ISSN: 1875-5992 (Online)
ISSN: 1871-5206 (Print)


Volume 16, 12 Issues, 2016


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Anti-Cancer Agents in Medicinal Chemistry

Formerly: Current Medicinal Chemistry - Anti-Cancer Agents

Aims & ScopeAbstracted/Indexed in

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  • 29th of 59 in Chemistry, Medicinal

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Editor-in-Chief:
Michelle Prudhomme
Universite Blaise Pascal - C.N.R.S
Aubiere Cedex
France


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Current: 2.469
5 - Year: 2.974

Upcoming Articles (E-Pub Abstracts ahead of Print)

Cordycepin Affects Multiple Apoptotic Pathways to Mediate Hepatocellular Carcinoma Cell Death


Yulin Zhou, Zhihua Guo, Qingfan Meng, Jiahui Lu, Ning Wang, Hui Liu, Qiming Liang, Yutong Quan, Di Wang and Jing Xie.


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Cetuximab immunoliposomes enhances delivery of 5-FU to skin squamous carcinoma cells


Raquel Petrilli, Josimar O. Eloy, Renata F. V. Lopez and Robert J Lee.


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Rapamycin-loaded immunoliposomes functionalized with trastuzumab: a strategy to enhance cytotoxicity to HER2-positive breast cancer cells


Josimar O. Eloy, Raquel Petrilli, Robert W. Brueggemeier, Juliana Maldonado Marchetti and Robert J Lee.


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Preparation and evaluation of in vitro self-assembling HSA nanoparticles for cabazitaxel


Na Qu, Yating Sun, Jing Xie and Lesheng Teng.


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Disulfiram’s anticancer activity: evidences and mechanisms


Yang Jiao, Bethany N Hannafon and Wei-Qun Ding.


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Effect of PUFAs oral administration on the amount of Apoptotic Caspases Enzymes in gastric cancer patients undergoing chemotherapy


Homayun Dolatkhah, Ahmad Movahedian, Mohammad-Hossein Somi, Mahmud Aghaei, Naser Samadi, Ahmad Mirza-Aghazade and Ali Esfahani.


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Use of azoles containing natural products in cancer prevention and treatment: An overview


Nasimudeen R. Jabir, Chelapram K. Firoz, Ashish Bhushan, Shams Tabrez and Mohammad A Kamal.


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The Role of Tumor Associated Macrophages in the Tumor Microenvironment: Mechanism and Functions


Jie Zhu, Binhua P. Zhou, Min Tao, Jingyi Liu and Wei Li.


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The cytotoxic effect of GW843682X on nasopharyngeal carcinoma


Qinyong Hu, Yuxin Chu, Weiguo Hu, Min Peng and Qibin Song.


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In Vivo Inhibition of Proteasome Activity and Tumour Growth by Murraya koenigii Leaf Extract in Breast Cancer Xenografts and by its active flavonoids in breast cancer cells


Bindu Noolu, Ramesh Gogulothu, Mehrajuddin Bhat, Syed SYH Qadri, V Sudhakar Reddy, G Bhanuprakash Reddy and Ayesha Ismail.


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Fe3O4 NANOPARTICLES MEDIATED SYNTHESIS OF NOVEL ISATIN-PYRIMIDINONE HYBRID MOLECULES AS ANTIOXIDANT AND CYTOTOXIC AGENTS


Srinubabu Maddela, Ajitha Makula and N Jayarambabu.


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Exploring the binding affinity of novel syringic acid analogues and critical determinants of selectivity as potent proteasome inhibitors


Srinivasulu Cheemanapalli, CM Anuradha, P Madhusudhana, M Mahesh, Pongali B Raghavendra and Chitta Suresh Kumar.


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New Approaches to Photodynamic Therapy from Type I, II and III to Type IV Using One or More Photons


Kathrin M. Scherer, Roger H. Bisby, Stanley W. Botchway and Anthony W Parker.


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Copper(II) complexes with saccharinate and glutamate as antitumor agents. Cyto- and genotoxicity in human osteosarcoma cells


J.F. Cadavid-Vargas, I.E. León, S.B. Etcheverry, E. Santi, M.H. Torre and AL Di Virgilio.


