Contents

Letters in Drug Design & Discovery, Volume 10 - Number 8

GRAPHICAL ABSTRACTS

, 10(8): i - v


DOI: 10.2174/1570180811310080001




Titanocene Y - Transport and Targeting of an Anticancer Drug Candidate

, 10(8): 675 - 682

Grainne Lally, Anthony Deally, Frauke Hackenberg, Susan J. Quinn and Matthias Tacke


DOI: 10.2174/15701808113100890027




Cytotoxic Effects of the Monomer and Dimer of 3, 4-seco-ent-kaurene from Croton Micans and their Interaction with Antitumoral Drugs on Cellular Line of Human Prostate Cancer

, 10(8): 683 - 688

Jennire Vivas, Felipe Sojo, Katiuska Chavez, Alírica I. Suarez and Francisco Arvelo


DOI: 10.2174/15701808113109990021




Synthesis and Biological Evaluation of 1, 3-Dihydroxyxanthone Mannich Base Derivatives as Potential Antitumor Agents

, 10(8): 689 - 698

Wenli Lan, Jingchen Wei, Jiangke Qin, Zhengmin Yang, Guifa Su and Zhikai Dai


DOI: 10.2174/15701808113100890029




Synthesis and Cytotoxic Evaluation for Some New Dihydropyrimidinone Derivatives for Anticancer Activity

, 10(8): 699 - 705

Onteddu. Surendranatha Reddy, Ch. Venkata Suryanarayana, N. Sharmila, G. V. Ramana, V. Anuradha and B. Hari Babu


DOI: 10.2174/15701808113109990007




Bifunctional Anti-HIV/TB Inhibitors: Perspective from In-Silico Design and Molecular Dynamics Simulations

, 10(8): 706 - 712

Lauren Blake and Mahmoud E. S. Soliman


DOI: 10.2174/15701808113109990023




Synthesis, Biological and Computational Evaluation of Novel Oxindole Derivatives as Inhibitors of Src Family Kinases

, 10(8): 713 - 718

Zühal Kilic-Kurt, Arzu Onay-Besikci and Sureyya Olgen


DOI: 10.2174/15701808113109070023




Pharmacophore Based 3D-QSAR Modeling and Molecular Docking of Leucettines as Potent Dyrk1A Inhibitors

, 10(8): 719 - 726

Anu Bahl, Prashant Joshi, Sandip B. Bharate and Harish Chopra


DOI: 10.2174/15701808113100890024




Synthesis and Biological Evaluations of 3-Benzothiazol-2-yl Coumarin Derivatives as MEK1 Inhibitors

, 10(8): 727 - 732

Chao Wang, Fengrong Xu, Yan Niu, Yun Wu, Jing Sun, Yihong Peng, Lei Liang and Ping Xu


DOI: 10.2174/15701808113109990012




Optimized Synthesis of Etidronate

, 10(8): 733 - 737

Rita Kovacs, David Illes Nagy, Alajos Grün, Gyorgy Tibor Balogh, Sandor Garadnay, Istvan Greiner and Gyorgy Keglevich


DOI: 10.2174/15701808113109990026




Synthesis of Allosamidin Analogue Di-N-acetyl-β-chitobiosyl N-Glycoaminooxazoline

, 10(8): 738 - 740

Gangliang Huang, Shuangquan Shu and Fei Cheng


DOI: 10.2174/15701808113109990008




Synthesis and In Vivo Antimalarial Activity of Novel Derivatives of 6- Mercaptopurine

, 10(8): 741 - 747

Roberta Reis Soares, Roberta C. N. R. Corrales, Fernanda Valerio Lopes, Marcio Jose M. Alves, Adilson David Da Silva and Clarice Abramo


DOI: 10.2174/15701808113109990017




Antibacterial Activity and Structure-Activity Relationship Studies of 4- aryl/alkyl-1-(diphenylacetyl)thiosemicarbazides

, 10(8): 748 - 757

Edyta Kusmierz, Agata Siwek, Urszula Kosikowska, Anna Malm, Joanna Stefanska, Katarzyna Dzitko and Monika Wujec


DOI: 10.2174/15701808113100890028




Evaluation of the Antimicrobial Activity of Some 4H-Pyrano[3,2-h]- quinoline,7H-Pyrimido[4',5':6,5]pyrano[3,2-h]quinoline Derivatives

, 10(8): 758 - 775

Hany M. Mohamed, Ibrahim A. Radini, Abdullah M. Al-Ghamdi and Ahmed M. El-Agrody


DOI: 10.2174/15701808113109990002




Synthesis of 4-(5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl)-6-(substituted phenyl)pyrimidin-2-ol Analogues as Anti-Inflammatory and Analgesic Agents

, 10(8): 776 - 782

Muhammad Jahangir Alam, Mohamed Jawed Ahsan, Ozair Alam and Suroor Ahmad Khan


DOI: 10.2174/15701808113100890022




Synthesis and Evaluation of In Vivo Anticonvulsant Activity of 2,5- Disubstituted-1,3,4-Oxadiazole Derivatives

, 10(8): 783 - 791

Kikkeri P. Harish, Kikkeri N. Mohana, Lingappa Mallesha, B. Veeresh, B. Madhava Reddy and Nagula Naresh Kumar


DOI: 10.2174/15701808113109990020




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