Home Page ::: Letters in Drug Design & Discovery

ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)


Volume 11, 10 Issues, 2014


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Letters in Drug Design & Discovery

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Editor-in-Chief:

Atta-ur-Rahman

, FRS
Honorary Life Fellow
Kings College
University of Cambridge
Cambridge
UK
Email: lddd@benthamscience.org

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Endorsement(s)

"Letters in Drug Design & Discovery should be available in every library in the pharmaceutical industry and in universities."

R. F. Borne, Associate Director
Laboratory for Applied Drug Design and Synthesis, The University of Mississippi, USA

Forthcoming Special Issue(s)

Theoretical Studies for Drug Design derived from natural products: Isolation, Characterization and Biological activity of metabolites in degenerative diseases


Guest Editor(s): Francisco J. Prado-Prado
Tentative Publication Date: November, 2015
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Authors' Comments
Thank you very much for asking me to give a feedback about the “Letters in Drug Design & Discovery”. I always feel very comfortable whenever I submit any article to publish in this journal.
The review process is fast and sound. I always receive prompt replies from Ms. Aiman Islam and Ambreen Irshad. Both are very sincere and helpful. So far, four of my articles have been published in this journal and hopefully this number will be increased in the coming years. Moreover, I encouraged many of my colleagues to submit their paper in this journal.
Finally, “Letters in Drug Design & Discovery” is a very good journal and I hope to have better relationship in future.

Dr. Imtaiyaz Hassan Hassan
Has contributed:

Letters in Drug Design & Discovery

,

Volume 12

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Number 2



Investigation of New Phenothiazine and Carbazole Derivatives as Potential Inhibitors of Human Farnesyltransferase

; Pp: 85 - 92

Gina-Mirabela Dumitriu, Alina Ghinet, Dalila Belei, Benoit Rigo, Philippe Gautret, Joelle Dubois and Elena Bicu


DOI: 10.2174/1570180811666140909010435


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A Divide-and-Conquer Strategy for the Prediction of Protein Contact Map

; Pp: 124 - 130

Cosme E. Santiesteban-Toca, Gerardo M. Casanola-Martin and Jesus S. Aguilar-Ruiz


DOI: 10.2174/1570180811666140909011206


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4-Substituted-2-Methoxyphenol: Suitable Building Block to Prepare New Bioactive Natural-like Hydroxylated Biphenyls

; Pp: 131 - 139

Maria Antonietta Dettori, Davide Fabbri, Marina Pisano, Carla Rozzo, Giuseppe Palmieri, Alessandro Dessi, Roberto Dallocchio and Giovanna Delogu


DOI: 10.2174/1570180811666140915222343


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Discovery of Novel HDAC Inhibitors by Structure-Based Optimization of Cinnamic Hydroxamic Scaffold


Chengqing Ning, Wenyuan Huang, Wen Wu, Cheng Lu, Yujun He, Lei Yao, Lifei Liu, Xiaohe Zhen, Xiaoyu Liu and Niefang Yu


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Development of Structure Activity Correlation Model on Azetidin-2-ones as Tubulin Polymerization Inhibitors


Vijay K. Patel, Kavibhushan S. Chouhan, Avineesh Singh, Deepak K Jain, Ravichandran Veerasamy, Pradeep K. Singour, Rajesh S. Pawar and Harish Rajak


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Synthesis and Biological Activity of Acylthiourea Derivatives Contain 1,2,3-Thiadiazole and 1,3,4-Thiadiazole


Ming-Yan Yang, Wen Zhao, Zhao-Hui Sun, Cheng-Xia Tan, Jian-Quan Weng and Xing-Hai Liu


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6, 7-Dimethoxyquinazolines as Potential Cytotoxic Agents: Synthesis and in Vitro Activity


Mange Ram Yadav, Bishram Singh Chauhan, Prashant Naik, Hardik Gandhi and Rajani Giridhar


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Synthesis of Derivatives of Artesunate α-Aminophosphonate and Their Antimicrobial Activities


Sheng He, Xilin Ouyang, Xiaochao Huang, Weisong Hu, Weilong Dai, Xiaoyan Tian, Yingming Pan, Shiwen Huang and Hengshan Wang


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Promising anticancer drug Candidates based on the 7-Methoxychromone Scaffold: Synthesis and Evaluation of Antiproliferative Activity


