Contents

Combinatorial Chemistry & High Throughput Screening, Volume 11 - Number 5

Editorial [Hot Topic: GPCR High Throughput Screening (Part 1) (Guest Editors: David P. Siderovski and Francis S. Willard)]

, 11(5): 336

Francis S. Willard and David P. Siderovski


DOI: 10.2174/138620708784534815




Functional Selectivity in GPCR Modulator Screening

, 11(5): 337 - 343

Terry Kenakin


DOI: 10.2174/138620708784534824




New Strategies in Drug Discovery for GPCRs: High Throughput Detection of Cellular ERK Phosphorylation

, 11(5): 344 - 356

Michael F. Crouch and Ron I.W. Osmond


DOI: 10.2174/138620708784534806




Label-Free Cell-Based Assays for GPCR Screening

, 11(5): 357 - 369

Ye Fang, Anthony G. Frutos and Ronald Verklereen


DOI: 10.2174/138620708784534789




State-Selective Binding Peptides for Heterotrimeric G-Protein Subunits:Novel Tools for Investigating G-Protein Signaling Dynamics

, 11(5): 370 - 381

Christopher A. Johnston, Francis S. Willard, J. Kevin Ramer, Rainer Blaesius, C. Natalia Roques and David P. Siderovski


DOI: 10.2174/138620708784534798




G Protein β γ Subunits as Targets for Small Molecule Therapeutic Development

, 11(5): 382 - 395

Alan V. Smrcka, David M. Lehmann and Axel L. Dessal


DOI: 10.2174/138620708784534761




A High Throughput Fluorescence Polarization Assay for Inhibitors of the GoLoco Motif/G-alpha Interaction

, 11(5): 396 - 409

Adam J. Kimple, Adam Yasgar, Mark Hughes, Ajit Jadhav, Francis S. Willard, Robin E. Muller, Christopher P. Austin, James Inglese, Gordon C. Ibeanu, David P. Siderovski and Anton Simeonov


DOI: 10.2174/138620708784534770




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