Contents

Current Topics in Medicinal Chemistry, Volume 16 - Number 4


Editorial


Metalloprotein Inhibitors for the Treatment of Human Diseases

, 16(4): 384 - 396

Yang Yang, Xue-Qin Hu, Qing-Shan Li, Xing-Xing Zhang, Ban-Feng Ruan, Jun Xu and Chenzhong Liao


DOI: 10.2174/1568026615666150813145218



Advances in Bacterial Methionine Aminopeptidase Inhibition

, 16(4): 397 - 414

Travis R. Helgren, Phumvadee Wangtrakuldee, Bart L. Staker and Timothy J. Hagen


DOI: 10.2174/1568026615666150813145410



Selective Histone Deacetylase Inhibitors with Anticancer Activity

, 16(4): 415 - 426

Nan Ma, Ying Luo, Ying Wang, Chenzhong Liao, Wen-Cai Ye and Sheng Jiang


DOI: 10.2174/1568026615666150813145629




6,7-Dihydroxyisoindolin-1-one and 7,8-Dihydroxy-3,4-Dihydroisoquinolin- 1(2H)-one Based HIV-1 Integrase Inhibitors

, 16(4): 435 - 440

Xue Zhi Zhao, Mathieu Métifiot, Steven J. Smith, Kasthuraiah Maddali, Christophe Marchand, Stephen H. Hughes, Yves Pommier, Terrence R. Burke and Jr.


DOI: 10.2174/1568026615666150813150058



Novel HIV-1 Integrase Inhibitor Development by Virtual Screening Based on QSAR Models

, 16(4): 441 - 448

Laura Guasch, Alexey V. Zakharov, Olga A. Tarasova, Vladimir V. Poroikov, Chenzhong Liao and Marc C. Nicklaus


DOI: 10.2174/1568026615666150813150433



Non-Zinc-Binding Inhibitors of MMP-13: GRID-Based Approaches to Rationalize the Binding Process

, 16(4): 449 - 459

Antonella Di Pizio, Mariangela Agamennone and Paolo Tortorella


DOI: 10.2174/1568026615666150813150631



In Vitro Inhibition of Glyoxalase І by Flavonoids: New Insights from Crystallographic Analysis

, 16(4): 460 - 466

Hong Zhang, Jing Zhai, Liping Zhang, Cuiyun Li, Yining Zhao, Yunyun Chen, Qing Li and Xiao Peng Hu


DOI: 10.2174/1568026615666150813150944




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