Contents
Letters in Drug Design & Discovery, Volume 10 - Number 5
Graphical Abstract
The Activity of Titanocene T Against Xenografted Caki-1 Tumors
, 10(5): 375 - 381Wolfgang Walther, Iduna Fichtner, Anthony Deally, Megan Hogan and Matthias Tacke
DOI: 10.2174/1570180811310050002
The Venom of the Centipede Scolopendra subspinipes mutilans Inhibits the Growth of Myelogenous Leukemia Cell Lines
, 10(5): 390 - 395Shiyan Xu, Fan Zhang, Hengyun Wang, Yu Liu, Dan Li, Zhe Wu and Zhonghua Liu
DOI: 10.2174/1570180811310050004
Further Insights in 5-phenyl-2-[2-(1-piperidinylcarbonyl) Phenyl]-2,3- dihydro-1H-pyrrolo[1,2-c]imidazol-1-ones, a Recently Disclosed Class of Neuropeptide S Antagonists
, 10(5): 396 - 401Gabriele Costantino, Marco Mor, Chiara Pecchini, Gian Paolo Vallerini, Elisa Della Turca, Fabrizio Micheli, Angela Worby, Romano Di Fabio, Angelo Giacometti, Adelheid Roth, Emilio Merlo-Pich, Matteo Biagetti, Giorgio Bonanomi, Dino Montanari, Luca Tarsi, Federica Tonelli, Raffaele Longhi and Anna Maria Capelli
DOI: 10.2174/1570180811310050005
Preparation and Cytotoxic Activities of Fatty Acid Derivatives of 20(S)- Protopanaxatriol
, 10(5): 402 - 409Nan-Nan Qiu, Jie Hu, Jin-Ping Liu, Fang Wang and Ping-Ya Li
DOI: 10.2174/1570180811310050006
Glyoxalase 1 and 2 Enzyme Inhibitory Activity of 6-Sulfamoylsaccharin and Sulfocoumarin Derivates
, 10(5): 410 - 414Marina Makrecka, Raivis Zalubovskis, Edijs Vavers, Jekaterina Ivanova, Aiga Grandane and Maija Dambrova
DOI: 10.2174/1570180811310050007
Aldose Reductase Inhibitory Potential of Several Thiazolyl-thiazolidine- 2,4-Diones
, 10(5): 415 - 419Net Das-Evcimen, Mutlu Sarıkaya, A. Selen Gurkan-Alp and Oya Bozdag-Dundar
DOI: 10.2174/1570180811310050008
Design, Synthesis and Evaluation of Quinoline-based Small Molecule Inhibitor of STAT3
, 10(5): 420 - 426Zhi-Bing Shi, Lei Zhang, Zheng-Yang Bin, Xiang-Rong Cao, Zhu-Nan Gong and Jian-Xin Li
DOI: 10.2174/1570180811310050009
QSAR Studies of Tetranortriterpenoid: An Analysis Through CoMFA and CPSA Parameters
, 10(5): 427 - 436K. Arvind, K. Anand Solomon and S.S. Rajan
DOI: 10.2174/1570180811310050010
Purification and Biological Evaluation of Some Bioactive Metabolomics as Antimicrobial Agent
, 10(5): 437 - 443Ramar Perumal Samy, Gautam Sethi and Vincent T.K Chow
DOI: 10.2174/1570180811310050011
Design, Synthesis, Crystal Structure, and Antimicrobial Evaluation of Novel Pyrazolyl-1,3,5-oxadiazoles, Pyrazolyl-1,2,4-triazoles and their Related Thioglycosides
, 10(5): 444 - 452Nora M. A. El-Ebiary, Emad M. El-Telbani, Randa H. Swellem, Ibrahim F. Zeid and Galal A. M. Nawwar
DOI: 10.2174/1570180811310050012
Synthesis and Biological Evaluation of some Amide Derivatives Bearing Benzothiazole and Piperidine Moieties as Antimicrobial Agents
, 10(5): 453 - 461Mehlika Dilek Altintop, Ahmet Ozdemir, Zafer Asim Kaplancikli, Gulhan Turan-Zitouni, Gokalp Iscan and Gulsen Akalin Ciftci
DOI: 10.2174/1570180811310050013
Synthesis and Biological Evaluation of Piperazinyl-2-(Benzo)thiophen/- furan-2-yl-acetonitriles as Strecker Reaction Products
, 10(5): 462 - 470Rahul V. Patel, Jigar K. Patel, Shivraj H. Nile and Se Won Park
DOI: 10.2174/1570180811310050014
Antimycobacterial Activity: Synthesis and Biological Evaluation of Novel Substituted (3E,5E)-3,5-diarylidene-1-phenethylpiperidine-4-one Derivatives
, 10(5): 471 - 476Mohamed Ashraf Ali, Venu Sanjeevi Lakshmipathi, Farzana Beevi, Raju Suresh Kumar, Rusli Ismail, Tan Soo Choon, Ang Chee Wei, Yeong Keng Yoon and Alireza Basiri
DOI: 10.2174/1570180811310050015
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