Contents

Current Medicinal Chemistry, Volume 11 - Number 6

Preface [Hot Topic: Emerging Kinase Targets and Kinase Inhibitor Discovery Methods (Guest Editor: Gary McCort)]

, 11(6): ii

Gary McCort


DOI: 10.2174/09298673104090600ii




Recent Kinase and Kinase Inhibitor X-ray Structures: Mechanisms of Inhibition and Selectivity Insights

, 11(6): 663 - 673

M. Cherry and D. H. Williams


DOI: 10.2174/0929867043455792




Stochastic Algorithm for Kinase Homology Model Construction

, 11(6): 675 - 692

A. Rayan, E. Noy, D. Chema, A. Levitzki and A. Goldblum


DOI: 10.2174/0929867043455701




Virtual Screening for Kinase Targets

, 11(6): 693 - 707

Ingo Muegge and Istvan J. Enyedy


DOI: 10.2174/0929867043455684




Property-Based Design of KDR Kinase Inhibitors

, 11(6): 709 - 719

Mark E. Fraley, William F. Hoffman, Kenneth L. Arrington, Randy W. Hungate, George D. Hartman, Rosemary C. McFall, Kathleen E. Coll, Keith Rickert, Kenneth A. Thomas and Georgia B. McGaughey


DOI: 10.2174/0929867043455729




AlphaScreen™ Kinase HTS Platforms

, 11(6): 721 - 730

Greg Warner, Chantal Illy, Liliana Pedro, Philippe Roby and Roger Bosse


DOI: 10.2174/0929867043455693




Development of Vascular Endothelial Growth Factor Receptor (VEGFR) Kinase Inhibitors as Anti-Angiogenic Agents in Cancer Therapy

, 11(6): 731 - 745

T. L. Underiner, B. Ruggeri and D. E. Gingrich


DOI: 10.2174/0929867043455756




4-Thiophenoxy-N-(3,4,5-Trialkoxyphenyl)Pyrimidine-2-Amines as Potent and Selective Inhibitors of the T-Cell Tyrosine Kinase p56lck

, 11(6): 747 - 753

D. F.C. Moffat, R. A. Allen, S. E. Rapecki, P. D. Davis, J. O'Connell, M. C. Hutchings, M. A. King, B. A. Boyce and M. J. Perry


DOI: 10.2174/0929867043455710




GSK-3 Inhibitors: Discoveries and Developments

, 11(6): 755 - 763

M. Alonso and A. Martinez


DOI: 10.2174/0929867043455738




Developing Inhibitors to Selectively Target Two-Component and Phosphorelay Signal Transduction Systems of Pathogenic Microorganisms

, 11(6): 765 - 773

K. Stephenson and J. A. Hoch


DOI: 10.2174/0929867043455765




Challenges in Antimicrobial Drug Discovery and the Potential of Nucleoside Antibiotics

, 11(6): 775 - 793

Suguna Rachakonda and Leanne Cartee


DOI: 10.2174/0929867043455774




Retinoids and Retinoid Receptors in the Control of Energy Balance: Novel Pharmacological Strategies in Obesity and Diabetes

, 11(6): 795 - 805

F. Villarroya, R. Iglesias and M. Giralt


DOI: 10.2174/0929867043455747




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