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Letters in Drug Design & Discovery

Volume 19, 12 Issues, 2022
ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)
This journal supports open access

Articles Ahead of Print






An Insight into Osmotic Drug Delivery Systems


Pankaj Bhateja, Rajesh Asija, Yogendra Singh and Mona Piplani*


DOI: 10.2174/1570180819666220430010228
View Abstract








Investigation of the Anticancer Potential of 2-alkoxycarbonylallyl Esters Against Metastatic Murine Breast Cancer Line 4T1 Targeting the EGFR: A Combined Molecular Docking, QSAR, and Machine Learning Approach


Babatunde Samuel Obadawo, Oluwatoba Emmanuel Oyeneyin*, Taoreed Olakunle Owolabi, Damilohun Samuel Metibemu, Nureni Ipinloju, Kehinde Henry Fagbohungbe, Helen Omonipo Modamori and Victor Olanrewaju Olatoye


DOI: 10.2174/1570180819666220512111613
View Abstract


The New Era of Drug Discovery: The Power of Computer-aided Drug Design (CADD)


Igor José dos Santos Nascimento*, Thiago Mendonça de Aquino and Edeildo Ferreira da Silva-Júnior


DOI: 10.2174/1570180819666220405225817
View Abstract




Piperazine-based Semicarbazone Derivatives as Potent Urease Inhibitors: Design, Synthesis, and Bioactivity Screening


Ebrahim Saeedian Moghadam, Abdullah Mohammed Al-Sadi, Meysam Talebi, Massoud Amanlou, Musa Shongwe, Mohsen Amini* and Raid Abdel-Jalil*


DOI: 10.2174/1570180819666220405234009
View Abstract







Design, Synthesis, and Evaluation of Isoindoline Derivatives as New Antidepressant Agents


Ai-Ling Sun, Chao-Chao Wang, Hao Zhou, Yi-Fei Lang, Shu-Yue Fu, Ren-Min Liu and Kang Lei*


DOI: 10.2174/1570180819666220301141149
View Abstract


Synthesis and Anticancer Activities of Novel Bis-chalcones Incorporating the 1,3-diphenyl-1H-pyrazole Moiety: In silico and In vitro Studies


Magda F. Mohamed, Farid M. Sroor*, Shahinda E. Elsayed, Karima F. Mahrous, Lamiaa Mageed, Mahmoud Khaled Hanafy, Sherif A. Ibrahim, Ahmed H. M. Elwahy and Ismail A. Abdelhamid


DOI: 10.2174/1570180819666220301151631
View Abstract




Synthesis of Novel Urea and Sulfonamide Derivatives of Isatin Schiff Bases as Potential Anti-cancer Agents


Ural U. Demirel, Süreyya Ölgen*, Ecem F. Karaman, Mehmet Tanol, Sibel Özden and Hakan Göker


DOI: 10.2174/1570180819666220224115908
View Abstract




Repurposing Novel Antagonists for Targeting p7 Viroporin of HCV Using In silico Approach


Varsha Dwivedi, Rakesh Kumar Gupta, Amita Gupta, Vijay K Chaudhary, Sanjay Gupta and Vandana Gupta*


DOI: 10.2174/1570180819666220124112150
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Novel S-Mercaptotriazolebenzothiazole-Based Derivatives as Antimicrobial Agents: Design, Synthesis, and In Vitro Evaluation


Alaa M. Alqahtani*, Asmaa G. Safi El-Din, Randa Abdou, Ali H. Amin, Hany H. Arab and Ahmed H. Abdelazeem


DOI: 10.2174/1570180819666220301154851
View Abstract


Potential of Caffeic Acid Derivatives as Antimalarial Leads


Gilles Degotte*, Bernard Pirotte, Michel Frédérich and Pierre Francotte


DOI: 10.2174/1570180819666220202160247
View Abstract







Thiamine: A Natural Peroxisome Proliferator-Activated Receptor Gamma (PPAR-γ) Activator


Parasuraman Aiya Subramani, Firdose Begum Shaik, R. Dinakaran Michael, Kalpana Panati and Venkata Ramireddy Narala*


DOI: 10.2174/1570180819666220127121403
View Abstract


Boesenbergia Pandurata as an Anti-Breast Cancer Agent: Molecular Docking and ADMET Study


Mohammad Rizki Fadhil Pratama, Ersanda Nurma Praditapuspa, Dini Kesuma, Hadi Poerwono, Tri Widiandani and Siswandono Siswodihardjo*


DOI: 10.2174/1570180819666211220111245
View Abstract





Synthesis and Antimicrobial Activity of Functional Derivatives of thiazolo[ 2,3-c][1,2,4]triazoles


Mikhailo Slivka*, Maksym Fizer, Ruslan Mariychuk, Marek Ostafin, Olexander Moyzesh, Galyna Koval, Oksana Holovko- Kamoshenkova, Ivan Rusyn and Vasy l Lendel


DOI: 10.2174/1570180819666220110145659
View Abstract






Gabapentin Antioxidant Derivatives with Anti-Inflammatory and Neuroprotective Potency


Georgios Papagiouvannis*, Panagiotis Theodosis-Nobelos, Paraskevi Tziona, Antonios Gavalas, Panos N. Kourounakis and Eleni A. Rekka


DOI: 10.2174/1570180818666211210161922
View Abstract








Editor-in-Chief

Ivana Cacciatore
Department of Pharmacy
University "G. d'Annunzio" of Chieti-Pescara
Chieti Scalo
(Italy)
Biography
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