Contents

Combinatorial Chemistry & High Throughput Screening, Volume 12 - Number 3

Screening of Antioxidant Phenolic Compounds Produced by In Vitro Shoots of Brassica oleracea L. var. costata DC

, 12(3): 230 - 240

Federico Ferreres, Carla Sousa, David M. Pereira, Patricia Valentao, Marcos Taveira, Anabela Martins, Jose A. Pereira, Rosa M. Seabra and Paula B. Andrade


DOI: 10.2174/138620709787581756




The Four Human γ-Aminobutyric Acid (GABA) Transporters: Pharmacological Characterization and Validation of a Highly Efficient Screening Assay

, 12(3): 241 - 249

Trine Kvist, Bolette Christiansen, Anders A. Jensen and Hans Brauner-Osborne


DOI: 10.2174/138620709787581684




Simultaneous Determination of LogD, LogP, and pKa of Drugs by Using a Reverse Phase HPLC Coupled with a 96-Well Plate Auto Injector

, 12(3): 250 - 257

Po-Chang Chiang and Yiding Hu


DOI: 10.2174/138620709787581693




Development and Validation of a High-Density Fluorescence Polarization-Based Assay for the Trypanosoma RNA Triphosphatase TbCet1

, 12(3): 258 - 268

Christophe Antczak, David Shum, Constantin Radu, Venkatraman E. Seshan and Hakim Djaballah


DOI: 10.2174/138620709787581729




Narrowing Laccase Substrate Specificity Using Active Site Saturation Mutagenesis

, 12(3): 269 - 274

Nirupama Gupta and Edgardo T. Farinas


DOI: 10.2174/138620709787581675




Design and Combinatorial Synthesis of a Library of Methylenesulfonamides and Related Compounds as Potential Kinase Inhibitors

, 12(3): 275 - 284

Jane E. Torr, Jonathan M. Large and Edward McDonald


DOI: 10.2174/138620709787581747




A Multi-Step NMR Screen for the Identification and Evaluation of Chemical Leads for Drug Discovery

, 12(3): 285 - 295

Kelly A. Mercier, Matthew D. Shortridge and Robert Powers


DOI: 10.2174/138620709787581738




High Throughput Screening Assay of α1G T-type Ca2+ Channels and Comparison with Patch-Clamp Studies

, 12(3): 296 - 302

Yoonjee Kim, Soonja Kang, Jae Yeol Lee and Hyewhon Rhim


DOI: 10.2174/138620709787581710




Docking-Based Virtual Screening: Recent Developments

, 12(3): 303 - 314

Tiziano Tuccinardi


DOI: 10.2174/138620709787581666




High Throughput Screening of Physicochemical Properties and In Vitro ADME Profiling in Drug Discovery

, 12(3): 315 - 329

Hong Wan and Anders G. Holmen


DOI: 10.2174/138620709787581701




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