ISSN: 1875-5992 (Online)
ISSN: 1871-5206 (Print)


Volume 16, 12 Issues, 2016


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Anti-Cancer Agents in Medicinal Chemistry

Formerly: Current Medicinal Chemistry - Anti-Cancer Agents

Aims & ScopeAbstracted/Indexed in

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  • 29th of 59 in Chemistry, Medicinal

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Editor-in-Chief:
Michelle Prudhomme
Universite Blaise Pascal - C.N.R.S
Aubiere Cedex
France


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Current: 2.469
5 - Year: 2.974

Upcoming Articles (E-Pub Abstracts ahead of Print)

Selective Toxicity of Apigenin on Cancerous Hepatocytes by Directly Targeting their Mitochondria


Enayatollah Seydi, Hamid Reza Rasekh, Ahmad Salimi, Zhaleh Mohsenifar and Jalal Pourahmad.


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Epidrugs in the immunotherapy of cutaneous and uveal melanoma


Mario Venza, Maria Visalli, Teresa Catalano, Concetta Beninati, Diana Teti and Isabella Venza.


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Epigenetic and miRNAs dysregulation in prostate cancer: the role of nutraceuticals


Alessandra Bosutti, Fabrizio Zanconati, Gabriele Grassi, Barbara Dapas, Sabina Passamonti and Bruna Scaggiante.


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Trans-platinum(II)/(IV) complexes with acetylpyridine ligands as antivascular agents in vitro: cytotoxic and antiangiogenic potential


Filipović Lana, Aranđelović Sandra, Krivokuća Ana, Janković Radmila, Dojčinović Biljana and Radulović Siniša.


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Melatonin regulates angiogenic and inflammatory proteins in MDA-MB-231 cell line and in co-culture with cancer-associated fibroblasts


Larissa Bazela Maschio-Signorini, Gabriela Bottaro Gelaleti, Marina Gobbe Moschetta, Thaiz Ferraz Borin, Bruna Victorasso Jardim-Perassi, Juliana Ramos Lopes, Jéssica Zani Lacerda, Rosimeire Aparecida Roela, Newton Antonio Bordin Júnior, Lizandra Akina Corrêa, Jessica Picinin Cardoso and Debora Aparecida Pires de Campos Zuccari.


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To Analyze the Amelioration of Phenobarbital Induced Oxidative Stress by Erucin, as Indicated by Biochemical and Histological Alterations


Rohit Arora, Sakshi Bhushan, Rakesh Kumar, Rahul Mannan, Pardeep Kaur, Bikram Singh, Ritika Sharma, Adarsh Pal Vig, Balbir Singh, Amrit Pal Singh and Saroj Arora.


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Naphthoflavones as antiproliferative agents : Design, synthesis and Biological evaluation


Dinesh Kumara, Onkar singh, Kunal Nepali, PMS Bedi, Arem Qayum, Shashank Singh and Subheet K Jain.


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The role of stromal components in pancreatic cancer progressionShort Title: stroma and pancreatic cancer


Mengdan Xu, Qiaoming Zhi, Binhua P. Zhou, Min Tao, Jingyi Liu and Wei Li.


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4-Anilinoquinazoline Derivatives with Epidermal Growth Factor Receptor Inhibitor Activity


Fang Liu, Yinjiu Huang, Hao Liu, Leina Li, Gang Liu, Yun Cheng, Yan Xu and Wenwen Chen.


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In vitro anticancer effects of two new potent hydrazide compounds in leukemic cells


Shahrzad Tavakolfar, Elham Musavi, Ali Almasirad, Amir Amanzadeh, Seyyed Mohamamd Atyabi, Parichehr Yaghamii, Somayeh Samiee-Sadr and Mona Salimi.


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Autophagy inhibits apoptosis induced by agrocybe aegerita lectin in hepatocellular carcinoma


Wei Liu, Guojun Yu, Wenhui Yu, Xiangdong Ye, Yanxia Jin, Alok Shrestha, Qing Yang and Hui Sun.


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Brain-metastatic breast cancer: clinical considerations and pharmacological approaches


Ana Carolina Andrade, Daniel Sartori Ferruzzi and Carolina Panis.


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Anticancer drug combinations, how far we can go through?


Da-Yong Lu, En-Hong Chen, Hong-Ying Wu, Ting-Ren Lu, Bin Xu and Jian Ding.


