Contents
Drug Metabolism Letters, Volume 10 - Number 3
Editorial
Research Article
New Screening Criteria Setting on Evaluation of Cytochrome P450 Induction Using HepaRG Cells with Multiplex Branched DNA Technologies in Early Drug Discovery
, 10(3): 152 - 160Akira Ogasawara, Nao Torimoto, Naoki Tsuda, Fumika Aohara, Rikiya Ohashi, Yasuhiro Yamada and Hideki Taniguchi
DOI: 10.2174/1872312810666160822110011
Research Article
Intracellular Retention of Three Quinuclidine Derivatives in Caco-2 Permeation Experiments: Mechanisms and Impact on Estimating Permeability and Active Efflux Ratio
, 10(3): 161 - 171Hong Jin, Sudarshan Kapadnis, Ting Chen, Dooyoung Lee, Andrew McRiner, Andrew Cook, Duane A. Burnett, Gerhard Koenig and Cuyue Tang
DOI: 10.2174/1872312810666160725123322
Research Article
Application of a “Fit for Purpose” PBPK Model to Investigate the CYP3A4 Induction Potential of Enzalutamide
, 10(3): 172 - 179Rangaraj Narayanan, Matthew Hoffmann, Gondi Kumar and Sekhar Surapaneni
DOI: 10.2174/1872312810666160729124745
Research Article
An Investigation of Sodium Fusidate and Recombinant Cytochrome P450 Enzymes Inhibition In-Vitro
, 10(3): 180 - 186John Mishriky, Jacqueline Balassone, Zenah Bashour, Simranjit Kaur, Vini Raman, Robel Getachew, Narin Osman, Daniel Guidone, Vincent Chan and Peter J. Little
DOI: 10.2174/1872312810666160607015045
Research Article
Inhibition of Procarcinogen Activating Enzyme CYP1A2 Activity and Free Radical Formation by Caffeic Acid and its Amide Analogues
, 10(3): 187 - 194Paitoon Narongchai, Kanokporn Niwatananun, Siripun Narongchai, Winthana Kusirisin and Churdsak Jaikang
DOI: 10.2174/1872312810666160608123113
Research Article
The Uremic Toxin Indoxyl-3-Sulfate Induces CYP1A2 In Primary Human Hepatocytes
, 10(3): 195 - 199Hong Liu, Rangaraj Narayanan, Matthew Hoffmann and Sekhar Surapaneni
DOI: 10.2174/1872312810666160719143703
Research Article
Identification and Characterization of the Human Cytosolic Sulfotransferases Mediating the Sulfation of Clioquinol and Iodoquinol
, 10(3): 200 - 205Akihiro Yamamoto, Maame Debrah-Pinamang, Nicholas J. DiModica, Katsuhisa Kurogi, Ali A. Naqvi, Ying Hui, Yoichi Sakakibara, Masahito Suiko and Ming-Cheh Liu
DOI: 10.2174/1872312810666160719142850
Research Article
UHPLC Quantitation Method for New Thiazolidinedione LPSF/GQ-02 and In Vitro/In Vivo Kinetic Studies
, 10(3): 206 - 212Carla Monalizi Vieira, Michel Leandro de Campos, Elias Carvalho Padilha, Marina Pitta, Ivan da Rocha Pitta, Maria do Carmo Alves de Lima and Rosângela Gonçalves Peccinini
DOI: 10.2174/1872312810666160725124554
Research Article
CYP2B6 and OPRM1 Receptor Polymorphisms at Methadone Clinics And Novel OPRM1 Haplotypes: A Cross-Sectional Study
, 10(3): 213 - 218Ahmad Abdulrahman AlMeman, Rusli Ismail and Markus Perola
DOI: 10.2174/1872312810666160810104040
Research Article
Effect of Cardiovascular Injury on Catabolism of Adenosine and Adenosine 5-‘Triphosphate in Systemic Blood in a Freely Moving Rat Model In Vivo
, 10(3): 219 - 226Pollen K. Yeung, Shyam S. Kolathuru and Remigius U. Agu
DOI: 10.2174/1872312810666160607013859
Webmaster Contact: info@benthamscience.org