Contents

Letters in Drug Design & Discovery, Volume 1 - Number 2

Molecular Modulation of Muscarinic Antagonists. Synthesis and Pharmacological Profile of 2,2-diphenyl-2-ethylthioacetic and 3,3-diphenyl-3- ethylthiopropionic Acid Derivatives Characterized by a Dipeptide Spacer

, 1(2): 91 - 96

S. Scapecchi, C. Martelli, P. Angeli, C. Bellucci, M. Buccioni, S. Dei, F. Gualtieri, G. Marucci, R. Matucci and M. N. Romanelli


DOI: 10.2174/1570180043485527




Quaternary Heteroarenium Salts as the Competitive Inhibitors of the Brain Acetylcholinesterase

, 1(2): 97 - 100

Kamil Kuca, Jiri Cabal, Jiri Patocka and Vlastimil Dohnal


DOI: 10.2174/1570180043485509




Distinct Dimerization Between α-Lactalbumin and Lysozyme Exhibiting Novel Antimicrobial Activity against Gram-positive and Gram-negative Bacteria

, 1(2): 101 - 109

Hisham R. Ibrahim, Norihiko Taniyama and Takayoshi Aoki


DOI: 10.2174/1570180043485554




Challenges of Anthrax Drug Design: In Search of “Achilles heel” of Bacillus anthracis

, 1(2): 110 - 114

Chantal Guidi-Rontani


DOI: 10.2174/1570180043485590




Comparative Study of 3D-QSAR Techniques on Angiotensin II Receptor (AT1) Antagonists

, 1(2): 115 - 120

P. A. Datar, E. C. Coutinho and Sudha Srivastava


DOI: 10.2174/1570180043485536




Diverse Peptidyl Privileged Structures as Potent Somatostatin Receptor Ligands

, 1(2): 121 - 125

Alexander Pasternak, Yanping Pan, Ralph T. Mosley, Susan P. Rohrer, Elizabeth T. Birzin, James Schaeffer, Arthur A. Patchett and Lihu Yang


DOI: 10.2174/1570180043485563




Rational Design of Chemokine SDF-1 Analogs with Agonist Activity for the CXCR4 Receptor and the Capacity to Rapidly Mobilize PMN and Hematopoietic Progenitor Cells in Mice

, 1(2): 126 - 134

Ahmed Merzouk, Donald Wong, Hassan Salari, Huimin Bian, Seiji Fukuda and Louis M. Pelus


DOI: 10.2174/1570180043485608




Thalidomide as an Antiangiogenic Drug in the Treatment of Multiple Myeloma

, 1(2): 135 - 136

Domenico Ribatti and Angelo Vacca


DOI: 10.2174/1570180043485491




Recombinant Murine Polyoma Virus-like-particles Induce Protective Antitumour Immunity

, 1(2): 137 - 147

M. Brinkman, J. Walter, I. Jennes, M. Neugebauer, W. Bertling, S. Grein, M. Thies, M. Weigand, T. Beyer and M. Herrmann


DOI: 10.2174/1570180043485545




Catecholamines, Sympathetic Innervation and Immunity: Role in Experimental and Rheumatoid Arthritis

, 1(2): 148 - 162

D. Lorton and C. Lubahn


DOI: 10.2174/1570180043485518




Steps towards Phage Display Libraries with an Extended Amino Acid Repertoire

, 1(2): 163 - 167

M. Bjorklund and E. Koivunen


DOI: 10.2174/1570180043485572




Urocortin: Cardiovascular Actions and Therapeutic Implications

, 1(2): 168 - 172

M. T. Rademaker


DOI: 10.2174/1570180043485482




Towards an Experimental de Novo Design Protocol. The use of Protein Crystallography to Deconvolute Dynamic Combinatorial Processes

, 1(2): 173 - 177

Robert E. Babine, Michael J. Rynkiewicz, Lei Jin and Sherin S. Abdel-Meguid


DOI: 10.2174/1570180043485617




Grid-Based Hydrogen Bond Potentials with Improved Directionality

, 1(2): 178 - 183

Ruth Huey, David S. Goodsell, Garrett M. Morris and Arthur J. Olson


DOI: 10.2174/1570180043485581




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