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Synthesis of Icaritin and β-anhydroicaritin Mannich Base Derivatives and Their Cytotoxic Activities on Three Human Cancer Cell Lines


Van-Son Nguyen, Ling Shi, Sheng-Chun Wang and Qiu-An Wang.


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Differential Cytotoxicity, Cellular Uptake, Apoptosis and Inhibition of BRCA1 Expression of BRCA1-Defective and Sporadic Breast Cancer Cells Induced by an Anticancer Ruthenium(II)-Arene Compound, RAPTA-EA1


Adisorn Ratanaphan, Tidarat Nhukeaw, Khwanjira Hongthong and Paul J Dyson.


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Effects of Epirubicin and Cisplatin against 4T1 Breast Cancer Cells are Enhanced by Myrtucommulone-A


Kenan izgi, Banu iskender, Cagri Sakalar, Aslıhan Arslanhan, Esra Hilal Yüksek, Esra Hizar and Halit Canatan.


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Synthesis and in vitro evaluation of the anticancer potential of new aminoalkanol derivatives of xanthone


Natalia Szkaradek, Daniel Sypniewski, Anna M. Waszkielewicz, Agnieszka Gunia-Krzyżak, Anna Galilejczyk, Sabina Gałka, Henryk Marona and Ilona Bednarek.


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Inhibitors of Cancer Stem Cells


María E. García-Rubiño, César Lozano-López and Joaquín M Campos.


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Omega-3 polyunsaturated fatty acids enhance cisplatin efficacy in gastric cancer cells by inducing apoptosis via ADORA1


Hong Sheng, Xuehua Chen, Binya Liu, Pu Li and Weixin Cao.


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Synthesis of Methotrexate Loaded Chitosan nanoparticles and in vitro evaluation of the potential in treatment of prostate cancer


Selvi Gunel N, Ozel B, Kipcak S, Aktan C, Akgun C, Ak G, Yilmaz H, Biray Avci C, Dodurga Y and Hamarat Sanlier S.


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HISTAMINE AND HISTAMINERGIC RECEPTORS IN COLORECTAL CANCER: FROM BASIC SCIENCE TO EVIDENCE-BASED MEDICINE


Giuseppe Losurdo, Mariabeatrice Principi, Bruna Girardi, Maria Pricci, Michele Barone, Enzo Ierardi and Alfredo Di Leo.


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Fab(nimotuzumab)-HYNIC-99mTc: Antibody fragmentation for molecular imaging agents


Victoria Calzada, María Fernanda García, Luis Michel Alonso-Martínez, Ximena Camacho, Enzo Goicochea, Marcelo Fernández, Abmel Xiques Castillo, Arlhee Díaz-Miqueli, Normando Iznaga-Escobar, René Leyva Montaña, Omar Alonso, Juan Pablo Gambini and Pablo Cabral.


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Anticancer Vitamin K3 analogues: A review


Kirti D. Badave, Ayesha A. Khan and Sandhya Y Rane.


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New 2-Imino-2H-Chromene-3(N-aryl)carboxamides as potential Cytotoxic Agents.


Rupinder Kaur Gill, Jyoti Kumari and Jitender Bariwal.


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Cytotoxicity and Anti-proliferative Properties of Heterocyclic Compounds Derived from Progesterone


Rafat M. Mohareb, Nadia Y. MegallyAbdo and Abeer A Mohamed.


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α(N)-Heterocyclic Thiosemicarbazones: Iron Chelators That Are Promising for Revival of Gallium in Cancer Chemotherapy


Shuhong Cao, Xiahui Chen, Ligen Chen and Jingwen Chen.


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RADIOPHARMACEUTICALS IN tumor hypoxia imaging: A review focused on MEDICINAL chemiSTRY aspects


Pablo Cabral and Hugo Cerecetto.


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New, Substituted Derivatives of Dicarboximides and their Cytotoxic Properties


Bożena Kuran, Mariola Napiórkowska, Jerzy Kossakowski, Marcin Cieślak, Julia Kaźmierczak-Barańska, Karolina Królewska and Barbara Nawrot.


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The synthetic oleanane triterpenoid HIMOXOL induces autophagy in breast cancer cells via ERK1/2 MAPK pathway and Beclin-1 up-regulation


Natalia Lisiak, Ewa Toton, Blazej Rubis, Barbara Majer and Maria Rybczynska.


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Circulating tumor cells: a new window for diagnosis and evaluation of cancer


Meihui Liu, Min Tang, Ming Li, Feng Gao, Can Shi, Jing Hou and Wenbin Zeng.


