Contents

Letters in Drug Design & Discovery, Volume 10 - Number 10

Graphical Abstracts:

, 10(10): i - vii


DOI: 10.2174/1570180811310100001




Synthesis and Antibacterial Activity of 4,5-disubstituted-1,2,4-triazole-3- thiones

, 10(10): 917 - 922

Tomasz Plech, Monika Wujec, Urszula Kosikowska and Anna Malm


DOI: 10.2174/15701808113109990082




Synthesis and Antibacterial Activity of Novel Chalcone Derivatives of Apocynin

, 10(10): 923 - 927

P. Janaki, B. Bhadraiah, P. Acharya Nagarjuna and N. J. P. Subhashini


DOI: 10.2174/15701808113109990081




Synthesis and Biological Evaluation of Halogenated 2-Arylimino-3-arythiazolidine- 4-ones Containing Benzoic Acid Fragments as Antibacterial Agents

, 10(10): 928 - 934

Jie Zhang, Likang Zheng, Huayong Liu, Dan Zhao, Di Qu and Shiqing Han


DOI: 10.2174/15701808113109990031




Design, Synthesis and Biological Evaluation of Novel Aminosaccharide Derivatives of Combretastatin A-4

, 10(10): 935 - 941

Yan Tang, Zhewei Tu, Jing Sun, Xiong Zhu, Kun Liu, Shuying He and Yungen Xu


DOI: 10.2174/15701808113109990024




Synthesis of pyridyl benzimidazoles encompassing 4-thiazolidinone derivatives as potential antimicrobial agents

, 10(10): 942 - 950

N C Desai, D D Pandya, G M Kotadiya and Priyanka Desai


DOI: 10.2174/15701808113109990029




Synthesis and Characterization of 1-carboxyphenothiazine Derivatives Bearing Nitrogen Mustard as Promising Class of Antitubercular Agents

, 10(10): 951 - 956

V.B. Kataria, M.J. Solanki, A.R. Trivedi and V.H. Shah


DOI: 10.2174/15701808113109990022




Design, Synthesis and Computational Studies of New Benzothiazole Substituted Quinazolines as Potential Antimicrobial Agents

, 10(10): 957 - 966

Amit B. Patel, Premlata Kumari, Suban K. Sahoo and Kishor H. Chikhalia


DOI: 10.2174/15701808113109990025




Design, Synthesis and Antimicrobial Activity of α-Aminophosphonates of Quinoline and their Molecular Docking Studies Against DNA Gyrase A

, 10(10): 967 - 976

Doddaga Srinivasulu, Muttana Vijaya Bhaskara Reddy, Donka Rajasekhar, Meriga Balaji and Chamarthi Nagaraju


DOI: 10.2174/15701808113109990035




Synthesis and Anti-Inflammatory Activity of Fused 1,2,4-triazolo-[3,4-b] [1,3,4]thiadiazole Derivatives of Phenothiazine

, 10(10): 977 - 983

S. Maddila, S. Gorle, M. Singh, P. Lavanya and S. B. Jonnalagadda


DOI: 10.2174/15701808113109990034




Synthesis and Evaluation of Vascular Endothelial Growth Factor Receptor-2 Inhibitory Activity of 6,7-Dimethoxycinnoline Derivatives

, 10(10): 984 - 988

Xingjun Yao, Hongfa Yang, Yanhui Wan, Li Bie, Xinrui Liu and Zhonghui Liu


DOI: 10.2174/15701808113109990027




Predicting Drug-Target Interactions of Nuclear Receptors Based on Molecular Descriptors Information

, 10(10): 989 - 994

Junxiang Wang, Weiming Yu, Zhibin Chen, Hengda Li and Zhenran Jiang


DOI: 10.2174/15701808113109100023




3D-QSAR Modeling Studies on Pyrrolopyridinone Derivatives as Inhibitors of Cdc7 Kinase

, 10(10): 995 - 1006

Xiangxiang Wu, Xin Zhu, Yimin Hou, Xuefen Wu and Huahui Zeng


DOI: 10.2174/15701808113109990039




Synthesis and Anthelmintic Evaluation of Novel Valerolactam- Benzimidazole Hybrids

, 10(10): 1007 - 1014

Beatriz Munguía, Pablo Mendina, Romina Espinosa, Andrea Lanz, Jenny Saldaña, María J. Andina, Ximena Ures, Andrés López, Eduardo Manta and Laura Domínguez


DOI: 10.2174/15701808113109990028




Biotin-Encoded and Fe3O4-Loaded Polymeric Nano Micelles: Preparation, Optimization and In Vitro Characterization

, 10(10): 1015 - 1023

Mohammad Hossein Ahmadi Azqhandi, Mohammad Reza Khanmohammadi, Bahman Vasheghani Farahani and Reza Najafipour


DOI: 10.2174/15701808113109990033




Synthesis and Anticonvulsant activity of Fluorinated Cyclic Enaminones

, 10(10): 1024 - 1031

Cosmas O. Okoro, John Apraku, Elisha O. Okoromoba and Olugbeminiyi O. Fadeyi


DOI: 10.2174/15701808113109990064




ACKNOWLEDGEMENTS TO REVIEWERS:

, 10(10): 1032


DOI: 10.2174/1570180811310100017




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