Letters in Drug Design & Discovery
Volume 18, 12 Issues, 2021
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access
Contents
Letters in Drug Design & Discovery, Volume 10 - Number 5
Graphical Abstract
The Activity of Titanocene T Against Xenografted Caki-1 Tumors
, 10(5): 375 - 381Wolfgang Walther, Iduna Fichtner, Anthony Deally, Megan Hogan and Matthias Tacke
DOI: 10.2174/1570180811310050002
The Venom of the Centipede Scolopendra subspinipes mutilans Inhibits the Growth of Myelogenous Leukemia Cell Lines
, 10(5): 390 - 395Shiyan Xu, Fan Zhang, Hengyun Wang, Yu Liu, Dan Li, Zhe Wu and Zhonghua Liu
DOI: 10.2174/1570180811310050004
Further Insights in 5-phenyl-2-[2-(1-piperidinylcarbonyl) Phenyl]-2,3- dihydro-1H-pyrrolo[1,2-c]imidazol-1-ones, a Recently Disclosed Class of Neuropeptide S Antagonists
, 10(5): 396 - 401Gabriele Costantino, Marco Mor, Chiara Pecchini, Gian Paolo Vallerini, Elisa Della Turca, Fabrizio Micheli, Angela Worby, Romano Di Fabio, Angelo Giacometti, Adelheid Roth, Emilio Merlo-Pich, Matteo Biagetti, Giorgio Bonanomi, Dino Montanari, Luca Tarsi, Federica Tonelli, Raffaele Longhi and Anna Maria Capelli
DOI: 10.2174/1570180811310050005
Preparation and Cytotoxic Activities of Fatty Acid Derivatives of 20(S)- Protopanaxatriol
, 10(5): 402 - 409Nan-Nan Qiu, Jie Hu, Jin-Ping Liu, Fang Wang and Ping-Ya Li
DOI: 10.2174/1570180811310050006
Glyoxalase 1 and 2 Enzyme Inhibitory Activity of 6-Sulfamoylsaccharin and Sulfocoumarin Derivates
, 10(5): 410 - 414Marina Makrecka, Raivis Zalubovskis, Edijs Vavers, Jekaterina Ivanova, Aiga Grandane and Maija Dambrova
DOI: 10.2174/1570180811310050007
Aldose Reductase Inhibitory Potential of Several Thiazolyl-thiazolidine- 2,4-Diones
, 10(5): 415 - 419Net Das-Evcimen, Mutlu Sarıkaya, A. Selen Gurkan-Alp and Oya Bozdag-Dundar
DOI: 10.2174/1570180811310050008
Design, Synthesis and Evaluation of Quinoline-based Small Molecule Inhibitor of STAT3
, 10(5): 420 - 426Zhi-Bing Shi, Lei Zhang, Zheng-Yang Bin, Xiang-Rong Cao, Zhu-Nan Gong and Jian-Xin Li
DOI: 10.2174/1570180811310050009
QSAR Studies of Tetranortriterpenoid: An Analysis Through CoMFA and CPSA Parameters
, 10(5): 427 - 436K. Arvind, K. Anand Solomon and S.S. Rajan
DOI: 10.2174/1570180811310050010
Purification and Biological Evaluation of Some Bioactive Metabolomics as Antimicrobial Agent
, 10(5): 437 - 443Ramar Perumal Samy, Gautam Sethi and Vincent T.K Chow
DOI: 10.2174/1570180811310050011
Design, Synthesis, Crystal Structure, and Antimicrobial Evaluation of Novel Pyrazolyl-1,3,5-oxadiazoles, Pyrazolyl-1,2,4-triazoles and their Related Thioglycosides
, 10(5): 444 - 452Nora M. A. El-Ebiary, Emad M. El-Telbani, Randa H. Swellem, Ibrahim F. Zeid and Galal A. M. Nawwar
DOI: 10.2174/1570180811310050012
Synthesis and Biological Evaluation of some Amide Derivatives Bearing Benzothiazole and Piperidine Moieties as Antimicrobial Agents
, 10(5): 453 - 461Mehlika Dilek Altintop, Ahmet Ozdemir, Zafer Asim Kaplancikli, Gulhan Turan-Zitouni, Gokalp Iscan and Gulsen Akalin Ciftci
DOI: 10.2174/1570180811310050013
Synthesis and Biological Evaluation of Piperazinyl-2-(Benzo)thiophen/- furan-2-yl-acetonitriles as Strecker Reaction Products
, 10(5): 462 - 470Rahul V. Patel, Jigar K. Patel, Shivraj H. Nile and Se Won Park
DOI: 10.2174/1570180811310050014
Antimycobacterial Activity: Synthesis and Biological Evaluation of Novel Substituted (3E,5E)-3,5-diarylidene-1-phenethylpiperidine-4-one Derivatives
, 10(5): 471 - 476Mohamed Ashraf Ali, Venu Sanjeevi Lakshmipathi, Farzana Beevi, Raju Suresh Kumar, Rusli Ismail, Tan Soo Choon, Ang Chee Wei, Yeong Keng Yoon and Alireza Basiri
DOI: 10.2174/1570180811310050015
Editor-in-Chief
K. Kuca
University of Hradec Kralove
Hradec Kralove
(Czech Republic)
Biography
University of Hradec Kralove
Hradec Kralove
Biography
Biography of K. Kuca
Kamil Kuca is working for several academic institutes (University of Hradec Kralove, Czech Republic; University Hospital Hradec Kralove, Czech republic; Florida International University, USA; Yangtze University, China; etc.). He is recently rector of the University of Hradec Kralove. He was also technology scout focused on biomedicine in the past. His research interests are toxicology, pharmacology, drug design, technology transfer, pharmacoeconomy, chemical and biological terrorism, etc. He was/is principal investigator on numerous national and international projects (EU, NATO, GACR, IGA MZ, MSMT etc.). He has published more than 350 IF research papers. He is working with several companies as a scientific consultant. He has lots of cooperators throughout the world (e.g. Korea, Croatia, United Arab Emirates, USA, France, Turkey, China, Singapore, Sweden, and Brazil). His Hindex is 36, number of citation in WoS is over 3000.
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Journal History
Letters in Drug Design & Discovery was introduced in 2004. Dr. Kamil Kuca serves as the Editor-in-Chief of the journal.
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