Letters in Drug Design & Discovery, Volume 11 - Number 3

Graphical Abstracts

, 11(3): i - vii

DOI: 10.2174/157018081103140203152259

Molecular Modeling and Docking Application to Evaluate Cruzain Inhibitory Activity by Chalcones and Hydrazides

, 11(3): 249 - 255

Drielli Gomes Vital, Marco Arribas and Gustavo Henrique Goulart Trossini

DOI: 10.2174/15701808113106660082

Synthesis and Anti-Proliferative Activity of New Biphenyle-Benzylidenethiazolidine- 2,4-dione Bis-Adducts Containing Various Heterocyclic Cores

, 11(3): 256 - 264

Maxime Meyer, Sandra Kuntz, Isabelle Grillier-Vuissoz, Helene Martin, Lysiane Richert, Stephane Flament, Yves Chapleur and Michel Boisbrun

DOI: 10.2174/15701808113106660080

Prediction of the Estrogen Receptor Binding Affinity for both hERα and hERβ by QSAR Approaches

, 11(3): 265 - 278

Changliang Deng, Xuanxuan Chen, Hongying Lu, Xin Yang, Feng Luan and Maria Natalia Dias Soeiro Cordeiro

DOI: 10.2174/15701808113109990067

Synthesis of Sulfur Containing Colchicine Derivatives and their Biological Evaluation as Cytotoxic Agents

, 11(3): 279 - 289

Joanna Kurek, Wladyslaw Boczon, Krzysztof Myszkowski, Marek Murias, Teresa Borowiak and Irena Wolska

DOI: 10.2174/15701808113106660086

Synthesis, Characterization, Antimycobacterial and Anticancer Evaluation of New 1,2,4-Triazole Derivatives

, 11(3): 290 - 296

G. Cihan-Ustundag, B. Simsek, E. Ilhan and G. Capan

DOI: 10.2174/157018081131000074

Triazole-linked Chalcone and Flavone Hybrid Compounds Based on AZT Exhibiting In Vitro Anti-Cancer Activity

, 11(3): 297 - 303

Nguyen Van Minh, Nguyen Le Anh, Do Thi Thao and Tran Khac Vu

DOI: 10.2174/157018081131000073

Synthesis, Evaluation and Molecular Docking Studies of 1,3,4-oxadiazole- 2-thiol Incorporating Fatty Acid Moiety as Antitumor and Antimicrobial Agents

, 11(3): 304 - 315

Fatma Salah El-Din Mohamed, Ahmed Ismail Hashem, Randa Helmy Swellem and Galal Abd El-Moaen Mohamed Nawwar

DOI: 10.2174/157018081131000072

Pharmacophore and 3D QSAR Study of TGFβ Inhibitors

, 11(3): 316 - 330

Mohamed Asraf Vazhapully, D. Vinod and N.H. Zeinul Hukuman

DOI: 10.2174/157018081131000071

Design and Synthesis of New Dual Binding Site Cholinesterase Inhibitors: in vitro Inhibition Studies with in silico Docking

, 11(3): 331 - 338

Muhammad Yar, Marek Bajda, Rana Atif Mehmood, Lala Rukh Sidra, Nisar Ullah, Lubna Shahzadi, Muhammad Ashraf, Tayaba Ismail, Sohail Anjum Shahzad, Zulfiqar Ali Khan, Syed Ali Raza Naqvi and Nasir Mahmood

DOI: 10.2174/15701808113106660078

A Combination of Pharmacophore and In silico Approaches for Identification of Potential Transthyretin Amyloidosis Inhibitors

, 11(3): 339 - 348

Zheng-Li Zhou, Hsuan-Liang Liu, Josephine W. Wu, Cheng-Wen Tsao, Wei-Hsi Chen, Kung-Tien Liu and Yih Ho

DOI: 10.2174/15701808113106660077

Synthesis, Characterization and Structure Activity Relationship Studies of Benzo[b]thiophene Derivatives as Promising Class of Antimicrobial Agents

, 11(3): 349 - 354

H.B. Ghodasara, R.G. Vaghasiya, V.K. Gothaliya and V.H. Shah

DOI: 10.2174/15701808113106660091

Synthesis and In Vitro Evaluation of Some Hydrazone Derivatives as Potential Antibacterial Agents

, 11(3): 355 - 362

Zafer Asim Kaplancikli, Mehlika Dilek Altintop, Ahmet Ozdemir, Gulhan Turan-Zitouni, Gamze Goger and Fatih Demirci

DOI: 10.2174/15701808113109990030

Identification of Interfacial Residues Involved in Hepcidin-Ferroportin Interaction

, 11(3): 363 - 374

Prasoon Kumar Thakur, Amresh Prakash, Parvez Khan, Robert E. Fleming, Abdul Waheed, Faizan Ahmad and Md. Imtaiyaz Hassan

DOI: 10.2174/15701808113106660088

Synthesis and Biological Evaluation of Novel N-[(7-pyridin-4-yl-2, 3- dihydro-benzofuran-2-yl) Methyl]-(4-methyl-1, 2, 3-thiadiazole-5-yl) Formamide as a Potent Immunosuppressant Agent

, 11(3): 375 - 379

Chen Fan, Yubin Wang, Peng Lu, Xiaojian Xue and Jinxiong She

DOI: 10.2174/15701808113106660084

Synthesis and Ultraviolet Absorption Characteristics of Chiral 3- arylidenenopinones from β-pinene

, 11(3): 380 - 386

Xu Xu, Yi-Qin Yang, Hai-Jun Xu, Lan Lan and Shi-Fa Wang

DOI: 10.2174/15701808113106660095

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