Combinatorial Chemistry & High Throughput Screening
Accelerated Technologies for Biotechnology, Bioassays, Medicinal Chemistry and Natural Products Research
Volume 24, 10 Issues, 2021
ISSN: 1875-5402 (Online)
ISSN: 1386-2073 (Print)
This journal supports open access
ISSN: 1875-5402 (Online)
ISSN: 1386-2073 (Print)
This journal supports open access
Contents
Combinatorial Chemistry & High Throughput Screening, Volume 8 - Number 4
G-Protein Coupled Receptor Assays: To Measure Affinity or Efficacy that is the Question
, 8(4): 285 - 292C. Williams and A. Sewing
DOI: 10.2174/1386207054020778
The CellCard(™) System: A Novel Approach to Assessing Compound Selectivity for Lead Prioritization of G Protein-Coupled Receptors
, 8(4): 293 - 299Oren Beske, Simon Goldbard and Pierre Turpin
DOI: 10.2174/1386207054020859
High Content Screening for G Protein-Coupled Receptors Using Cell-Based Protein Translocation Assays
, 8(4): 301 - 309Charlotta Granas, Betina Kerstin Lundholt, Arne Heydorn, Viggo Linde, Hans-Christian Pedersen, Christian Krog-Jensen, Mette M. Rosenkilde and Len Pagliaro
DOI: 10.2174/1386207054020741
Using IMAP Technology to Identify Kinase Inhibitors: Comparison with a Substrate Depletion Approach and Analysis of the Nature of False Positives
, 8(4): 319 - 325P. Singh, B. Lillywhite, C. Bannaghan and P. Broad
DOI: 10.2174/1386207054020769
Substrate Specificity and Novel Selective Inhibitors of TNF-α Converting Enzyme (TACE) from Two-Dimensional Substrate Mapping
, 8(4): 327 - 339Millard H. Lambert, R. Kevin Blackburn, Theresa D. Seaton, Daniel B. Kassel, Daniel S. Kinder, M. Anthony Leesnitzer, D. Mark Bickett, Janet R. Warner, Marc W. Andersen, Jennifer G. Badiang, David J. Cowan, Michael D Gaul, Kimberly G. Petrov, Michael H. Rabinowitz, Robert W. Wiethe, J. David Becherer, Darryl L. McDougald, David L. Musso, Robert C. Andrews and Marcia L. Moss
DOI: 10.2174/1386207054020840
Rat PXR Reporter-Gene Activity Correlates with the Induction of CYP3A in Rat Precision-Cut Liver Slices
, 8(4): 341 - 346Xiaoming Cui, Ann Thomas, Diana Montgomery, Chunyan Gu, Richard A. Morrison, Ronald E. White and K. -C. Cheng
DOI: 10.2174/1386207054020822
Identification of Nitric Oxide Donors by Biomimetic HTS Application
, 8(4): 347 - 352Gyorgy T. Balogh, Balazs Dalmadi, Attila Bielik and Gyorgy M. Keseru
DOI: 10.2174/1386207054020831
Recent Advances in Analytical Construct Resins
, 8(4): 361 - 371D. M. Whitehead, S. C. McKeown and A Routledge
DOI: 10.2174/1386207054020804
Editor-in-Chief
Gerald H. Lushington
LiS Consulting, Lawrence
KS
(USA)
Biography
LiS Consulting, Lawrence
KS
Biography
Biography of Gerald H. Lushington
Dr. Gerald Lushington received his Ph.D. in Chemistry from the University of New Brunswick. The author of 181 journal articles, nine book chapters and four patents, Lushington is currently Principal Consultant at LiS Consulting, and serves as Adjunct Professor of Food Nutrition Dietetic Health at Kansas State University. With more than 25 years experience in the application of molecular modeling, simulation and informatics to a diverse range of scientific applications, Lushington's primary areas of focus are in drug discovery and pharmacology.
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Journal History
Combinatorial Chemistry & High Throughput Screening Journal was launched in 1998. Dr. Gerald H. Lushington serves as the Editor-in-Chief of the journal.
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