Contents
Letters in Drug Design & Discovery, Volume 11 - Number 5
Graphical Abstract
Synthesis of Oxygenated Chalcones with Anti-Staphylococcal Activity
, 11(5): 525 - 530Luciana Dalla-Vechia, Cíntia Janine Kiekow, Ivana Correa Ramos Leal, Katia Regina Netto Dos Santos, Simone Cristina Baggio Gnoatto, Hugo Verli, Rodrigo Octavio Mendonca Alves de Souza and Grace Gosmann
DOI: 10.2174/1570180810666131125221032
Designing New 5-Nitroimidazoles: Towards Safer Anti-infectious Agents
, 11(5): 531 - 559Maxime D. Crozet, Thierry Terme and Patrice Vanelle
DOI: 10.2174/1570180810666131122010615
Novel Urea/Thiourea Derivatives of Quinazolin-4(3H)-one: Design, Synthesis, Antimicrobial and Anti-TB Study
, 11(5): 560 - 571Dhruvin R. Shah, Rahul P. Modh, Dhara V. Desai and Kishor H. Chikhalia
DOI: 10.2174/1570180810666131122003517
Novel 4-bromo-2-(3-methyl-1-(substituted-phenylsulfonyl)-4,5-dihydro-1- H-pyrazol-5-yl)phenol Derivatives: Synthesis and Antibacterial Activity
, 11(5): 572 - 577Qing Chenga, Ying-Ming Jia, Fei-Hu Cheng and Xin-Hua Liu
DOI: 10.2174/1570180810666131122234935
Synthesis and Anticancer Activity of Some 2-[3/4-(2-Substituted Phenyl-2- oxoethoxy)benzylidene]-6-substituted-2,3-dihydro-1H-inden-1-one Derivatives
, 11(5): 578 - 585Nalan Gundogdu-Karaburun, Ahmet Cagri Karaburun, Seref Demirayak, Ismail Kayagil and Leyla Yurttas
DOI: 10.2174/1570180811666140403001212
Synthesis and Antitumor Activities of α-,γ-mangostin Derivatives
, 11(5): 586 - 593Kai Cheng, Gui-lin Zhang, Sheng-xiang Qiu, Yan-qing Liu, Yan-fei Wang, Song Liu, Yan Shan, Bo Yu and Yu Lu
DOI: 10.2174/1570180811666131217003216
A Facile Synthesis and Anticancer Activity Evaluation of Spiro Analogues of Benzothiazolylchromeno/pyrano Derivatives
, 11(5): 594 - 600Anand Kumar Arya, Kulbhushan Rana and Mahendra Kumar
DOI: 10.2174/1570180811666131210000903
Design, Synthesis and In-Vitro Evaluation of Polymer-linked Prodrug of Methotrexate for the Targeted Delivery to the Colon
, 11(5): 601 - 610Nishu Singla, Rajiv Sharma and T.R. Bhardwaj
DOI: 10.2174/1570180811666131217002719
Potent Neuroprotective Activity of Monoterpene Derived 4-[(3aR,7aS)- 1,3,3a,4,5,7a-Hexahydro-3,3,6-trimethylisobenzofuran-1-yl]-2-methoxyphenol in MPTP Mice Model
, 11(5): 611 - 617Alla V. Pavlova, Irina V. Il'ina, Ekaterina A. Morozova, Dina V. Korchagina, Svetlana Yu. Kurbakova, Irina V. Sorokina, Tatyana G. Tolstikova, Konstantin P. Volcho and Nariman F. Salakhutdinov
DOI: 10.2174/1570180811666131210000316
QSAR Study on Diketo Acid and Carboxamide Derivatives as Potent HIV- 1 Integrase Inhibitor
, 11(5): 618 - 627Arodola Olayide Adebimpe, Radha Charan Dash and Mahmoud E. S. Soliman
DOI: 10.2174/1570180811666131217003010
Synthesis and Anticonvulsant Activity Evaluation of 4-butyl-5-(4- alkoxyphenyl)-2H-1,2,4-triazole-3(4H)-ones
, 11(5): 628 - 635Zi-Shi Zhu, Shi-Ben Wang, Xian-Qing Deng, Da-Chuan Liu and Zhe-Shan Quan
DOI: 10.2174/1570180810666131122003939
Artificial Neural Networks Modeling of Release of Olanzapine From Glycerol Monooleate Matrices
, 11(5): 636 - 648G. Bagheri, E. Vasheghani-Farahani, M. Ardjmand, H. Attar and F. A. Dorkoosh
DOI: 10.2174/1570180811666131227193958
4D-QSAR Model for Compounds with Binding Affinity Towards Dopamine D2 Receptors
, 11(5): 649 - 664Daniela Rodrigues Silva, Teodorico C. Ramalho and Elaine F. F. da Cunha
DOI: 10.2174/1570180810666131113213448
A Combined DFT and QSAR Calculations to Study Substituted Biphenyl imidazoles as Bombesin Receptor Subtype-3 Agonists
, 11(5): 665 - 676Mohsen Shahlaei, Amin Nowroozi and Reza Khodarahmi
DOI: 10.2174/1570180811666131203002858
Synthesis and In Vivo Hepatoprotective Activity of Some Novel Andrographolide Derivatives
, 11(5): 677 - 685Chunlei Tang, Guolong Gu, Baowei Yang, Xuekun Wang, Hai Qian, Wenlong Huang, Xiaoyun Zhu and Jing Li
DOI: 10.2174/1570180810666131123002409
Development of Pyrazole Compounds as Antidiabetic Agent: A Review
, 11(5): 686 - 703Prasanna A. Datar and Sonali R. Jadhav
DOI: 10.2174/1570180810666131113212354
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