Hoang Le Tuan Anh, Nguyen Thi Cuc, Pham Hai Yen, Nguyen Xuan Nhiem, Bui Huu Tai, Do Thi Thao, Nguyen Hoai Nam, Chau Van Minh, Phan Van Kiem and Young Ho Kim


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Design, Synthesis and Biological Evaluation of Novel Fluorinated Heterocyclic Hybrid Molecules based on Triazole & Quinoxaline Scaffolds Lead to Highly Potent Antimalarials and Antibacterials


Adimulam Chandra Shekhar, Boddupally Pedda Venkat Lingaiah, Pamulaparthy Shanthan Rao, Banda Narsaiah, Aparna Devi Allanki and Puran Singh Sijwali


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Synthesis and Anticancer Activity of 7, 8-Dihydroxy-4-Arylcoumarins


Jianrui Wu, Ting Peng, Fang Chen, Yixin Leng, Linjiang Tong, Mengyuan Li, Rong Qu, Hua Xie, Jian Ding and Wenhu Duan


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The Disulfide Analogues of Isophosphoramide Mustard for Anticancer Therapy


Joanna Cytarska, Krzysztof Skowerski, Szymon Jaworski, Konrad Misiura, Beata Filip-Psurska and Joanna Wietrzyk


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First Discovery of Tylophora Alkaloids as HIV Inhibitors


Ziwen Wang, Mingxiao Wang, Lei Wang, Xue Yao, Yue Li, Juan Tan, Wentao Qiao, Yunqi Geng, Yuxiu Liu and Qingmin Wang


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Identification of Pyrazole Derivative as an Antiviral Agent Against Chikungunya Through HTVS


Surender Singh Jadav, Barij Nayan Sinha, Boris Pastorino, Xavier de Lamballerie, Rolf Hilgenfeld and Venkatesan Jayaprakash


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Modeling the Active Conformation of Human µ Opioid Receptor

, 2014; 11(9): 1053 - 1061

Agnieszka A. Kaczor, Damian Bartuzi and Dariusz Matosiuk


DOI: 10.2174/1570180811666140322001506
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In Vitro and In Vivo Investigations into the Carbene Copper Bromide Anticancer Drug Candidate WBC4

, 2014; 11(7): 825 - 832

Wolfgang Walther, Iduna Fichtner, Frauke Hackenberg, Wojciech Streciwilk and Matthias Tacke


DOI: 10.2174/1570180811666140529004102
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Analysis of Proteasome Inhibition Prediction Using Atom-Based Quadratic Indices Enhanced by Machine Learning Classification Techniques

, 2014; 11(6): 705 - 711

Gerardo M. Casanola-Martin, Huong Le-Thi-Thu, Yovani Marrero-Ponce, Juan A Castillo- Garit, Francisco Torrens, Facundo Perez-Gimenez and Concepcion Abad


DOI: 10.2174/1570180811666140122001144
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Potent Neuroprotective Activity of Monoterpene Derived 4-[(3aR,7aS)- 1,3,3a,4,5,7a-Hexahydro-3,3,6-trimethylisobenzofuran-1-yl]-2-methoxyphenol in MPTP Mice Model

, 2014; 11(5): 611 - 617

Alla V. Pavlova, Irina V. Il'ina, Ekaterina A. Morozova, Dina V. Korchagina, Svetlana Yu. Kurbakova, Irina V. Sorokina, Tatyana G. Tolstikova, Konstantin P. Volcho and Nariman F. Salakhutdinov


DOI: 10.2174/1570180811666131210000316
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Synthesis and Anti-Proliferative Activity of New Biphenyle-Benzylidenethiazolidine- 2,4-dione Bis-Adducts Containing Various Heterocyclic Cores

, 2014; 11(3): 256 - 264

Maxime Meyer, Sandra Kuntz, Isabelle Grillier-Vuissoz, Helene Martin, Lysiane Richert, Stephane Flament, Yves Chapleur and Michel Boisbrun


DOI: 10.2174/15701808113106660080
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Biochemical Changes Evidenced in Alzheimer's Disease: A Mini-Review

, 2014; 11(2): 240 - 248

Luciana Scotti, Francisco Jaime Bezerra Mendonça Junior, Marcelo Sobral da Silva, Ivan R. Pitta and Marcus Tullius Scotti


DOI: 10.2174/15701808113109990063
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