Contents

Current Topics in Medicinal Chemistry, Volume 11 - Number 17

Editorial [Hot Topic: New Developments in the Medicinal Chemistry of Vanilloid TRPV1 and Related Receptors (Guest Editor: Arpad Szallasi)]

, 11(17): 2116 - 2117

Arpad Szallasi


DOI: 10.2174/156802611796904906




Therapeutic Targeting of TRP Channels - The TR(i)P to Pain Relief

, 11(17): 2118 - 2130

Samer R. Eid


DOI: 10.2174/156802611796904898




TRP Channel Gating Physiology

, 11(17): 2131 - 2150

Andres Nieto-Posadas, Andres Jara-Oseguera and Tamara Rosenbaum


DOI: 10.2174/156802611796904870




TRPV1 Activation is Not An All-Or-None Event: TRPV1 Partial Agonism/Antagonism and Its Regulatory Modulation

, 11(17): 2151 - 2158

Peter M. Blumberg, Larry V. Pearce and Jeewoo Lee


DOI: 10.2174/156802611796904825




Therapeutic Targeting of TRPV1 by Resiniferatoxin, from Preclinical Studies to Clinical Trials

, 11(17): 2159 - 2170

Igor Kissin and Arpad Szallasi


DOI: 10.2174/156802611796904924




The Vanilloid Agonist Resiniferatoxin for Interventional-Based Pain Control

, 11(17): 2171 - 2179

Michael J. Iadarola and Andrew J. Mannes


DOI: 10.2174/156802611796904942




TRPV1 Signaling: Mechanistic Understanding and Therapeutic Potential

, 11(17): 2180 - 2191

Rong Xia, Tarek A. Samad, Joan Btesh, Lin-Hua Jiang, Ibrahim Kays, Louise Stjernborg and Niek Dekker


DOI: 10.2174/156802611796904843




Disease-Related Changes in TRPV1 Expression and Its Implications for Drug Development

, 11(17): 2192 - 2209

Louis S. Premkumar and Mahendra Bishnoi


DOI: 10.2174/156802611796904834




Analgesic Potential of TRPV3 Antagonists

, 11(17): 2210 - 2215

Regina M. Reilly and Philip R. Kym


DOI: 10.2174/156802611796904889




TRPV4 Agonists and Antagonists

, 11(17): 2216 - 2226

Fabien Vincent and Matthew A.J. Duncton


DOI: 10.2174/156802611796904861




Transient Receptor Potential A1 Modulators

, 11(17): 2227 - 2236

Tim Strassmaier and Rajagopal Bakthavatchalam


DOI: 10.2174/156802611796904915




TRPM8 Biology and Medicinal Chemistry

, 11(17): 2237 - 2252

Jeff DeFalco, Matthew A.J. Duncton and Daniel Emerling


DOI: 10.2174/156802611796904933




Inhibition of the Function of TRPV1-Expressing Nociceptive Sensory Neurons by Somatostatin 4 Receptor Agonism: echanism and Therapeutical Implications

, 11(17): 2253 - 2263

Janos Szolcsanyi, Erika Pinter, Zsuzsanna Helyes and Gabor Petho


DOI: 10.2174/156802611796904852




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