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L-Canavanine Potentiates Cytotoxicity of Chemotherapeutic Drugs in Human Breast Cancer Cells


Agustina D. R. Nurcahyanti and Michael Wink.


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Radiolabeled nanoparticles for cancer diagnosis and therapy


Jacek Koziorowski, Adina E. Stanciu, Vanessa Gómez-Vallejo and Jordi Llop.


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Recent advances in heterocyclic tubulin inhibitors targeting the colchicine binding site


Xiaoxin Wu, Qinghui Wang and Wei Li.


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Targeting the Folate Receptor: Effects of Conjugating Folic Acid to DOX Loaded Polymeric Micelles


Mohamed A. Elkhodiry, Ghaleb A Husseini and Diana Velluto.


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Macromolecular Drug Targets in Cancer Treatment and Thiosemicarbazides as Anticancer Agents


Ş. Güniz Küçükgüzela and Göknil Pelin Coşkuna.


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Lenalidomide in an in vitro Dendritic Cell Model for Malignant Gliomas


Caspar D. Kühnöl, Martin S. Staege and Christof M Kramm.


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Design and Synthesis of Some Novel Estrogen Receptor Modulators as Anti-Breast Cancer Agents: In vitro & In vivo Screening, Docking Analysis


Pritam N. Dube and Santosh N Mokale.


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Ethanolic extract of Algerian Propolis and galangin decreased murine melanoma tumour progression


L Benguedouar, M Lahouel, S. C. Gangloff, A Durlach, F Grange, P Bernard and F Antonicelli.


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5' Adenosine Monophosphate-Activated Protein Kinase Modulators as Anticancer Agents


Abhishek Thakur, Nirnoy Dan, Soumendranath Bhakat, Venkatesan Jayaprakash and Sugato Banerjee.


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Review Article: Novel Therapeutic Strategies Against Cancer: Marine-derived Drugs May Be The Answer?


Maria Alessandra Gammone, Graziano Riccioni, Fabio Galvano and Nicolantonio D'Orazio.


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Molecular Mechanisms of Anti-cancer Activities of β-elemene: Targeting Hallmarks of Cancer


Shiyu Jiang, Chunhua Ling, Wei Li, Hongxin Jiang, Qiaoming Zhi and Min Jiang.


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Juglone exerts cytotoxic, anti-proliferative and anti-invasive effects on Glioblastoma multiforme in a cell culture model


Dziugas Meskelevicius, Kastytis Sidlauskas, Ruta Bagdonaviciute, Julius Liobikas and Daiva Majiene.


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Peroxisome Proliferator-activated Receptors and their ligands in cancer drug resistance: opportunity or challenge


Bahman Yousefi, Nosratollah Zarghami, Nasser Samadi and Maryam Majidinia.


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8-bromo-7-methoxychrysin reversed M2 polarization of tumor-associated macrophages induced by liver cancer stem-like cells


Shuwen Sun, Yinghong Cui, Kaiqun Ren, Meifang Quan, Zhenwei Song, Hui Zou, Duo Li, Yu Zheng and Jianguo Cao.


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Fibroblast Growth Factor Receptor (FGFR): A new target for non-small cell lung cancer therapy


Federica Biello, Giovanni Burrafato, Erika Rijavec, Carlo Genova, Giulia Barletta, Anna Truini, Simona Coco, Maria Giovanna Dal Bello, Angela Alama, Francesco Boccardo and Francesco Grossi.


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Synthesis of Combretastatin A-4 analogs and their biological activity


Agnieszka Głowacka, Monika Gensicka, Grzegorz Cholewinski and Krystyna Dzierzbicka.


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Synthesis of New Benzimidazole and Benzothiazole Disulfide Metal Complexes as G-quadruplex Binding Ligands


Kawkab Saour and Dunya Lafta.


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Synthesis of arylamino-1,3,5-triazines functionalized with alkylating 2-chloroethylamine fragment and studies of their cytotoxicity on the breast cancer MCF-7 cell line


Justyna Fraczyk, Beata Kolesinska, Monika Swiontek, Wojciech Lipinski, Danuta Drozdowska and Zbigniew Jerzy Kaminski.


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Docking studies of glutamine valproic acid derivative (S)-5-amino-2-(heptan-4-ylamino)-5-oxopentanoic acid (Gln-VPA) on HDAC8 with biological evaluation in HeLa cells


F Martínez-Ramos, GR Luna-Palencia, I Vásquez-Moctezuma, D Méndez-Luna, MJ Fragoso-Vázquez, J Trujillo-Ferrara, MA Meraz-Ríos, JE Mendieta-Wejebe and J Correa-Basurto.


