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"Letters in Drug Design & Discovery should be available in every library in the pharmaceutical industry and in universities."

R. F. Borne, Associate Director
Laboratory for Applied Drug Design and Synthesis, The University of Mississippi, USA

Forthcoming Special Issues

Opportunities and challenges in anticandidal drug discovery and development

Guest Editor(s): Mohammad Abid
Tentative Publication Date: September, 2018
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Published Special Issues


Letters in Drug Design & Discovery, Volume 15, Number 03
Guest Editor(s): Gokhan Zengin, Marcello Locatelli

Authors' Comments
I would like to thank Bentham Science Publishers for their peerless effort to keep up scientists and students updated with the latest science and research work. Actually, Bentham assists researchers to achieve their goals to spread their reputation worldwide. I have experienced sincere, efficient and effective communication while dealing with Bentham team members. I intend to submit my work to Bentham and try to pick up journals that match my research profile. I have submitted a recent work to Medicinal Chemistry and nowadays I am drafting a manuscript targeting Current Pharmaceutical Design. Honestly, no words neither sentences would express my gratefulness and admiration. Bentham has offered my institution three months trial to access their journal lists and surf on its Board. This free access trial fulfills my literature review and broadens my horizon to absorb the recent research in pharmaceutical sciences and medicinal chemistry. Finally, I wish Bentham more success and achievement!

Dima Sabbah
(Department of Pharmacy, Faculty of Pharmacy, Al-Zaytoonah University of Jordan, Amman, Jordan)

Letters in Drug Design & Discovery


Volume 15


Number 9

Biography   Open Access

Research Article

Research Article

Research Article

Design, Synthesis and anti-HIV-1 Activity of Modified Styrylquinolines

, 15(9): 937 - 944

Shivani Mahajan, Shiv Gupta, Nisha Jariwala, Deepali Bhadane , Late K.K. Bhutani, Smita Kulkarni* and Inder Pal Singh*

DOI: 10.2174/1570180815666171212143339

Research Article

Research Article

Synthesis and Mosquiticidal Activity of Novel Hydrazone Containing Pyrimidine Derivatives against Aedes aegypti

, 15(9): 951 - 956

Zhong-Hua Shen, Zhao-Hui Sun, James J. Becnel, Alden Estep , David E. Wedge*, Cheng-Xia Tan, Jian-Quan Weng, Liang Han and Xing-Hai Liu*

DOI: 10.2174/1570180815666180102141640

Research Article

Research Article

Articles Ahead of Print

3D QSAR Based Virtual Screening of Pyrido[1,2-a] Benzimidazoles as Potent Antimalarial Agents

Kalicharan Sharma, Apeksha Srivastava, Pooja Tiwari, Shweta Sharma, Mohammad Shaquiquzzaman, M. Mumtaz Alam and Mymoona Akhter*

View Abstract

Assessing the Antimalarial Potentials of Phytochemicals: Virtual Screening, Molecular Dynamics and In-Vitro Investigations

Saumya K. Patel, Mohd Athar, Prakash C Jha*, Vijay Khedkar, Yogesh T. Jasrai, Himanshu A. Pandya, Linz-Buoy George and H. Highland

View Abstract

Aurones as New Porcine Pancreatic α-Amylase Inhibitors

Khashayar Roshanzamir, Elaheh Kashani-Amin, Azadeh Ebrahim-Habibi and Latifeh Navidpour*

View Abstract

Synthesis of 3-furanyl-4,5-dihydroisoxazole Derivatives via Cycloaddition and their Antibacterial Evaluation

Gabriela Andrade Danin Barbosa, Alcino Palermo de Aguiar*, Erika Martins de Carvalho and Joseli Maria da Rocha Nogueira

View Abstract

Total Synthesis and Antibacterial Screening of (±)-6,8-Dihydroxy-3- undecyl-3,4-dihydroisochromen-1-one; A Structural Analog of Metabolites from Ononis natrix

Hummera Rafique*, Aamer Saeed, Ehsan Ullah Mughal, Muhammad Naveed Zafar, Amara Mumtaz, Naghmana Kausar and Kiran Hina

View Abstract

A Study on the Synthesis of Risedronic Acid; The Role of an Ionic Liquid Additive

David Illes Nagy, Alajos Grun, Julia Sinkovicz, Sandor Garadnay, Istvan Greiner and Gyorgy Keglevich*

View Abstract

Synthesis and Anticancer Activity of Some 1H-inden-1-one Substituted (Heteroaryl)Acetamide Derivatives

Ahmet Cagri Karaburun, Nalan Gundogdu-Karaburun*, Leyla Yurttas, Ismail Kayagil and Seref Demirayak

View Abstract

Oxime K033-Reactivation Activity of Cholinesterases Inhibited by Various Nerve Agents and Organophosphorus Pesticides

Kamil Kuca*, Kamil Musilek, Daniel Jun, Jaroslav Pejchal, Ondrej Krejcar, Marek Penhaker, Qinghua Wu, Raquel O. Lopes, Teodorico C. Ramalho, Tanos C. C. Franca, Eugenie Nepovimova and Ondrej Soukup

View Abstract

Abstracts Ahead of Print

3D-QSAR Studies of S-DABO Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors

Yueping Wang, Jie Chang, Jiangyuan Wang, Peng Zhong, Yufang Zhang, Christopher Cong Lai and Yanping He*

View Abstract

Synthesis, Anti-inflammatory, Antimicrobial Potential and Molecular Docking Studies of 4,5-Disubstituted-1,2,4-Triazole Thioacetate Derivatives

