Home Page ::: Letters in Drug Design & Discovery

ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)


Volume 11, 10 Issues, 2014


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Letters in Drug Design & Discovery

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Editor-in-Chief:

Atta-ur-Rahman

, FRS
Honorary Life Fellow
Kings College
University of Cambridge
Cambridge
UK
Email: lddd@benthamscience.org

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"Letters in Drug Design & Discovery should be available in every library in the pharmaceutical industry and in universities."

R. F. Borne, Associate Director
Laboratory for Applied Drug Design and Synthesis, The University of Mississippi, USA

Authors' Comments
Thank you very much for asking me to give a feedback about the “Letters in Drug Design & Discovery”. I always feel very comfortable whenever I submit any article to publish in this journal.
The review process is fast and sound. I always receive prompt replies from Ms. Aiman Islam and Ambreen Irshad. Both are very sincere and helpful. So far, four of my articles have been published in this journal and hopefully this number will be increased in the coming years. Moreover, I encouraged many of my colleagues to submit their paper in this journal.
Finally, “Letters in Drug Design & Discovery” is a very good journal and I hope to have better relationship in future.

Dr. Imtaiyaz Hassan Hassan
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Letters in Drug Design & Discovery

,

Volume 11

-

Number 9



Synthesis and In vitro Evaluation of Thiadiazole Derivatives as AChE, Bu- ChE and LOX Inhibitors

; Pp: 1062 - 1069

Mehlika Dilek Altintop, Ahmet Ozdemir, Usama Abu Mohsen, Halide Edip Temel, Gulsen Akal n Ciftci and Zafer Asim Kaplancikli


DOI: 10.2174/1570180811666140529004517


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Synthesis and Antifungal Activity of 1,3,4-Thiadiazole Derivatives Containing Pyridine Group

; Pp: 1107 - 1111

Lin-Jiong Zhang, Ming-Yan Yang, Zhao-Hui Sun, Cheng-Xia Tan, Jian-Quan Weng, Hong-Ke Wu and Xing-Hai Liu


DOI: 10.2174/1570180811666140610212731


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Identification of Novel GSK1070916 Analogs as Potential Aurora B Inhibitors: Insights from Molecular Dynamics and MM/GBSA based Rescoring


Faraz Shaikh, Soumendranath Bhakat, Abhishek Thakur, Ashish Radadia, Mahmoud E. S. Soliman and Anamik Shah


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Theoretical Modelling of Potential Chk1 Inhibitors


Pedro M.M. Araújo, Luís Pinto da Silva and Joaquim C.G. Esteves da Silva


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Pd/C-Catalyzed Synthesis of (E)-2-Arylmethylideneindolin-3-ols under Ultrasound: Their Initial Evaluation as Potential Anti-Proliferative Agents


Ponugubati Radhakrishna Murthi, Namburi Suresh, Chekuri Sharmila, Rani, Mandava Venkata Basaveswara Rao and Manojit Pal


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Design, Synthesis and Biological Evaluation of Benzimidazole-Pyridine-Piperidine Hybrids as a new class of potent Antimicrobial Agents


Kothapally Beulah, Akula Ravi Kumar, Boddupally Peda Venkat Lingaiah, Pamulaparthy Shanthan Rao, Banda Narsaiah, Aaramadaka Sunil Kumar Reddy and Upadhyayula Surya Narayana Murty


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Synthesis, Characterization and Microbial Activity of new Bisphenol-CDerivatives


Bhavin B. Dhaduk, Chirag B. Patel and Parsotam H.Parsania


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4-Substituted-2-Methoxyphenol: Suitable Building Block to Prepare New Bioactive Natural-like Hydroxylated Biphenyls


Maria Antonietta Dettori, Davide Fabbri, Marina Pisano, Carla Rozzo, Giuseppe Palmieri, Alessandro Dessì, Roberto Dallocchio and Giovanna Delogu


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Hybrid Pharmacophore Design and Synthesis of Naphthalimide-Benzimidazole Conjugates asPotential Anticancer Agents


