Contents

Letters in Drug Design & Discovery, Volume 10 - Number 9

GRAPHICAL ABSTRACTS

, 10(9): i - v


DOI: 10.2174/15701808113100990001




The Identification of the SIRT1 Activator SRT2104 as a Clinical Candidate

, 10(9): 793 - 797

Pui Yee Ng, Jean E. Bemis, Jeremy S. Disch, Chi B. Vu, Christopher J. Oalmann, Amy V. Lynch, David P. Carney, Thomas V. Riera, Jeffrey Song, Jesse J. Smith, Siva Lavu, Angela Tornblom, Meghan Duncan, Marie Yeager, Kristina Kriksciukaite, Akanksha Gupta, Vipin Suri, Peter J. Elliot, Jill C. Milne, Joseph J. Nunes, Michael R. Jirousek, George P. Vlasuk, James L. Ellis and Robert B. Perni


DOI: 10.2174/15701808113100990021




Synthesis, Antimicrobial Activities and Molecular Docking Studies of Novel 6-Hydroxybenzofuran-3(2H)-one Based 2,4-Disubstituted 1,3- Thiazoles

, 10(9): 798 - 807

Krzysztof Z. La czkowski, Konrad Misiura, Anna Biernasiuk, Anna Malm, Agata Siwek and Tomasz Plech


DOI: 10.2174/15701808113109990010




Pharmacophore Modeling and 3D QSAR Studies of Novel Human Carbonic Anhydrase IX Inhibitors

, 10(9): 808 - 816

Kalyan K. Sethi and Saurabh M. Verma


DOI: 10.2174/15701808113100990026




Synthesis and Biological Evaluation of Atorvastatin Derivatives as Novel HMG-CoA Reductase Inhibitors

, 10(9): 817 - 822

Jiayi Tong, Naxin Wang and Hua Xiao


DOI: 10.2174/15701808113106660020




3D-QSAR and Docking Studies of N-hydroxy 1,8-naphthyridine 2-one Analogs as Ribonuclease H Inhibitors

, 10(9): 823 - 835

Brijesh Patel, Saurabh M. Verma and Kalyan K. Sethi


DOI: 10.2174/15701808113109990059




QSAR of Pyrazole Oxadiazole Derivatives as s1p1 Agonists Studied by CoMFA, CoMSIA and Docking

, 10(9): 836 - 852

Baokun Li, Tingjun Hou, Chongqian Zhang and Youyong Li


DOI: 10.2174/15701808113109990001




Computational Simulations as Preformulation Perspective for the Delivery of NSAIDs Using β-Cyclodextrin

, 10(9): 853 - 858

Amrish Kumar, Dinesh Kumar Mishra, Manoj Gautam and Suresh Thareja


DOI: 10.2174/15701808113109990016




Transition Metal Complexes of 8-Aminoquinoline-5-Substituted Uracils with Antioxidative and Cytotoxic Activities

, 10(9): 859 - 864

Ratchanok Pingaew, Apilak Worachartcheewan, Veda Prachayasittikul, Supaluk Prachayasittikul, Somsak Ruchirawat and Virapong Prachayasittikul


DOI: 10.2174/15701808113109990004




Studies on Synthesis of Novel Triazolalkyl Tagged Trifluoromethyl Substituted Pyrimidine Derivatives and their Evaluation for Cytotoxic Activity

, 10(9): 865 - 871

Punna Nagender, Gannarapu Malla Reddy, Royya Naresh Kumar, Anugu Chandrashekar Reddy, Loka Reddy Velatooru, Rajesh Pamanji, Janapala Venkateswara Rao and Banda Narsaiah


DOI: 10.2174/1570180811310090010




Design, Synthesis and In-Vitro Cytotoxicity of Novel Platinum (II) Complexes with Phthalate as the Leaving Group

, 10(9): 872 - 878

Rajiv Sharma, Ravindra K. Rawal, Manav Malhotra, Tripti Gaba, A. K. Sharma and T. R. Bhardwaj


DOI: 10.2174/15701808113109990018




Synthesis and Biological Evaluation of Novel β-Carboline Derivatives as Antiproliferative Agents

, 10(9): 879 - 885

Jing Chen, Wenting Du, Xuefen Tao, Jiawei Huang, Yuliang Song and Huazhou Ying


DOI: 10.2174/15701808113109990009




Synthesis and Antiproliferative Activity of New Polyoxo 2-Benzyl-2,3- dihydrobenzofurans and Their Related Compounds

, 10(9): 886 - 894

Ping Qi, Jianhua Jiang, Huan Qi, Yinghua Jin, Qirong Shen, Yingliang Wu, Hongrui Song and Weige Zhang


DOI: 10.2174/15701808113109990011




Synthesis, Evaluation of Analgesic and Gastric Ulcerogenic Activities and the Metabolites in Rat Plasma of Hydantoin Ibuprofen Conjugates

, 10(9): 895 - 899

Cuiying Mao, Ping Yang, Yongsheng Wang, Lan Qiao, Bing Chen, Shihan Wang, Yang Xu and Haibin Lu


DOI: 10.2174/15701808113109990005




Synthesis and Anticonvulsant Activity of Some Non-Classical Dihydropyridine Like Structures

, 10(9): 900 - 905

Mohammad Sharifzadeh, Hamid Reza khademi, Ali Almasirad, Zahra rezayan, Mohsen Rezayan Ghayahbashi and Mohsen Amini


DOI: 10.2174/15701808113109990015




Synthesis and in vivo Antihyperlipidemic Potential of Novel Substituted Thieno[3,2-d]pyrimidines

, 10(9): 906 - 915

Riyaj Shaukat Tamboli, Rakesh Devidas Amrutkar, Kishor Sanchlal Jain and Muthu Kumaradoss Kathiravan


DOI: 10.2174/15701808113109990019




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