Contents

Letters in Drug Design & Discovery, Volume 10 - Number 1

Graphical Abstract

Graphical Abstracts

, 10(1): i - iv


DOI: 10.2174/157018081130901000i




Editorial

Editorial

, 10(1): 1

Atta-ur-Rahman


DOI: 10.2174/1570180811309010001




Search for Molecular Basis of Antifungal Activity of Thiosemicarbazide Derivatives: A Combined in vitro Antifungal and Enzymatic Studies with in Silico Docking

, 10(1): 2 - 10

Agata Siwek, Pawel Staczek, Aleksandra Strzelczyk and Joanna Stefanska


DOI: 10.2174/1570180811309010002




Boronic Acid Based Inhibitors of Autotaxin: Understanding their Biological Role in Terms of Quantitative Structure Activity Relationships (QSAR)

, 10(1): 11 - 18

Sotirios Katsamakas and Dimitra Hadjipavlou-Litina


DOI: 10.2174/1570180811309010011




Synthesis and Biological Study of Novel Indole-3-Imine-2-on Derivatives as Src Kinase and Glutathione S-Transferase Inhibitors

, 10(1): 19 - 26

Z. Kilic Kurt, D. Aydin, Y. G. Isgor, B. S. Isgor and S. Olgen


DOI: 10.2174/1570180811309010019




Synthesis and Anti-HIV Evaluation of Novel 1,2,4-triazole Derivatives as Potential Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors

, 10(1): 27 - 34

Zhenyu Li, Yuan Cao, Peng Zhan, Christophe Pannecouque, Jan Balzarini, Erik De Clercq and Xinyong Liu


DOI: 10.2174/1570180811309010027




Synthesis and Evaluation of Anticonvulsant Activity of Some N-[(4-Chlor- 2-methylphenoxy)ethyl]- and N-[(4-Chlor-2-methylphenoxy)acetyl]aminoalkanols

, 10(1): 35 - 43

Anna M. Waszkielewicz, Edward Szneler, Marek Cegla and Henryk Marona


DOI: 10.2174/1570180811309010035




Synthesis and Antimicrobial Activity of some Amide Derivatives Bearing Thiazole, Benzhydryl and Piperidine Moieties

, 10(1): 44 - 48

Ahmet Ozdemir


DOI: 10.2174/1570180811309010044




Protein Interaction Networks in Metallo Proteins and Docking Approaches of Metallic Compounds with TIMP and MMP in Control of MAPK Pathway

, 10(1): 49 - 55

Kaladhar Svgk Dowluru, Potladurthi Chandra Sai, Padmanabhuni Venkata Nageswara Rao, Amajala Krishna chaitanya, Duddukuri Govinda Rao, Vadlapudi Varahala Rao, Potladurthi Suresh, Erva Rajeswara Reddy, Sudabattula Vijaya kumar, Divyakolu Vinod Kumar and Gajjala Bhaskar Reddy


DOI: 10.2174/1570180811309010049




Evaluation of In-Vitro Multidrug Resistance Reversal Activities of HZ08 analogues with Improved Soluble Property

, 10(1): 56 - 60

Xiaobu Lan, Haiyan Lin, Chunlei Tang, Xiaoyun Zhu, Hai Qian, Wenlong Huang and Yunman Li


DOI: 10.2174/1570180811309010056




Synthesis and Antiproliferative Evaluation of Hybrids of Indolin-2-one and Quinazoline-4(3H)-one Linked via Imine Bond

, 10(1): 61 - 66

Wei-Yao Wu, Sheng-Li Cao, Bei-Bei Mao, Ji Liao, Zhong-Feng Li, Hao-Bin Song and Xingzhi Xu


DOI: 10.2174/1570180811309010061




Identification of Leads from Marine Seaweeds against Human β-tubulin

, 10(1): 67 - 74

Selvaa Kumar C, Nikhil Gadewal and Sudheer M.M. Mohammed


DOI: 10.2174/1570180811309010067




Design, Synthesis and Evaluation of Novel 2-piperidinyl Quinoline Chalcones/ Amines as Potential Antidepressant Agents

, 10(1): 75 - 85

Obaid Afzal, Sandhya Bawa, Suresh Kumar, Rajiv Kumar and Md Quamrul Hassan


DOI: 10.2174/1570180811309010075




Synthesis, Characterization, Antimicrobial Activity of Novel N-Substituted β-Hydroxy Amines and βHydroxy Ethers Contained Chiral Benzoxazine Fluoroquinolones

, 10(1): 86 - 93

B. Guruswamy and R. Arul


DOI: 10.2174/1570180811309010086




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