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New poly(3-hydroxybutyrate) microparticles with paclitaxel sustained release for intraperitoneal administration


A.P. Bonartsev, A.L. Zernov, S.G. Yakovlev, I.I. Zharkova, V.L. Myshkina, T.K. Mahina, G.A. Bonartseva, N.V. Andronova, G.B. Smirnova, J.A. Borisova, M.S. Kalishjan, K.V. Shaitan and HM Treshalina.


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Lichen acids may be used as a potential drug for cancer therapy; by inhibiting mitochondrial thioredoxin reductase purified from rat lung


Ilknur Ozgencli, Harun Budak, Mehmet Ciftci and Mustafa Anar.


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Synthesis and Anticancer Study of novel 4H-Chromen Derivatives


Xiaolin Lu, Gaochao Dong, Ying Zheng, Chao Zhang, Yang Qiu, Tao Lu and Xiang Zhou.


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Novel 2-Thienyl- and 2-Benzothienyl-Substituted 6-(2-Imidazolinyl)Benzothiazoles: Synthesis; in vitro Evaluation of Antitumor Effects and Assessment of Mitochondrial Toxicity


Livio Racané, Mirela Sedić, Nataša Ilić, Maja Aleksić, Sandra Kraljević Pavelić and Grace Karminski-Zamola.


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Aryl maleimides as apoptosis inducers on L5178-Y murine leukemia cells (in silico, in vitro and ex vivo study)


Erik Andrade-Jorge, Marycarmen Godínez-Victoria, Luvia Enid Sánchez-Torres, Luis Humberto Fabila-Castillo and José G Trujillo-Ferrara.


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Design, synthesis and evaluation of 5-pyridin-4-yl-2-thioxo-[1,3,4]oxadiazol-3-yl derivatives as anti-angiogenic agents Targeting VEGFR-2.


Umesh Bhanushali, Samidha Kalekar-Joshi, Renuka Kulkarni-Munshi, Swapna Yellanki, Raghavender Medishetty, Pushkar Kulkarni and C S Ramaa.


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Heterocyclic drug-polymer conjugates for cancer targeted drug delivery


Harmeet Kaur, Sapna D. Desai, Virender Kumar, Pooja Rathi and Jasbir Singh.


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Thiazolidinone constraint combretastatin analogs as novel antitubulin agents: Design, synthesis, biological evaluation and docking studies


Sahil Sharma, Manish Kumar Gupta, Ajit Kumar Saxena and Preet Mohinder Singh Bedi.


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Oleic Acid Protects Against Oxidative Stress Exacerbated by Cytarabine and Doxorubicin in Rat Brain


David Calderón Guzmán, Norma Osnaya Brizuela, Maribel Ortíz Herrera, Hugo Juárez Olguín, Ernestina Hernández García, Armando Valenzuela Peraza and Gerardo Barragán Mejía.


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Breast Cancer: Current Molecular Therapeutic Targets and New Players


Siddavaram Nagini.


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Selective Toxicity of Apigenin on Cancerous Hepatocytes by Directly Targeting their Mitochondria


Enayatollah Seydi, Hamid Reza Rasekh, Ahmad Salimi, Zhaleh Mohsenifar and Jalal Pourahmad.


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Epidrugs in the immunotherapy of cutaneous and uveal melanoma


Mario Venza, Maria Visalli, Teresa Catalano, Concetta Beninati, Diana Teti and Isabella Venza.


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Epigenetic and miRNAs dysregulation in prostate cancer: the role of nutraceuticals


Alessandra Bosutti, Fabrizio Zanconati, Gabriele Grassi, Barbara Dapas, Sabina Passamonti and Bruna Scaggiante.


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Trans-platinum(II)/(IV) complexes with acetylpyridine ligands as antivascular agents in vitro: cytotoxic and antiangiogenic potential


Filipović Lana, Aranđelović Sandra, Krivokuća Ana, Janković Radmila, Dojčinović Biljana and Radulović Siniša.


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Melatonin regulates angiogenic and inflammatory proteins in MDA-MB-231 cell line and in co-culture with cancer-associated fibroblasts


Larissa Bazela Maschio-Signorini, Gabriela Bottaro Gelaleti, Marina Gobbe Moschetta, Thaiz Ferraz Borin, Bruna Victorasso Jardim-Perassi, Juliana Ramos Lopes, Jéssica Zani Lacerda, Rosimeire Aparecida Roela, Newton Antonio Bordin Júnior, Lizandra Akina Corrêa, Jessica Picinin Cardoso and Debora Aparecida Pires de Campos Zuccari.