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Synthesis and Cytotoxicity of Two Active Metabolites of Larotaxel


Jianwei Li, Anping Li, Minghua Li, Yufeng Qiao and Hui Zhang.


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Synthesis of 4-piperidone based curcuminoids with anti-inflammatory and anti-proliferation potential in human cancer cell lines


Amit Anthwal, Kundan Singh, M.S.M. Rawat, Amit K. Tyagi, Ashanul Haque, Imran Ali and Diwan S Rawat.


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Role of carboxypeptidase N invasion and migration in breast cancer


Ranliang Cui, Peng Zhang and Yueguo Li.


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The utility of chemotherapy in the treatment of metastatic prostate cancer


Kanika Gupta, Jacob Elkon, Ehab El-Bahesh and Jeanny B Aragon-Ching.


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Natural Product-Derived Spirooxindole Fragments Serve as Privileged Substructures for Discovery of New Anticancer Agents


Bin Yu, Yi-Chao Zheng, Xiao-Jing Shi, Ping-Ping Qi and Hong-Min Liu.


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Lgr5 contributes to intestinal metaplasia during gastric carcinogenesis: a meta-analysis


Ye Han, Hugang Shen, Xiaofeng Xue, Bin Yuan, Yuting Kuang, Qiaoming Zhi and Hong Zhao.


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The prognostic value of serum LDH levels in patients with hepatocellualr carcinoma after hepatic resection


Wen-Jie Hu, Shun-Jun Fu, Jing-Fang Diao, Dai-Wei Wan, Zhi-Jian Tan, Qiao-Ming Zhi and Jun-Ming He.


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Guaraná a richest caffeine food increase oxaliplatin sensitivity of colorectal HT-29 cells by apoptosis pathway modulation


Francine Carla Cadoná, Alencar Kolinski Machado, Verônica Farina Azzolin, Fernanda Barbisan, Eduardo Bortoluzzi Dornelles, Werner Glanzner, Paulo Bayard Dias Gonçalves, Charles Elias Assmann, Euler Esteves Ribeiro and Ivana Beatrice Mânica da Cruz.


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New Pyrano[2,3-d:6,5-d']dipyrimidine Derivatives - Synthesis, in vitro Cytotoxicity Activity and Computational Studies


Suresh Maddila, Sreekantha B Jonnalagadda, Kovashnee Naicker, Sridevi Gorle, Surjyakant Rana, Kotaiah Yalagala, Surya N. Maddila, Moganavelli Singh and Parvesh Singh.


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A Novel Method to Synthesize 4-Aryl-1H-1,2,3-Triazoles and their Anti-hepatoma Activity


Xiaolong Li, Yun He, Li Hai, Tao Zhang and Yong Wu.


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Blood-Brain Barrier and Breast Cancer Resistance Protein: a limit to the therapy of CNS tumors and neurodegenerative diseases


Anna Lisa Iorio, Martina da Ros, Ornella Fantappiè, Maurizio Lucchesi, Ludovica Facchini, Alessia Stival, Sabrina Becciani, Milena Guidi, Claudio Favre, Maurizio de Martino, Lorenzo Genitori and Iacopo Sardi.


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Yin and yang of polyphenols in cancer prevention. A short review.


Jolie Kiemlian Kwee.


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Long noncoding RNA C21orF96 promotes the migration, invasion and lymph node metastasis in gastric cancer


Ziguo Yang, Qiaoming Zhi, Dan Wang, Li Zhang, Yuting Kuang, Ruizhen Miao, Yulong Shi and Xiaobo Guo.


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Determination of the Antiproliferative Activity of New Theobromine Derivatives and Evaluation of Their In Vitro Hepatotoxic Effects


Maya Georgieva, Magdalena Kondeva-Burdina, Javor Mitkov, Virginia Tzankova, Georgi Momekov and Alexander Zlatkov.


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Chemical Structure Characteristics and Bioactivity of Small Molecule FAK Inhibitors


Fang-Yuan CAO, Xiao-Ping ZHOU, Jing SU, Xiao-Hong YANG, Feng-Hui MU, Jia-Yi SHEN and Wei SUN.


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Nanoliposome is a promising carrier of protein and peptide biomolecule for the treatment of cancer


Tapan Kumar Giri, Ayan Giri, Tapan Kumar Barman and Subhasis Maity.


