Contents

Letters in Drug Design & Discovery, Volume 10 - Number 2

Graphical Abstract

Graphical Abstracts

, 10(2): i - iv


DOI: 10.2174/157018013804725099




Antibacterial Activity and Structure-activity Relationship Studies of 4- substituted-5-(diphenylmethyl)-2,4-dihydro-3H-1,2,4-triazole-3-thiones

, 10(2): 95 - 101

Edyta Kusmierz, Agata Siwek, Urszula Kosikowska, Anna Malm, Joanna Stefanska, Katarzyna Dzitko and Monika Wujec


DOI: 10.2174/157018013804725198




Synthesis and Antibacterial Activity of Oxime Ester Derivatives from Dehydroabietic Acid

, 10(2): 102 - 110

Cui Yan-Jie, Rao Xiao-Ping, Shang Shi-Bin, Song Jie and Gao Yan-Qing


DOI: 10.2174/157018013804725071




Novel 2-pyrazolin-1-ylthiazoles as Potential Antimicrobial Agents

, 10(2): 111 - 118

Bakr Fathy Abdel-Wahab, Ashraf Sediek, Hanan Ahmed Mohamed and Ghada Elsayed Ahmed Awad


DOI: 10.2174/157018013804725143




Synthesis, Molecular Docking and In Vitro Antimicrobial Studies of New Hexahydroindazole Derivatives of Curcumin

, 10(2): 119 - 128

Dileep Kumar, Harish B.G, Mayank Gangwar, Manish Kumar, Dharmendra Kumar, RaginiTilak, Gopal Nath, Ashok kumar and Sushil Kumar Singh


DOI: 10.2174/157018013804725161




Combined Three Dimensional Quantitative Structure Activity Relationships (3D-QSAR) Modeling and Molecular Docking Studies on Naphthoquinone Analogs as Proteasome Inhibitors

, 10(2): 129 - 144

Guanhong Xu, Zhou Zhou and Fei Li


DOI: 10.2174/157018013804725125




Synthesis, Genotoxicity and UV-protective Activity of New Benzofuroxans Substituted by Aromatic Amines

, 10(2): 145 - 154

Elena Alexandrovna Chugunova, Marina Alexandrovna Sazykina, Elmira Mingaleevna Gibadullina, Alexander Romanovich Burilov, Ivan Sergeevich Sazykin, Vladimir Anatolevich Chistyakov, Rezeda Eduardovna Timasheva, Dmitry Borisovich Krivolapov and Regis Goumont


DOI: 10.2174/157018013804725080




Synthesis and Anti-HIV-Evaluation of Novel Andrographolide Derivatives

, 10(2): 155 - 163

Guolong Gu, Haiyan Lin, Yajuan Liu, Liumeng Yang, Yongtang Zheng, Bin Wang, Chunlei Tang, Hai Qian and Wenlong Huang


DOI: 10.2174/157018013804725107




Screening of Few Epoxides as mt-MAPK Inhibitor Preventing Granuloma Formation to Serve as Tubercular Antidote

, 10(2): 164 - 168

Abhishek Chowdhury, Paulomi Paul, Pankaj Chetia and Manabendra Dutta Choudhury


DOI: 10.2174/157018013804725189




Design and Synthesis of Novel Cannabinoid Ligands Based on a 1,2,3- triazole Scaffold

, 10(2): 169 - 172

Przemyslaw W. Szafranski, Karol Dyduch, Tomasz Kosciolek, Tomasz P. Wrobel, Maria Gomez-Canas, Maria Gomez-Ruiz, Javier Fernandez-Ruiz and Jacek Mlynarski


DOI: 10.2174/157018013804725134




Anticonvulsant Activity and 5-HT1A/5-HT7 Receptors Affinity of Piperazine Derivatives of 3,3-Diphenyl- and 3,3-Dimethyl-succinimides

, 10(2): 173 - 182

Jolanta Obniska, Iwona Chlebek, Krzysztof Kaminski, Andrzej J. Bojarski and Grzegorz Satala


DOI: 10.2174/157018013804725116




High-Efficiency Synthesis of N,N ’ -Diacetyl-β-Chitobiosyl Allosamizoline

, 10(2): 183 - 185

Hualiang Huang


DOI: 10.2174/157018013804725170




Synthesis and Antioxidant Activity of 1,2,4-Triazole linked Thieno[2,3- d]pyrimidine Derivatives

, 10(2): 186 - 193

Suresh Maddila, Avula S. Kumar, Sridevi Gorle, M. Singh, Palakondu Lavanya and S.B. Jonnalagadda


DOI: 10.2174/157018013804725152




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