Contents

Current Topics in Medicinal Chemistry, Volume 10 - Number 3

Editorial [Hot topic: The Medicinal Chemistry of Protease Inhibitors (Guest Editors: Wibke E. Diederich and Christof Wegscheid-Gerlach)]

, 10(3): 231

Wibke E. Diederich and Christof Wegscheid-Gerlach


DOI: 10.2174/156802610790725443




Proteasome Inhibitors: Recent Advances and New Perspectives In Medicinal Chemistry

, 10(3): 232 - 256

E. Genin, M. Reboud-Ravaux and J. Vidal


DOI: 10.2174/156802610790725515




Entering the Era of Non-Basic P1 Site Groups: Discovery of Xarelto™ (Rivaroxaban)

, 10(3): 257 - 269

Alexander Straub, Susanne Roehrig and Alexander Hillisch


DOI: 10.2174/156802610790725506




Calpains: Attractive Targets for the Development of Synthetic Inhibitors

, 10(3): 270 - 293

Markus Pietsch, Krystle C. H. Chua and Andrew D. Abell


DOI: 10.2174/156802610790725489




Development of Nitrile-Based Peptidic Inhibitors of Cysteine Cathepsins

, 10(3): 294 - 322

Maxim Frizler, Marit Stirnberg, Mihiret Tekeste Sisay and Michael Gutschow


DOI: 10.2174/156802610790725452




Recent Advances in Targeting Viral Proteases for the Discovery of Novel Antivirals

, 10(3): 323 - 345

Holger Steuber and Rolf Hilgenfeld


DOI: 10.2174/156802610790725470




Proteases of Plasmodium falciparum as Potential Drug Targets and Inhibitors Thereof

, 10(3): 346 - 367

Christof Wegscheid-Gerlach, Hans-Dieter Gerber and Wibke E. Diederich


DOI: 10.2174/156802610790725461




Enzyme Kinetics and Hit Validation in Fluorimetric Protease Assays

, 10(3): 368 - 382

Stephanie Ludewig, Markus Kossner, Markus Schiller, Knut Baumann and Tanja Schirmeister


DOI: 10.2174/156802610790725498




Webmaster Contact: info@benthamscience.org
Copyright © 2018 Bentham Science