Contents

Letters in Drug Design & Discovery, Volume 11 - Number 5

Graphical Abstract

Graphical Abstracts

, 11(5): i - viii


DOI: 10.2174/157018081105140424145741




Synthesis of Oxygenated Chalcones with Anti-Staphylococcal Activity

, 11(5): 525 - 530

Luciana Dalla-Vechia, Cíntia Janine Kiekow, Ivana Correa Ramos Leal, Katia Regina Netto Dos Santos, Simone Cristina Baggio Gnoatto, Hugo Verli, Rodrigo Octavio Mendonca Alves de Souza and Grace Gosmann


DOI: 10.2174/1570180810666131125221032




Designing New 5-Nitroimidazoles: Towards Safer Anti-infectious Agents

, 11(5): 531 - 559

Maxime D. Crozet, Thierry Terme and Patrice Vanelle


DOI: 10.2174/1570180810666131122010615




Novel Urea/Thiourea Derivatives of Quinazolin-4(3H)-one: Design, Synthesis, Antimicrobial and Anti-TB Study

, 11(5): 560 - 571

Dhruvin R. Shah, Rahul P. Modh, Dhara V. Desai and Kishor H. Chikhalia


DOI: 10.2174/1570180810666131122003517




Novel 4-bromo-2-(3-methyl-1-(substituted-phenylsulfonyl)-4,5-dihydro-1- H-pyrazol-5-yl)phenol Derivatives: Synthesis and Antibacterial Activity

, 11(5): 572 - 577

Qing Chenga, Ying-Ming Jia, Fei-Hu Cheng and Xin-Hua Liu


DOI: 10.2174/1570180810666131122234935




Synthesis and Anticancer Activity of Some 2-[3/4-(2-Substituted Phenyl-2- oxoethoxy)benzylidene]-6-substituted-2,3-dihydro-1H-inden-1-one Derivatives

, 11(5): 578 - 585

Nalan Gundogdu-Karaburun, Ahmet Cagri Karaburun, Seref Demirayak, Ismail Kayagil and Leyla Yurttas


DOI: 10.2174/1570180811666140403001212




Synthesis and Antitumor Activities of α-,γ-mangostin Derivatives

, 11(5): 586 - 593

Kai Cheng, Gui-lin Zhang, Sheng-xiang Qiu, Yan-qing Liu, Yan-fei Wang, Song Liu, Yan Shan, Bo Yu and Yu Lu


DOI: 10.2174/1570180811666131217003216




A Facile Synthesis and Anticancer Activity Evaluation of Spiro Analogues of Benzothiazolylchromeno/pyrano Derivatives

, 11(5): 594 - 600

Anand Kumar Arya, Kulbhushan Rana and Mahendra Kumar


DOI: 10.2174/1570180811666131210000903




Design, Synthesis and In-Vitro Evaluation of Polymer-linked Prodrug of Methotrexate for the Targeted Delivery to the Colon

, 11(5): 601 - 610

Nishu Singla, Rajiv Sharma and T.R. Bhardwaj


DOI: 10.2174/1570180811666131217002719




Potent Neuroprotective Activity of Monoterpene Derived 4-[(3aR,7aS)- 1,3,3a,4,5,7a-Hexahydro-3,3,6-trimethylisobenzofuran-1-yl]-2-methoxyphenol in MPTP Mice Model

, 11(5): 611 - 617

Alla V. Pavlova, Irina V. Il'ina, Ekaterina A. Morozova, Dina V. Korchagina, Svetlana Yu. Kurbakova, Irina V. Sorokina, Tatyana G. Tolstikova, Konstantin P. Volcho and Nariman F. Salakhutdinov


DOI: 10.2174/1570180811666131210000316




QSAR Study on Diketo Acid and Carboxamide Derivatives as Potent HIV- 1 Integrase Inhibitor

, 11(5): 618 - 627

Arodola Olayide Adebimpe, Radha Charan Dash and Mahmoud E. S. Soliman


DOI: 10.2174/1570180811666131217003010




Synthesis and Anticonvulsant Activity Evaluation of 4-butyl-5-(4- alkoxyphenyl)-2H-1,2,4-triazole-3(4H)-ones

, 11(5): 628 - 635

Zi-Shi Zhu, Shi-Ben Wang, Xian-Qing Deng, Da-Chuan Liu and Zhe-Shan Quan


DOI: 10.2174/1570180810666131122003939




Artificial Neural Networks Modeling of Release of Olanzapine From Glycerol Monooleate Matrices

, 11(5): 636 - 648

G. Bagheri, E. Vasheghani-Farahani, M. Ardjmand, H. Attar and F. A. Dorkoosh


DOI: 10.2174/1570180811666131227193958




4D-QSAR Model for Compounds with Binding Affinity Towards Dopamine D2 Receptors

, 11(5): 649 - 664

Daniela Rodrigues Silva, Teodorico C. Ramalho and Elaine F. F. da Cunha


DOI: 10.2174/1570180810666131113213448




A Combined DFT and QSAR Calculations to Study Substituted Biphenyl imidazoles as Bombesin Receptor Subtype-3 Agonists

, 11(5): 665 - 676

Mohsen Shahlaei, Amin Nowroozi and Reza Khodarahmi


DOI: 10.2174/1570180811666131203002858




Synthesis and In Vivo Hepatoprotective Activity of Some Novel Andrographolide Derivatives

, 11(5): 677 - 685

Chunlei Tang, Guolong Gu, Baowei Yang, Xuekun Wang, Hai Qian, Wenlong Huang, Xiaoyun Zhu and Jing Li


DOI: 10.2174/1570180810666131123002409




Development of Pyrazole Compounds as Antidiabetic Agent: A Review

, 11(5): 686 - 703

Prasanna A. Datar and Sonali R. Jadhav


DOI: 10.2174/1570180810666131113212354




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