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To Analyze the Amelioration of Phenobarbital Induced Oxidative Stress by Erucin, as Indicated by Biochemical and Histological Alterations


Rohit Arora, Sakshi Bhushan, Rakesh Kumar, Rahul Mannan, Pardeep Kaur, Bikram Singh, Ritika Sharma, Adarsh Pal Vig, Balbir Singh, Amrit Pal Singh and Saroj Arora.


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The role of stromal components in pancreatic cancer progressionShort Title: stroma and pancreatic cancer


Mengdan Xu, Qiaoming Zhi, Binhua P. Zhou, Min Tao, Jingyi Liu and Wei Li.


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4-Anilinoquinazoline Derivatives with Epidermal Growth Factor Receptor Inhibitor Activity


Fang Liu, Yinjiu Huang, Hao Liu, Leina Li, Gang Liu, Yun Cheng, Yan Xu and Wenwen Chen.


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In vitro anticancer effects of two new potent hydrazide compounds in leukemic cells


Shahrzad Tavakolfar, Elham Musavi, Ali Almasirad, Amir Amanzadeh, Seyyed Mohamamd Atyabi, Parichehr Yaghamii, Somayeh Samiee-Sadr and Mona Salimi.


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Autophagy inhibits apoptosis induced by agrocybe aegerita lectin in hepatocellular carcinoma


Wei Liu, Guojun Yu, Wenhui Yu, Xiangdong Ye, Yanxia Jin, Alok Shrestha, Qing Yang and Hui Sun.


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Brain-metastatic breast cancer: clinical considerations and pharmacological approaches


Ana Carolina Andrade, Daniel Sartori Ferruzzi and Carolina Panis.


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Anticancer drug combinations, how far we can go through?


Da-Yong Lu, En-Hong Chen, Hong-Ying Wu, Ting-Ren Lu, Bin Xu and Jian Ding.


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Synthesis of Icaritin and β-anhydroicaritin Mannich Base Derivatives and Their Cytotoxic Activities on Three Human Cancer Cell Lines


Van-Son Nguyen, Ling Shi, Sheng-Chun Wang and Qiu-An Wang.


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Differential Cytotoxicity, Cellular Uptake, Apoptosis and Inhibition of BRCA1 Expression of BRCA1-Defective and Sporadic Breast Cancer Cells Induced by an Anticancer Ruthenium(II)-Arene Compound, RAPTA-EA1


Adisorn Ratanaphan, Tidarat Nhukeaw, Khwanjira Hongthong and Paul J Dyson.


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Effects of Epirubicin and Cisplatin against 4T1 Breast Cancer Cells are Enhanced by Myrtucommulone-A


Kenan izgi, Banu iskender, Cagri Sakalar, Aslıhan Arslanhan, Esra Hilal Yüksek, Esra Hizar and Halit Canatan.


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Synthesis and in vitro evaluation of the anticancer potential of new aminoalkanol derivatives of xanthone


Natalia Szkaradek, Daniel Sypniewski, Anna M. Waszkielewicz, Agnieszka Gunia-Krzyżak, Anna Galilejczyk, Sabina Gałka, Henryk Marona and Ilona Bednarek.


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Inhibitors of Cancer Stem Cells


María E. García-Rubiño, César Lozano-López and Joaquín M Campos.


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Synthesis of Methotrexate Loaded Chitosan nanoparticles and in vitro evaluation of the potential in treatment of prostate cancer


Selvi Gunel N, Ozel B, Kipcak S, Aktan C, Akgun C, Ak G, Yilmaz H, Biray Avci C, Dodurga Y and Hamarat Sanlier S.


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HISTAMINE AND HISTAMINERGIC RECEPTORS IN COLORECTAL CANCER: FROM BASIC SCIENCE TO EVIDENCE-BASED MEDICINE


Giuseppe Losurdo, Mariabeatrice Principi, Bruna Girardi, Maria Pricci, Michele Barone, Enzo Ierardi and Alfredo Di Leo.


