Contents

Letters in Drug Design & Discovery, Volume 11 - Number 6

Analysis of Proteasome Inhibition Prediction Using Atom-Based Quadratic Indices Enhanced by Machine Learning Classification Techniques

, 11(6): 705 - 711

Gerardo M. Casanola-Martin, Huong Le-Thi-Thu, Yovani Marrero-Ponce, Juan A Castillo- Garit, Francisco Torrens, Facundo Perez-Gimenez and Concepcion Abad


DOI: 10.2174/1570180811666140122001144



Synthesis and Antioxidant Activity of Novel Quinazolinones Functionalized with Urea/Thiourea/Thiazole Derivatives as 5-Lipoxygenase Inhibitors

, 11(6): 712 - 720

Maralekere K. Prashanth and Hosakere D. Revanasiddappa


DOI: 10.2174/1570180811666131230235157



Design, Synthesis and Biological Evaluation of Some Oxadiazole Derivatives as Novel Amide-Based Inhibitors of Soluble Epoxide Hydrolase

, 11(6): 721 - 730

Elham Rezaee Zavareh, Mahdi Hedayati, Laleh Hoghooghi Rad, Azin Kiani, Soraya Shahhosseini, Mehrdad Faizi and Sayyed Abbas Tabatabai


DOI: 10.2174/1570180811666140220005530



A Potential Anticancer Agent 1,2-di(quinazolin-4-yl)diselane

, 11(6): 731 - 735

Yinjiu Huang, Gang Liu, Xiaomei Hu, Hao Liu, Jianguo Hu, Zhenzhong Feng, Bi Tang, Jun Qian, Qiyi Wang and Xuehui Long


DOI: 10.2174/1570180811666140214204858



Synthesis and Anti-Cancer Activities of Aryl Benzyl Ethers with Fluoro Substituents

, 11(6): 736 - 741

Yi Jiang, Hong Xu, Li Liu, Rui He, Xiaomei Song and Na Li


DOI: 10.2174/1570180811666140130232233



Anticancer Activity and DNA Binding of 4-Alkylenediamines Modified Naphthalimide Derivatives

, 11(6): 742 - 748

Ke-Rang Wang, Feng Qian, Zi-Bo Yang, Hong-Wei An, Dan Han, Hua Chen, Ping-Zhu Zhang and Xiao-Liu Li


DOI: 10.2174/1570180811666140121234834



Design, Synthesis and Biological Evaluation of 5-Amino-1H-pyrazole-4- carboxamide Derivatives as Potential Antitumor Agents

, 11(6): 749 - 755

Baowei Yang, Wukun Liu, Yicheng Mei, Dandan Huang, Hai Qian, Wenlong Huang and Ronald Gust


DOI: 10.2174/1570180811666140115234123



Synthesis of Novel Macrocyclic Tetraamides

, 11(6): 756 - 761

Barun Kumar Mehta, Dandela Rambabu, Guttikonda Raja, ASG. Prasad, Jim-Min Fang and Mandava Venkata Basaveswara Rao


DOI: 10.2174/1570180811666140116215724



Design, Synthesis and Biological Evaluation of 2, 4, 5-Triphenylimidazole Derivatives with Preliminary SAR

, 11(6): 762 - 769

Chunqi Hu, Jianfeng Shen, Kejun Bian, Ruoyu Zhang and Liping Deng


DOI: 10.2174/1570180811666140116214111



Pharmacokinetic Analysis of Tetramethylpyrazine Bis-Nitrone TN-2 in Rats and its Protein Binding In Vitro

, 11(6): 770 - 777

Yewei Sun, Kaiyi Liao, Sai Li, Zaijun Zhang, Pei Yu and Yuqiang Wang


DOI: 10.2174/1570180811666140121234608



Novel 4-Oxothienopyrimidinyl Propanoic Acid Derivatives as AMPActivated Protein Kinase (AMPK) Activators

, 11(6): 778 - 785

Pradip K. Sasmal, Mahaboobi Jaleel, P. Tirumala Rao, M. Munikumar, Megha Bhattacharya, Nutakki Ravi Kumar, Poondla. Neelima, Khaji Abdul Rawoof, P. Narasimha Rao, Chandrasekhar Abbineni, M. Roshaiah, S. Sridhar, Thammera Ranjith Kumar, Menon C. A. Vinu, Vijay Potluri, Parimal Misra, Rashmi Talwar and Saibal Kumar Das


DOI: 10.2174/1570180811666140122003044



Influence of the Preparation Method on the Dissolution Properties of Piroxicam - Cyclodextrins Systems

, 11(6): 786 - 808

F. Bouchal, M. Skiba, S. Fatmi, N. Chaffai and M. Lahiani-Skiba


DOI: 10.2174/1570180811666140207215957



Positively Charged Nitrogen is Not Indispensable Requirement for Binding of Nitrogenous κ-Opioid Agonists: Insights from Docking Studies

, 11(6): 809 - 813

Indrani Bera and Nanda Ghoshal


DOI: 10.2174/1570180811666140220004853



Synthesis and Biological Activity of Thiazole Dithiocarbamate Derivatives

, 11(6): 814 - 823

Nalan Gundogdu-Karaburun


DOI: 10.2174/1570180811999140515100911




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