Ahmed Kamal, Pogula Praveen Kumar, Mohammed Naseer Ahmed Khan, Bobburi Naga Sheshadri and Olepu Srinivas


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Quantitative Structure – Activity Relationship Study on Saponins as Cytotoxicity Enhancers


Reneta Gevrenova, Alexander Weng, Laurence Voutguenne-Nazabadioko, Mayank Thakur and Irini Doytchinova


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A Divide-and-Conquer Strategy for the Prediction of Protein Contact Map


Cosme E. Santiesteban-Toca, Gerardo M. Casanola-Martin and Jesus S. Aguilar-Ruiz


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Non-Classical Therapeutic Approach in the Treatment of Alzheimer's Disease: A Mini Review


Vladan Bajic, Biljana Spremo-Potparevic, Lada Zivković, Emina Sudar, Sonja Zafirovic, Milan Obradovic and Esma R. Isenovic


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Investigation of new Phenothiazine and Carbazole Derivatives as Potential Inhibitors of Human Farnesyltransferase


Gina-Mirabela Dumitriu, Alina Ghinet, Dalila Belei, Benoît Rigo, Philippe Gautret, Joelle Dubois and Elena Bicu


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Mannich Base Derivatives as the Potential Candidates of Human Topoisomerase II Inhibitors


Huseyin Istanbullu, Muge Senarisoy, Ercin Erciyas and Zeki Topcu


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In Vitro and In Vivo Investigations into the Carbene Copper Bromide Anticancer Drug Candidate WBC4

, 2014 :11(7); 825 - 832

Wolfgang Walther, Iduna Fichtner, Frauke Hackenberg, Wojciech Streciwilk and Matthias Tacke


DOI: 10.2174/1570180811666140529004102
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Modeling the Active Conformation of Human µ Opioid Receptor

, 2014 :11(9); 1053 - 1061

Agnieszka A. Kaczor, Damian Bartuzi and Dariusz Matosiuk


DOI: 10.2174/1570180811666140322001506
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Analysis of Proteasome Inhibition Prediction Using Atom-Based Quadratic Indices Enhanced by Machine Learning Classification Techniques

, 2014 :11(6); 705 - 711

Gerardo M. Casanola-Martin, Huong Le-Thi-Thu, Yovani Marrero-Ponce, Juan A Castillo- Garit, Francisco Torrens, Facundo Perez-Gimenez and Concepcion Abad


DOI: 10.2174/1570180811666140122001144
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Potent Neuroprotective Activity of Monoterpene Derived 4-[(3aR,7aS)- 1,3,3a,4,5,7a-Hexahydro-3,3,6-trimethylisobenzofuran-1-yl]-2-methoxyphenol in MPTP Mice Model

, 2014 :11(5); 611 - 617

Alla V. Pavlova, Irina V. Il'ina, Ekaterina A. Morozova, Dina V. Korchagina, Svetlana Yu. Kurbakova, Irina V. Sorokina, Tatyana G. Tolstikova, Konstantin P. Volcho and Nariman F. Salakhutdinov


DOI: 10.2174/1570180811666131210000316
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Synthesis and Anti-Proliferative Activity of New Biphenyle-Benzylidenethiazolidine- 2,4-dione Bis-Adducts Containing Various Heterocyclic Cores

, 2014 :11(3); 256 - 264

Maxime Meyer, Sandra Kuntz, Isabelle Grillier-Vuissoz, Helene Martin, Lysiane Richert, Stephane Flament, Yves Chapleur and Michel Boisbrun


DOI: 10.2174/15701808113106660080
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Biochemical Changes Evidenced in Alzheimer's Disease: A Mini-Review

, 2014 :11(2); 240 - 248

Luciana Scotti, Francisco Jaime Bezerra Mendonça Junior, Marcelo Sobral da Silva, Ivan R. Pitta and Marcus Tullius Scotti


DOI: 10.2174/15701808113109990063
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