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Anticancer Vitamin K3 analogues: A review


Kirti D. Badave, Ayesha A. Khan and Sandhya Y Rane.


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Cytotoxicity and Anti-proliferative Properties of Heterocyclic Compounds Derived from Progesterone


Rafat M. Mohareb, Nadia Y. MegallyAbdo and Abeer A Mohamed.


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α(N)-Heterocyclic Thiosemicarbazones: Iron Chelators That Are Promising for Revival of Gallium in Cancer Chemotherapy


Shuhong Cao, Xiahui Chen, Ligen Chen and Jingwen Chen.


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RADIOPHARMACEUTICALS IN tumor hypoxia imaging: A review focused on MEDICINAL chemiSTRY aspects


Pablo Cabral and Hugo Cerecetto.


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Circulating tumor cells: a new window for diagnosis and evaluation of cancer


Meihui Liu, Min Tang, Ming Li, Feng Gao, Can Shi, Jing Hou and Wenbin Zeng.


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Review Article: Novel Therapeutic Strategies Against Cancer: Marine-derived Drugs May Be The Answer?


Maria Alessandra Gammone, Graziano Riccioni, Fabio Galvano and Nicolantonio D'Orazio.


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Molecular Mechanisms of Anti-cancer Activities of β-elemene: Targeting Hallmarks of Cancer


Shiyu Jiang, Chunhua Ling, Wei Li, Hongxin Jiang, Qiaoming Zhi and Min Jiang.


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Peroxisome Proliferator-activated Receptors and their ligands in cancer drug resistance: opportunity or challenge


Bahman Yousefi, Nosratollah Zarghami, Nasser Samadi and Maryam Majidinia.


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8-bromo-7-methoxychrysin reversed M2 polarization of tumor-associated macrophages induced by liver cancer stem-like cells


Shuwen Sun, Yinghong Cui, Kaiqun Ren, Meifang Quan, Zhenwei Song, Hui Zou, Duo Li, Yu Zheng and Jianguo Cao.


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Fibroblast Growth Factor Receptor (FGFR): A new target for non-small cell lung cancer therapy


Federica Biello, Giovanni Burrafato, Erika Rijavec, Carlo Genova, Giulia Barletta, Anna Truini, Simona Coco, Maria Giovanna Dal Bello, Angela Alama, Francesco Boccardo and Francesco Grossi.


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Synthesis of Combretastatin A-4 analogs and their biological activity


Agnieszka Głowacka, Monika Gensicka, Grzegorz Cholewinski and Krystyna Dzierzbicka.


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Natural Product-Derived Spirooxindole Fragments Serve as Privileged Substructures for Discovery of New Anticancer Agents


Bin Yu, Yi-Chao Zheng, Xiao-Jing Shi, Ping-Ping Qi and Hong-Min Liu.


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Lgr5 contributes to intestinal metaplasia during gastric carcinogenesis: a meta-analysis


Ye Han, Hugang Shen, Xiaofeng Xue, Bin Yuan, Yuting Kuang, Qiaoming Zhi and Hong Zhao.


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The prognostic value of serum LDH levels in patients with hepatocellualr carcinoma after hepatic resection


Wen-Jie Hu, Shun-Jun Fu, Jing-Fang Diao, Dai-Wei Wan, Zhi-Jian Tan, Qiao-Ming Zhi and Jun-Ming He.


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Guaraná a richest caffeine food increase oxaliplatin sensitivity of colorectal HT-29 cells by apoptosis pathway modulation


Francine Carla Cadoná, Alencar Kolinski Machado, Verônica Farina Azzolin, Fernanda Barbisan, Eduardo Bortoluzzi Dornelles, Werner Glanzner, Paulo Bayard Dias Gonçalves, Charles Elias Assmann, Euler Esteves Ribeiro and Ivana Beatrice Mânica da Cruz.


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New Pyrano[2,3-d:6,5-d']dipyrimidine Derivatives - Synthesis, in vitro Cytotoxicity Activity and Computational Studies


Suresh Maddila, Sreekantha B Jonnalagadda, Kovashnee Naicker, Sridevi Gorle, Surjyakant Rana, Kotaiah Yalagala, Surya N. Maddila, Moganavelli Singh and Parvesh Singh.


