Contents

Letters in Drug Design & Discovery, Volume 11 - Number 8

Synthesis and Antitubercular Activities in Vitro of New p-Aminosalicylic Ester Imines

, 11(8): 953 - 959

Michael J. Hearn, Daniel J. Smaltz and Michael H. Cynamon


DOI: 10.2174/1570180811666140516233652



Synthesis and Antimicrobial Activities of (4,5,6,7-Tetrahydro-1H-indazol- 2(3H)-yl)thiazole Derivatives

, 11(8): 960 - 967

Krzysztof Z. Laczkowski, Konrad Misiura, Anna Biernasiuk and Anna Malm


DOI: 10.2174/1570180811666140516233913



Synthesis and Antimycobacterial Activity of Highly Functionalised Pyrrolothiazole Derivatives

, 11(8): 968 - 974

Abdulrahman I. Almansour, Venu Sanjeevi Lakshmipathi, Elumalai Manogaran, Mohamed Ashraf Ali, Farzana Beevi, Tan Soo Choon, Ang Chee Wei, Raju Suresh Kumar and Mohammad Asad


DOI: 10.2174/1570180811666140506204239



Synthesis and Biological Activity of Novel 1-((benzofuran-2-yl)methyl)-1Htriazole Derivatives

, 11(8): 975 - 984

Yi-Min Shi, Li-Juan Yang, Wen Chen, Cheng-Jun Sun, Xiao-Liang Xu, Shu-Ya Zhou, Hong- Bin Zhang and Xiao-Dong Yang


DOI: 10.2174/1570180811666140423214501



Synthesis, Biological Evaluation and the Rationalisation of the Inhibitory Activity of a Range of Sulfonate Derivatives of Estrone (E1) in the Design of Reversible Inhibitors of Estrone Sulfatase (ES)

, 11(8): 985 - 992

Mohsen Akbarzadeh, Timothy Cartledge and Sabbir Ahmed


DOI: 10.2174/1570180811666140226235116



Synthesis and Evaluation of 4-arylmethyl Curcumin Analgues as Potent Hsp90 Inhibitors

, 11(8): 993 - 999

Yang Liu, Min Ye, Qundan Wu, Lixian Wu and Jianhua Xu


DOI: 10.2174/1570180811666140512221037



Synthesis and Biochemical Evaluation of a Range of 4-(n-alkanesulfonate) benzyl Imidazole-Based Compounds as Inhibitors of Rat Testicular 17α-hydroxylase/17,20-lyase (P45017α) in the Treatment of Hormone- Dependent Prostate Cancer

, 11(8): 1000 - 1009

Pallav S. Shah, Imran Shahid, Wai-Yee Lee, Caroline P. Owen and Sabbir Ahmed


DOI: 10.2174/1570180811666131230235538



Library of Synthetic Compounds Based on Pyrazole Unit: Design and Screening Against Breast and Colorectal Cancer

, 11(8): 1010 - 1016

Farid Abrigach, Mohamed Khoutoul, Noureddine Benchat, Smaail Radi, Nihed Draoui, Olivier Feron, Olivier Riant and Rachid Touzani


DOI: 10.2174/1570180811666140512220842



Quantitative Structure-Retention Relationships Studies of Selected Groups of Compounds Characterized by Different Pharmacological Activity Using Multiple Linear Regression Procedure

, 11(8): 1017 - 1039

Jolanta Stasiak, Marcin Koba and Tomasz Baczek


DOI: 10.2174/1570180811666140506204742



Synthesis and Anticonvulsant Activity of N-(trans)- 3-phenylprop-2-en-1-yl (Cinnamyl) Derivatives of Aminoalkanols

, 11(8): 1040 - 1052

Agnieszka Gunia-Krzyzak, Anna M. Waszkielewicz, Karolina Sloczynska, Magda Borczuch- Kostanska, Marek Cegla, Grzegorz Satala, Andrzej J. Bojarski and Henryk Marona


DOI: 10.2174/1570180811666140423203639




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