ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)


Volume 14, 12 Issues, 2017


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Letters in Drug Design & Discovery

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University of Texas
San Antonio, TX
USA


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Laboratory for Applied Drug Design and Synthesis, The University of Mississippi, USA

Forthcoming Special Issue(s)

Opportunities and challenges in anticandidal drug discovery and development


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Tentative Publication Date: July, 2017
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Letters in Drug Design & Discovery

,

Volume 14

-

Number 10



Research Article

Research Article

Research Article

Synthesis and Biological Evaluation of 1,3,4-Thiadiazole Linked Phthalimide Derivatives as Anticancer Agents

, 14(10): 1138 - 1144

Zahra Rezaei, Setareh Moghimi, Rezvan Javaheri, Mehdi Asadi, Mohammad Mahdavi, Shabnam Shabani, Najmeh Edraki, Omidreza Firuzi, Maliheh Safavi, Mohsen Amini, Ali Asadipour, Elnaz Zeinalzadeh, Loghman Firoozpour and Alireza Foroumadi


DOI: 10.2174/1570180814666170127164759


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Research Article

Design, Synthesis and Antibacterial Activities of New Azo-compounds: An Experimental and a Computational Approach

, 14(10): 1145 - 1154

Jamshaid Ashraf, Ehsan Ullah Mughal, Shahzad Murtaza, Amina Sadiq, Sheraz Ahmad Khan Tanoli, Amara Mumtaz, Abdul Hameed, Khalid Mohammed Khan, Ishtiaq Ahmed, Bilal Khalid and Asif Javid


DOI: 10.2174/1570180814666170306124134


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Research Article

Development of Novel Selective Pharmacophore for Tankyrase Inhibitors

, 14(10): 1164 - 1175

Xin Qiao, Ting Ran, Yan-Min Zhang, Jing Pan, Ling-Feng Yin, Wei-Neng Zhou, Lu Zhu, Jun-Nan Zhao, Hai-Chun Liu, Shuai Lu, Tao Lu, Ya-Dong Chen and Yu-Lei Jiang


DOI: 10.2174/1570180814666170118151011


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Research Article

Ultrasound-Assisted 3-Component Reaction in Acetic Acid Alone: Catalyst / Promoter / Ligand Free Synthesis of Bioactive Pyrazolo[1,5-a]pyrimidines

, 14(10): 1176 - 1183

Namburi Suresh, Bodapati Veera Durgarao, A. Ratnakar, Sunder Kumar Kolli, Mohd Ashraf Ashfaq, Mandava V. Basaveswara Rao and Manojit Pal


DOI: 10.2174/1570180814666170126120408


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Computational Approach to the Discovery of Phytochemical Molecules with Therapeutic Potential Targets to the PKCZ protein


Poliany G. Freitas, Thiago C. Elias, Icaro A. Pinto, Luciano T. Costa, Paulo VSD de Carvalho, Daniel Q. Omote, Ihosvany Camps, Tati Ishikawa, Helen A. Arcuri, Susana Vinga, Arlindo L. Oliveira, Walter F.A. Junior and Nelson J. F. da Silveira


View Abstract



Fighting Against Alzheimer's Disease: Synthesis of New Pyrazoline and Benzothiazole Derivatives as New Acetylcholinesterase and MAO Inhibitors


Gülhan Turan-Zitouni, Weiam Hussein, Begüm Nurpelin Sağlık, Merve Baysal and Zafer Asım Kaplancıklı


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Synthesis, Biological Evaluation, Molecular Docking Study and Acute Oral Toxicity Study of Coupled Imidazole-Pyrimidine Derivatives


Shailee V. Tiwari, Anna Pratima G. Nikalje, Deepak K. Lokwani, Aniket P. Sarkate and Kizukala Jamir


View Abstract



Synthesis and Antioxidant Evaluation of a New Class of Thienopyrimidinerhodanine Hybrids


Kerru Nagaraju , Venkata H.S.S. Bhaskaruni, Ravada Kishore , Suresh Maddila, Parvesh Singh and Jonnalagadda B. Sreekantha


View Abstract



Anti-MRSA (Multidrug Resistant Staphylococcus aureus) Activity of 3-Substituted Coumarins


Uzma Salar, Khalid Mohammed Khan, Humaira Muhammad, Muhammed Imran Fakhri, Sanaullah , Shahnaz Perveen and M. Iqbal Choudhary


View Abstract



Nalidixic Acid Schiff Bases: Synthesis and Biological Evaluation


Asif Husain, Munendra Mohan Varshney, Versha Parcha, Aftab Ahmad and Shahalam Khan


View Abstract



Exploration of Some Thiazolidine-2,4-dione and 2-Oxoindoline Derivatives Incorporating 3,4,5-Trimethoxybenzyl Moiety as Novel Anticancer Agents


Le Cong Huan, Hai Pham-The, Huong Le-Thi-Thu, Tran Phuong Thao , Do Nguyet Que , Nguyen-Thu Trang, Phan Thi Phuong Dung, Minji Pyo, Sang-Bae Han , Nguyen Thi Thuan and Nguyen-Hai Nam


View Abstract



Synthesis of New Thiazolyl-Pyrazoline Derivatives and Evaluation of Their Antimicrobial, Cytotoxic and Genotoxic Effects


Belgin Sever, Mehlika Dilek Altıntop, Hulya Karaca Gencer, Handan Acelya Kapkac, Ozlem Atlı, Merve Baysal and Ahmet Ozdemir


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Synthesis, antioxidant and antimicrobial activities of metal complexes of 2-thiouracil-hydroxyquinoline derivatives


Apilak Worachartcheewan, Ratchanok Pingaew, Decha Lekcharoen, Supaluk Prachayasittikul, Somsak Ruchirawat and Virapong Prachayasittikul


View Abstract



Highly Functionalized Tryptamine-Azole-Fluoroquinolone Hybrids: Microwave Irradiated and Conventional Synthesis, Antibacterial Activity Evaluation


Yıldız Uygun Cebeci, Serap Basoglu Ozdemir,, Hacer Bayrak, Sule Ceylan, Ahmet Demirbas, Neslihan Demirbas and Sengul Alpay Karaoglu


View Abstract



Illicium verum extract exhibited anti-inflammatory action in rodents


Shagufta Khan, Huma Aslam Bhatti, Ghulam Abbas, Muhammad Ali Versiani, Shaheen Faizi, Salman Khalid Ahmed, Saad Jawaid , Anita Naushir Akbar Ali , Rabia Jamy , Fatima Shahid and Ahsana Dar Farooq


View Abstract



Novel Hybrid Molecules of Isoxazole Chalcone Derivatives: Synthesis And Study of Invitro Cytotoxic Activities


Arunkumar Thiriveedhi, Ratnakaram Venkata Nadh , Navuluri Srinivasu and Kishore Kaushal


View Abstract



Antimicrobial Activities of Synthetic Arylidine Nicotinic and Isonicotinic Hydrazones


Muhammad Hayat, Khalid Mohammed Khan, Sumayya Saeed, Uzma Salar, Momin Khan, Taimoor Baig, Aqeel Ahmad, Shahnaz Perveen and Muhammad Taha


View Abstract



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