Muhammad Nouman Arif, Humaira Nadeem*, Rehan Zafar Paracha, Arifullah Khan, Imran Khanzada and Fawad Ali

View Abstract

Synthesis and Biological Activity Evaluation of N-(arylsulfonyl) Valine Hydrazones and Assistance of NMR Spectroscopy for Definitive 3D Structure

Sevil Senkardes, Esra Tatar, Ridvan Nepravishta, Dorisa Cela, Maurizio Paci, Ozlem Bingol Ozakpinar, Turgut Sekerler, Erik De Clercq, Christophe Pannecouque, S. Guniz Kucukguzel* and Ilkay Kucukguzel

View Abstract

Molecular modeling of an orphan GPR18 receptor

Kamil J. Kuder , Tadeusz Karcz, Maria Kaleta and Katarzyna Kiec-Kononowicz*

View Abstract

Identification of New Inhibitors of Mutant Isocitrate Dehydrogenase 2 through Molecular Similarity-based Virtual Screening

Lijun Yang, Stefan Pusch, Tianfang Ma, Qihua Zhu, Yungen Xu, Andreas von Deimling, Xiaoming Zha* and Tsygankova Victoria Jennings

View Abstract

Paclitaxel-Tyroserleutide Conjugates Self-assembly into Nanocarrier for Drug Delivery

Yongjia Liu, Leilei Shi, Bangshang Zhu*, Yue Su, Hui Li and Xinyuan Zhu

View Abstract

Synthesis and biological evaluation of some novel thiophene-bearing quinazoline derivatives as EGFR inhibitors

Min Zou, Bo Jin, Yanrong Liu, Huiping Chen, Zhuangli Zhang, Changzheng Zhang, Zhihong Zhao and Liyun Zheng*

View Abstract

2-Acryloyl-4,5-methylenedioxyphenol: A Small Molecule Endowed with Antidermatophytic Activity

Marco Zuccolo, Sabrina Dallavalle*, Raffaella Cincinelli, Luce Mattio, Stefania Mazzini, Michelandrea De Cesare and Loana Musso

View Abstract

Cytotoxicity of sodium arsenite-loaded anti-HER2 immunoliposomes against HER2-expressing human breast cancer cell lines

Moslem Afrakhteh, Alireza Kheirollah, Aminollah Pourshohod, Mohammad Ali Ghaffari, Mostafa Jamalan* and Majid Zeinali

View Abstract

Caffeic Acid Phenethyl Ester Effects: In silico Study of its Osteoimmunological Mechanisms

Ghulam Murtaza*, Yuhao Zhao, Xiaokun Pang, Xiaoxin Xu, Xincan Jiang, Dongbin Zhao, Yanxu Ma and Akriti Nepal

View Abstract

Editor's Choice

Synthesis and Mosquiticidal Activity of Novel Hydrazone Containing Pyrimidine Derivatives against Aedes aegypti

, 2018; 15(9): 951 - 956

Zhong-Hua Shen, Zhao-Hui Sun, James J. Becnel, Alden Estep, David E. Wedge*, Cheng-Xia Tan, Jian-Quan Weng, Liang Han and Xing-Hai Liu*

DOI: 10.2174/1570180815666180102141640

Inhibitory Effects of 1,4-disubstituted Thiosemicarbazide Derivatives on Streptococcus mutans and Streptococcus sanguinis Mono-species Biofilms

, 2018; 15(8): 843 - 850

Malgorzata Miazga-Karska, Maciej Wos, Agnieszka A. Kaczor, Anna Pachuta-Stec, Grazyna Ginalska and Monika Pitucha*

DOI: 10.2174/1570180814666171012164241

Enhancement Antimicrobial Activity of Clarithromycin by Amine Functionalized Mesoporous Silica Nanoparticles as Drug Delivery System

, 2018; 15(7): 787 - 795

Pegah Khosravian, Mehdi Khoobi, Mehdi Shafiee Ardestani, Mohammad Porgham Daryasari, Malihe Hassanzadeh, Payam Ghasemi-Dehkordi, Massoud Amanlou and Hamid Akbari Javar*

DOI: 10.2174/1570180815666180117155818

Synthesis and Mosquitocidal Activity of a Series of Hydrazone Derivatives against Aedes aegypti

, 2018; 15(6): 671 - 677

Mehlika Dilek Altintop*, Nurhayat Tabanca, James J. Becnel, Jeffrey R. Bloomquist, Zafer Asim Kaplancikli and Ahmet Ozdemir

DOI: 10.2174/1570180814666171002155548

Antimicrobial, Gastroprotective and Healing Effect of the Hydroalcoholic Extract of Astronium fraxinifolium

, 2018; 15(3): 325 - 334

Anita Oliveira Brito Pereira Bezerra Martins, Ana Luiza Albuquerque Siebra, Cicera Datiane de Morais Oliveira, Gerlania Oliveira Leite, Henrique Douglas Melo Coutinho, Margareth Linde Athayde, Aline Augusti Bolignon, Jacqueline Cosmo Andrade, Larissa Rolim Oliveira, Marta Regina Kerntopf, Roseli Barbosa, Francisco Rafael Alves Santana Cesario, Thales Silva Coutinho, Lucindo Jose Quintans-Junior and Irwin Rose Alencar de Menezes*

DOI: 10.2174/1570180814666170213160114

Synthesis and Antimicrobial Activity of Some Novel Substituted 3-(Thiophen-2-yl)pyrazole-based Heterocycles

, 2017; 14(11): 1316 - 1323

Bakr F. Abdel-Wahab*, Abdelbasset A. Farahat, Ghada E. A. Awad and Gamal A. El-Hiti*

DOI: 10.2174/1570180814666170327162447

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