ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)

Volume 14, 12 Issues, 2017

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Letters in Drug Design & Discovery

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G. Perry

University of Texas
San Antonio, TX

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"Letters in Drug Design & Discovery should be available in every library in the pharmaceutical industry and in universities."

R. F. Borne, Associate Director
Laboratory for Applied Drug Design and Synthesis, The University of Mississippi, USA

Forthcoming Special Issue(s)

Opportunities and challenges in anticandidal drug discovery and development

Guest Editor(s): Mohammad Abid
Tentative Publication Date: July, 2017
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I'm really pleased with all the experience of publishing in Bentham Science, surely I'd recommend you to my colleagues.

Mariagracia Vera
(Laboratorio de Síntesis Orgánica, Diseño y Evaluación Farmacológica de Nuevos Productos, Departamento de Química, Facultad Experimental de Ciencias, Universidad del Zulia, Maracaibo, Venezuela)

Letters in Drug Design & Discovery


Volume 14


Number 10

Research Article

Research Article

Research Article

Synthesis and Biological Evaluation of 1,3,4-Thiadiazole Linked Phthalimide Derivatives as Anticancer Agents

, 14(10): 1138 - 1144

Zahra Rezaei, Setareh Moghimi, Rezvan Javaheri, Mehdi Asadi, Mohammad Mahdavi, Shabnam Shabani, Najmeh Edraki, Omidreza Firuzi, Maliheh Safavi, Mohsen Amini, Ali Asadipour, Elnaz Zeinalzadeh, Loghman Firoozpour and Alireza Foroumadi

DOI: 10.2174/1570180814666170127164759

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Research Article

Design, Synthesis and Antibacterial Activities of New Azo-compounds: An Experimental and a Computational Approach

, 14(10): 1145 - 1154

Jamshaid Ashraf, Ehsan Ullah Mughal, Shahzad Murtaza, Amina Sadiq, Sheraz Ahmad Khan Tanoli, Amara Mumtaz, Abdul Hameed, Khalid Mohammed Khan, Ishtiaq Ahmed, Bilal Khalid and Asif Javid

DOI: 10.2174/1570180814666170306124134

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Research Article

Development of Novel Selective Pharmacophore for Tankyrase Inhibitors

, 14(10): 1164 - 1175

Xin Qiao, Ting Ran, Yan-Min Zhang, Jing Pan, Ling-Feng Yin, Wei-Neng Zhou, Lu Zhu, Jun-Nan Zhao, Hai-Chun Liu, Shuai Lu, Tao Lu, Ya-Dong Chen and Yu-Lei Jiang

DOI: 10.2174/1570180814666170118151011

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Research Article

Ultrasound-Assisted 3-Component Reaction in Acetic Acid Alone: Catalyst / Promoter / Ligand Free Synthesis of Bioactive Pyrazolo[1,5-a]pyrimidines

, 14(10): 1176 - 1183

Namburi Suresh, Bodapati Veera Durgarao, A. Ratnakar, Sunder Kumar Kolli, Mohd Ashraf Ashfaq, Mandava V. Basaveswara Rao and Manojit Pal

DOI: 10.2174/1570180814666170126120408

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Computational Approach to the Discovery of Phytochemical Molecules with Therapeutic Potential Targets to the PKCZ protein

Poliany G. Freitas, Thiago C. Elias, Icaro A. Pinto, Luciano T. Costa, Paulo VSD de Carvalho, Daniel Q. Omote, Ihosvany Camps, Tati Ishikawa, Helen A. Arcuri, Susana Vinga, Arlindo L. Oliveira, Walter F.A. Junior and Nelson J. F. da Silveira

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Fighting Against Alzheimer's Disease: Synthesis of New Pyrazoline and Benzothiazole Derivatives as New Acetylcholinesterase and MAO Inhibitors

Gülhan Turan-Zitouni, Weiam Hussein, Begüm Nurpelin Sağlık, Merve Baysal and Zafer Asım Kaplancıklı

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Synthesis, Biological Evaluation, Molecular Docking Study and Acute Oral Toxicity Study of Coupled Imidazole-Pyrimidine Derivatives

Shailee V. Tiwari, Anna Pratima G. Nikalje, Deepak K. Lokwani, Aniket P. Sarkate and Kizukala Jamir

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Synthesis and Antioxidant Evaluation of a New Class of Thienopyrimidinerhodanine Hybrids

Kerru Nagaraju , Venkata H.S.S. Bhaskaruni, Ravada Kishore , Suresh Maddila, Parvesh Singh and Jonnalagadda B. Sreekantha

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Anti-MRSA (Multidrug Resistant Staphylococcus aureus) Activity of 3-Substituted Coumarins

Uzma Salar, Khalid Mohammed Khan, Humaira Muhammad, Muhammed Imran Fakhri, Sanaullah , Shahnaz Perveen and M. Iqbal Choudhary

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Nalidixic Acid Schiff Bases: Synthesis and Biological Evaluation

Asif Husain, Munendra Mohan Varshney, Versha Parcha, Aftab Ahmad and Shahalam Khan

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Exploration of Some Thiazolidine-2,4-dione and 2-Oxoindoline Derivatives Incorporating 3,4,5-Trimethoxybenzyl Moiety as Novel Anticancer Agents

Le Cong Huan, Hai Pham-The, Huong Le-Thi-Thu, Tran Phuong Thao , Do Nguyet Que , Nguyen-Thu Trang, Phan Thi Phuong Dung, Minji Pyo, Sang-Bae Han , Nguyen Thi Thuan and Nguyen-Hai Nam

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Synthesis of New Thiazolyl-Pyrazoline Derivatives and Evaluation of Their Antimicrobial, Cytotoxic and Genotoxic Effects

Belgin Sever, Mehlika Dilek Altıntop, Hulya Karaca Gencer, Handan Acelya Kapkac, Ozlem Atlı, Merve Baysal and Ahmet Ozdemir

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Synthesis, antioxidant and antimicrobial activities of metal complexes of 2-thiouracil-hydroxyquinoline derivatives

Apilak Worachartcheewan, Ratchanok Pingaew, Decha Lekcharoen, Supaluk Prachayasittikul, Somsak Ruchirawat and Virapong Prachayasittikul

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Highly Functionalized Tryptamine-Azole-Fluoroquinolone Hybrids: Microwave Irradiated and Conventional Synthesis, Antibacterial Activity Evaluation

Yıldız Uygun Cebeci, Serap Basoglu Ozdemir,, Hacer Bayrak, Sule Ceylan, Ahmet Demirbas, Neslihan Demirbas and Sengul Alpay Karaoglu

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Illicium verum extract exhibited anti-inflammatory action in rodents

Shagufta Khan, Huma Aslam Bhatti, Ghulam Abbas, Muhammad Ali Versiani, Shaheen Faizi, Salman Khalid Ahmed, Saad Jawaid , Anita Naushir Akbar Ali , Rabia Jamy , Fatima Shahid and Ahsana Dar Farooq

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Novel Hybrid Molecules of Isoxazole Chalcone Derivatives: Synthesis And Study of Invitro Cytotoxic Activities

Arunkumar Thiriveedhi, Ratnakaram Venkata Nadh , Navuluri Srinivasu and Kishore Kaushal

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Antimicrobial Activities of Synthetic Arylidine Nicotinic and Isonicotinic Hydrazones

Muhammad Hayat, Khalid Mohammed Khan, Sumayya Saeed, Uzma Salar, Momin Khan, Taimoor Baig, Aqeel Ahmad, Shahnaz Perveen and Muhammad Taha

View Abstract


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