Contents

Letters in Drug Design & Discovery, Volume 10 - Number 5

Graphical Abstract

Graphical Abstracts

, 10(5): i - v


DOI: 10.2174/1570180811310050001




The Activity of Titanocene T Against Xenografted Caki-1 Tumors

, 10(5): 375 - 381

Wolfgang Walther, Iduna Fichtner, Anthony Deally, Megan Hogan and Matthias Tacke


DOI: 10.2174/1570180811310050002




Synthesis and Biological Evaluation of 3-Chloro-4-(indol-3-yl)-2,5- pyrroledione Derivatives as Antitumor Agents

, 10(5): 382 - 389

Yuchen Lin and Jing Chen


DOI: 10.2174/1570180811310050003




The Venom of the Centipede Scolopendra subspinipes mutilans Inhibits the Growth of Myelogenous Leukemia Cell Lines

, 10(5): 390 - 395

Shiyan Xu, Fan Zhang, Hengyun Wang, Yu Liu, Dan Li, Zhe Wu and Zhonghua Liu


DOI: 10.2174/1570180811310050004




Further Insights in 5-phenyl-2-[2-(1-piperidinylcarbonyl) Phenyl]-2,3- dihydro-1H-pyrrolo[1,2-c]imidazol-1-ones, a Recently Disclosed Class of Neuropeptide S Antagonists

, 10(5): 396 - 401

Gabriele Costantino, Marco Mor, Chiara Pecchini, Gian Paolo Vallerini, Elisa Della Turca, Fabrizio Micheli, Angela Worby, Romano Di Fabio, Angelo Giacometti, Adelheid Roth, Emilio Merlo-Pich, Matteo Biagetti, Giorgio Bonanomi, Dino Montanari, Luca Tarsi, Federica Tonelli, Raffaele Longhi and Anna Maria Capelli


DOI: 10.2174/1570180811310050005




Preparation and Cytotoxic Activities of Fatty Acid Derivatives of 20(S)- Protopanaxatriol

, 10(5): 402 - 409

Nan-Nan Qiu, Jie Hu, Jin-Ping Liu, Fang Wang and Ping-Ya Li


DOI: 10.2174/1570180811310050006




Glyoxalase 1 and 2 Enzyme Inhibitory Activity of 6-Sulfamoylsaccharin and Sulfocoumarin Derivates

, 10(5): 410 - 414

Marina Makrecka, Raivis Zalubovskis, Edijs Vavers, Jekaterina Ivanova, Aiga Grandane and Maija Dambrova


DOI: 10.2174/1570180811310050007




Aldose Reductase Inhibitory Potential of Several Thiazolyl-thiazolidine- 2,4-Diones

, 10(5): 415 - 419

Net Das-Evcimen, Mutlu Sarıkaya, A. Selen Gurkan-Alp and Oya Bozdag-Dundar


DOI: 10.2174/1570180811310050008




Design, Synthesis and Evaluation of Quinoline-based Small Molecule Inhibitor of STAT3

, 10(5): 420 - 426

Zhi-Bing Shi, Lei Zhang, Zheng-Yang Bin, Xiang-Rong Cao, Zhu-Nan Gong and Jian-Xin Li


DOI: 10.2174/1570180811310050009




QSAR Studies of Tetranortriterpenoid: An Analysis Through CoMFA and CPSA Parameters

, 10(5): 427 - 436

K. Arvind, K. Anand Solomon and S.S. Rajan


DOI: 10.2174/1570180811310050010




Purification and Biological Evaluation of Some Bioactive Metabolomics as Antimicrobial Agent

, 10(5): 437 - 443

Ramar Perumal Samy, Gautam Sethi and Vincent T.K Chow


DOI: 10.2174/1570180811310050011




Design, Synthesis, Crystal Structure, and Antimicrobial Evaluation of Novel Pyrazolyl-1,3,5-oxadiazoles, Pyrazolyl-1,2,4-triazoles and their Related Thioglycosides

, 10(5): 444 - 452

Nora M. A. El-Ebiary, Emad M. El-Telbani, Randa H. Swellem, Ibrahim F. Zeid and Galal A. M. Nawwar


DOI: 10.2174/1570180811310050012




Synthesis and Biological Evaluation of some Amide Derivatives Bearing Benzothiazole and Piperidine Moieties as Antimicrobial Agents

, 10(5): 453 - 461

Mehlika Dilek Altintop, Ahmet Ozdemir, Zafer Asim Kaplancikli, Gulhan Turan-Zitouni, Gokalp Iscan and Gulsen Akalin Ciftci


DOI: 10.2174/1570180811310050013




Synthesis and Biological Evaluation of Piperazinyl-2-(Benzo)thiophen/- furan-2-yl-acetonitriles as Strecker Reaction Products

, 10(5): 462 - 470

Rahul V. Patel, Jigar K. Patel, Shivraj H. Nile and Se Won Park


DOI: 10.2174/1570180811310050014




Antimycobacterial Activity: Synthesis and Biological Evaluation of Novel Substituted (3E,5E)-3,5-diarylidene-1-phenethylpiperidine-4-one Derivatives

, 10(5): 471 - 476

Mohamed Ashraf Ali, Venu Sanjeevi Lakshmipathi, Farzana Beevi, Raju Suresh Kumar, Rusli Ismail, Tan Soo Choon, Ang Chee Wei, Yeong Keng Yoon and Alireza Basiri


DOI: 10.2174/1570180811310050015




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