Bentham Science Logo

Track Your Manuscript:


Letters in Drug Design & Discovery

Volume 17, 12 Issues, 2020
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

In the current pandemic scenario, publication process of all articles related to Coronavirus will be expedited, for timely publication of much needed research

Contents

Letters in Drug Design & Discovery, Volume 11 - Number 4


In Vitro Antitumoral Activity of Palladium(II) and Platinum(II) Complexes with O,O'-Dialkyl Esters of Ethylene-bis(S)-Leucine

, 11(4): 387 - 394

Jelena M. Vujic, Goran N. Kaluderovic, Tatjana P. Stanojkovic, Jadranka A. Antic and Srecko R. Trifunovic


DOI: 10.2174/15701808113106660092



Synthesis and Antitumor Invasive Activity of Novel Ionone Alkaloid Derivatives

, 11(4): 395 - 402

Hai-Jun Fang, Qian Liu, Chun-Chun Gan, Mei-Na Jin, Nan Qin and Hong-Quan Duan


DOI: 10.2174/15701808113106660094



Toward the Identification of Novel Carbonic Anhydrase XIV Inhibitors using 3D-QSAR Pharmacophore Model, Virtual Screening and Molecular Docking Study

, 11(4): 403 - 412

Tao Liu, Lu Zhou, Taijin Wang, Lufen He and Xiangyang Tang


DOI: 10.2174/15701808113106660083



Synthesis of 2,5-Disubstituted-1,3,4-oxadiazole Analogs as Novel Anticancer and Antimicrobial Agents

, 11(4): 413 - 419

Mohamed Jawed Ahsan, Jyotika Sharma, Sandeep Bhatia, Pramod Kumar Goyal, Kailash Shankhala and Mukand Didel


DOI: 10.2174/1570180810666131113211647



QSAR Study of H1N1 Neuraminidase Inhibitors from Influenza a Virus

, 11(4): 420 - 427

Apilak Worachartcheewan, Chanin Nantasenamat, Chartchalerm Isarankura-Na-Ayudhya and Virapong Prachayasittikul


DOI: 10.2174/15701808113106660085



In-Vitro Antiproliferative Activity of New Tetrahydroisoquinolines (THIQs) on Ishikawa Cells and their 3D Pharmacophore Models

, 11(4): 428 - 436

Suresh Kumar V. K. Eyunni, Madhavi Gangapuram and Kinfe K. Redda


DOI: 10.2174/1570180811666131203002502



Synthesis, In Vitro Activity and Rationalisation of a Series of Dialkyl Esters of 5-Aminosulfonylisophthanoate as Potential Estrone Sulfatase (ES) Inhibitors

, 11(4): 437 - 443

Sabbir Ahmed and Chirag K. Patel


DOI: 10.2174/15701808113106660081



Design and Synthesis of Novel 2- Substituted Benzothiazole Compounds as PTP1B Inhibitors

, 11(4): 444 - 453

Arun P. Chandrasekharappa, Sangamesh E. Badiger, Pramod K. Dubey, Sunil K. Panigrahi and Sekhar Reddy VVV. Manukonda


DOI: 10.2174/15701808113106660076



Diverse Models for the Prediction of Dual mTOR and PI3Kα Inhibitory Activities of Substituted 4-morpholinopyrrolopyrimidines

, 11(4): 454 - 473

Monika Gupta and A. K. Madan


DOI: 10.2174/15701808113106660089



Synthesis, Molecular Docking and In Vitro Antimicrobial Studies of Novel Pyrazole Analogues of Curcumin

, 11(4): 474 - 483

Dileep Kumar, Harish B. G., Mayank Gangwar, Manish Kumar, Dharmendra Kumar, Ragini Tilak, Gopal Nath, Ashok Kumar and Sushil Kumar Singh


DOI: 10.2174/15701808113106660087



Improved Synthesis of Antiviral Drug Valacyclovir Hydrochloride

, 11(4): 484 - 487

Keshava Navin Kumar Reddy, Murugulla Adharvana Chari, Mayur. D. Khunt, B. Ramachandra Reddy, Vurimidi Himabindu and Ghanta Mahesh Reddy


DOI: 10.2174/15701808113106660090



Synthesis and Evaluation of Anticonvulsant Activities of Triazole- Incorporated Benzothiazoles

, 11(4): 488 - 494

Ming-Xia Song, Hong Zeng, Xian-Qing Deng and Zhe-Shan Quan


DOI: 10.2174/15701808113106660093



Improvement of Generic Sevoflurane by a New Production Process

, 11(4): 495 - 501

Tomo Hayase, Shigekazu Sugino, Shun-suke Tachibana, Naoyuki Hirata and Michiaki Yamakage


DOI: 10.2174/1570180810666131113211447



The Study of the Biological Activity of Amino-Substituted Benzofuroxans

, 11(4): 502 - 512

Elena A. Chugunova, Alexandra D. Voloshina, Rezeda E. Mukhamatdinova, Igor V. Serkov, Alexey N. Proshin, Elmira M. Gibadullina, Alexander R. Burilov, Natalia V. Kulik, Vladimir V. Zobov, Dmitry B. Krivolapov, Alexey B. Dobrynin and Regis Goumont


DOI: 10.2174/1570180810666131122010403



Computer-Aided Perspective for the Design of Flexible HIV Non- Nucleoside Reverse Transcriptase Inhibitors (NNRTIs): de-novo Drug Design, Virtual Screening and Molecular Dynamics Simulations

, 11(4): 513 - 524

Suri Moonsamy and Mahmoud E. S. Soliman


DOI: 10.2174/15701808113109990048




Editor-in-Chief

K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)

Biography
View Full Editorial Board

Journal History

Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
Scopus CiteScore Metrics: 1.05

Advertisement

How to write and publish your papers in high impact journalsCovid Resource Center

Related Journals

Related eBooks

eBooks Catalog