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Recent Progress of Allicin on Cell Growth Inhibition and Apoptosis in Gastric Cancer Cells


Runlan Luo, Dengyang Fang, Hongdong Hang and Zeyao Tang.


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Leuckart synthesis and pharmacological assessment of novel acetamide derivatives


Priyanka Rani, Dilipkumar Pal, Rahul Rama Hegde and Syed Riaz Hashim.


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Hepato and Cardiotoxicity of Chemotherapeutic Treatment Evaluated by Means of Small Animal Imaging.


Fiorella Carla Tesán, Mariano Portillo, Diego Martinel-Lamas, Vanina Araceli Medina, María Jimena Salgueiro and Marcela Zubillaga.


View Abstract


Nano-Hydroxyapatite Doped with Ho-166 as Drug Delivery System for Bone Cancer Therapy


Franciana Maria Rosa da Silva, Julio Cezar de Almeida Junior, Elizabeth Eugênio de Mello Oliveira, Marta de Souza Albernaz, Alexandre Malta Rossi and Ralph Santos-Oliveira.


View Abstract


PERSPECTIVES OF BENZIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS IN THE NEW ERA


Snehlata Yadav, Balasubramanian Narasimhan and Harmeet kaur.


View Abstract


Biological Potential of Halfsandwich Ruthenium(II) and Iridium(III) Complexes


Gerd Ludwig, Marija Mojić, Mirna Z. Bulatović, Sanja Mijatović, Danijela Maksimović-Ivanić, Dirk Steinborn and Goran N Kaluđerović.


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A review on novel breast cancer therapies: Photodynamic therapy and plant derived agent induced cell death mechanisms


Blassan Plackal Adimuriyil George and Heidi Abrahamse.


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15,16-dihydrotanshinone I induces apoptosis and inhibits the proliferation, migration of human osteosarcoma cell line 143B in vitro


Xuepeng Chen, Qihong Li, Yan He, Hongjiang Du, Zhajun Zhan, Hong zhao, Jiejun Shi, Qingsong Ye and Ji'an Hu.


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Indole-3-ethylsulfamoylphenylacrylamides with Potent Anti-proliferative and Anti-angiogenic Activities


Samir Mehndiratta, Shiow-Lin Pan, Sunil Kumar and Jing-Ping Liou.


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Flavonoids with Therapeutic Potential in Prostate Cancer


Bao Vue, Sheng Zhang and Qiao-Hong Chen.


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Research Progress on the Antitumor Effects of Rhein: Literature Review


Chao Wu, Hongyan Cao, Hua Zhou, Lin Sun, Jingui Xue, Jianyuan Li, Yanqin Bian, Runfei Sun, Shu Dong, Ping Liu and Mingyu Sun.


View Abstract


1, 3, 6-Trihydroxy-7-methyl-9, 10-anthracenedione isolated from genus Lindera with anti-cancer activity


Guoqing Wei, Hui Chen, Fangyuan Nie, Xiaofeng Ma and Hezhong Jiang.


View Abstract


O-6-methylguanine-DNA Methyltransferase Inhibits Gastric Carcinoma Cell Migration and Invasion by Downregulation of Matrix Metalloproteinase 2


Chenglong Li, Li Deng, Qiaoming Zhi, Qingyou Meng, Aimin Qian, Hongfei Sang, Jiazeng Xia and Xiaoqiang Li.


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Isolation, purification and characterization of a novel steroidal saponin cholestanol glucoside from Lasiodiplodia theobromae that induces apoptosis in A549 cells.


Jinu Mathew Valayil, Gini C Kuriakose and Jayabaskaran C.


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Synthesis of Diflunisal thiazolidinones as anticancer agents


Sevil Şenkardeş, Özlem Bingöl Özakpınar, Derya Özsavcı, Azize Şener, Özge Çevik and ŞGüniz Küçükgüzel.


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Up-regulated circulating miR-106a by DNA methylation promised a potential diagnostic and prognostic marker for gastric cancer


Renshun Yuan, Gang Wang, Qiaoming Zhi, Huabin Chen, Ye Han, Bin Wang, Zhongyang Kou, Hao Hu, Zhaoji Guo, Xiaofeng Xue and Hong Zhao.


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Clinical Significance of miR-1826 as a Novel Prognostic Biomarker in Colorectal Cancer


You Hu, Bin Yi, Songbing He, Pengfei Liu, Lei Wang, Jing Yu, Daiwei Wan, Jin Zhou, Xinguo Zhu and Qiaoming Zhi.


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