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A Novel Method to Synthesize 4-Aryl-1H-1,2,3-Triazoles and their Anti-hepatoma Activity


Xiaolong Li, Yun He, Li Hai, Tao Zhang and Yong Wu.


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Long noncoding RNA C21orF96 promotes the migration, invasion and lymph node metastasis in gastric cancer


Ziguo Yang, Qiaoming Zhi, Dan Wang, Li Zhang, Yuting Kuang, Ruizhen Miao, Yulong Shi and Xiaobo Guo.


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Chemical Structure Characteristics and Bioactivity of Small Molecule FAK Inhibitors


Fang-Yuan CAO, Xiao-Ping ZHOU, Jing SU, Xiao-Hong YANG, Feng-Hui MU, Jia-Yi SHEN and Wei SUN.


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Hepato and Cardiotoxicity of Chemotherapeutic Treatment Evaluated by Means of Small Animal Imaging.


Fiorella Carla Tesán, Mariano Portillo, Diego Martinel-Lamas, Vanina Araceli Medina, María Jimena Salgueiro and Marcela Zubillaga.


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Nano-Hydroxyapatite Doped with Ho-166 as Drug Delivery System for Bone Cancer Therapy


Franciana Maria Rosa da Silva, Julio Cezar de Almeida Junior, Elizabeth Eugênio de Mello Oliveira, Marta de Souza Albernaz, Alexandre Malta Rossi and Ralph Santos-Oliveira.


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PERSPECTIVES OF BENZIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS IN THE NEW ERA


Snehlata Yadav, Balasubramanian Narasimhan and Harmeet kaur.


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Biological Potential of Halfsandwich Ruthenium(II) and Iridium(III) Complexes


Gerd Ludwig, Marija Mojić, Mirna Z. Bulatović, Sanja Mijatović, Danijela Maksimović-Ivanić, Dirk Steinborn and Goran N Kaluđerović.


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15,16-dihydrotanshinone I induces apoptosis and inhibits the proliferation, migration of human osteosarcoma cell line 143B in vitro


Xuepeng Chen, Qihong Li, Yan He, Hongjiang Du, Zhajun Zhan, Hong zhao, Jiejun Shi, Qingsong Ye and Ji'an Hu.


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Flavonoids with Therapeutic Potential in Prostate Cancer


Bao Vue, Sheng Zhang and Qiao-Hong Chen.


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Research Progress on the Antitumor Effects of Rhein: Literature Review


Chao Wu, Hongyan Cao, Hua Zhou, Lin Sun, Jingui Xue, Jianyuan Li, Yanqin Bian, Runfei Sun, Shu Dong, Ping Liu and Mingyu Sun.


View Abstract


1, 3, 6-Trihydroxy-7-methyl-9, 10-anthracenedione isolated from genus Lindera with anti-cancer activity


Guoqing Wei, Hui Chen, Fangyuan Nie, Xiaofeng Ma and Hezhong Jiang.


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O-6-methylguanine-DNA Methyltransferase Inhibits Gastric Carcinoma Cell Migration and Invasion by Downregulation of Matrix Metalloproteinase 2


Chenglong Li, Li Deng, Qiaoming Zhi, Qingyou Meng, Aimin Qian, Hongfei Sang, Jiazeng Xia and Xiaoqiang Li.


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Synthesis of Diflunisal thiazolidinones as anticancer agents


Sevil Şenkardeş, Özlem Bingöl Özakpınar, Derya Özsavcı, Azize Şener, Özge Çevik and ŞGüniz Küçükgüzel.


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Up-regulated circulating miR-106a by DNA methylation promised a potential diagnostic and prognostic marker for gastric cancer


Renshun Yuan, Gang Wang, Qiaoming Zhi, Huabin Chen, Ye Han, Bin Wang, Zhongyang Kou, Hao Hu, Zhaoji Guo, Xiaofeng Xue and Hong Zhao.


View Abstract


Clinical Significance of miR-1826 as a Novel Prognostic Biomarker in Colorectal Cancer


You Hu, Bin Yi, Songbing He, Pengfei Liu, Lei Wang, Jing Yu, Daiwei Wan, Jin Zhou, Xinguo Zhu and Qiaoming Zhi.


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