Henryk Marona


DOI: 10.2174/1570180811666140423203639




Editor-in-Chief

K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
Biography
View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 1.05

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