E-Pub Articles Ahead of Print ::: Medicinal Chemistry

ISSN: 1875-6638 (Online)
ISSN: 1573-4064 (Print)


Volume 13, 8 Issues, 2017


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Medicinal Chemistry

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Editor-in-Chief:
Atta-ur-Rahman
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Kings College
University of Cambridge
Cambridge
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Email: mc@benthamscience.org

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Articles Ahead of Print

Synthesis and Ativiral Activity of 5-(Benzylthio)-4-carbamyl-1,2,3-triazoles Against Human Cytomegalovirus (CMV) and Varicella-zoster Virus (VZV)


Yi-ning Wen, Zhi-feng Zhang, Ning-ning Liu, Graciela Andrei, Robert Snoeck, Yu-hong Xiang, Dominique Schols, Xue Chen, Zhuo-yong Zhang, Qing-shan Zhang and Qin-pei Wu.


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Additive Effect of MCP in Combination with Cefotaxime Against Staphylococcus aureus


Elias Dahdouh, Salah El-Khatib, Elias Baydoun and Roula M Abdel-Massih.


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A Simple Method to Predict Blood-Brain Barrier Permeability of Drug- Like Compounds Using Classification Trees


Juan A. Castillo-Garit, Gerardo M. Casañola-Martin, Huong Le-Thi-Thu, Hai Pham-The and Stephen J Barigye.


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Prospects of Gene Therapy for Pulmonary Diseases: Progress and Limitations


Garyfalia Karponi, Nikolaos Zogas, Kalliopi Domvri, Paul Zarogoulidis, Georgia Trakada, Stefanos Roumeliotis, Wolfgang Hohenforst-Schmidt, Kaid Darwiche, Lutz Freitag and Konstantinos Zarogoulidis.


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Synthesis and Biological Evaluation of Hybrid 1,5- and 2,5-Disubstituted Indoles as Potentially New Antitubercular Agents


Ana Soares, Mónica S. Estevão, M. Manuel B. Marques, Vasily Kovalishyn, Diogo A.R.S. Latino, João Aires-de-Sousa, Jorge Ramos, Miguel Viveiros and Filomena Martins.


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A Concise Update on the Relevance of Secretory Phospholipase A2 Group IIA and Its Inhibitors to Cancer


Juan Chen, Long Ye, Yu Sun and Yoshikazhu Takada.


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Bioactive Constituents from an Endophytic Fungus, Penicillium polonicum NFW9, Associated with Taxus fauna


Nighat Fatima, Tawanun Sripisut, Ui Joung Youn, Safia Ahmed, Ihsan Ul-Haq, Ulyana Muñoz-Acuña, Charles J. Simmons, Muneer Ahmed Qazi, Muniba Jadoon, Ghee Teng Tan, Esperanza J. Carcache de Blanco and Leng Chee Chang.


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Medicinal Chemistry Approaches of Controlling Gastrointestinal Side Effects of Non-Steroidal Anti-Inflammatory Drugs. Endogenous Protective Mechanisms and Drug Design


Paraskevi Tziona, Panagiotis Theodosis-Nobelos and Eleni A Rekka.


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A New Anti-Aging Lysophosphatidic Acid from Arabidopsis thaliana


Yujuan Sun, Yanhui Wang, Guangfa Wang, Lan Xiang and Jianhua Qi.


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Aryl/heteroaryl Substituted Celecoxib Derivatives as COX-2 Inhibitors: Synthesis, Anti-inflammatory Activity and Molecular Docking Studies


Golla Madhava, Katla Venkata Ramana, Saddala Madhu Sudhana, Devineni Subba Rao, Kuntrapakam Hema Kumar, Valluru Lokanatha, Asupatri Usha Rani and Chamarthi Naga Raju.


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Derivatives of 6-Nitrobenzimidazole Inhibit Fructose-Mediated Protein Glycation and Intracellular Reactive Oxygen Species Production


Humera Jahan, Muhammad Iqbal Choudhary, Zarbad Shah, Khalid M. Khan and Atta-ur-Rahman.


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Effect of Inhibition of Intestinal Cholesterol Absorption on the Prevention of Cholesterol Gallstone Formation


Piero Portincasa and David Q-H Wang.


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Synthesis of Adamantane Aminoethers with Antitubercular Potential


Angeliki-Sofia Foscolos, Ioannis Papanastasiou, Andrew Tsotinis, Nicolas Kolocouris, George B. Foscolos, Anthony Vocat and Stewart T Cole.


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Harmaline and its Derivatives Against the Infectious Multi-Drug Resistant Escherichia coli


Hina Siddiqui, Sehar Tasneem, Saba Farooq, Amtul Sami, Atta -Ur- Rahman and Muhammad Iqbal Choudhary.


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Titanocenes as Anticancer Agents: Recent Insights


Hana Skoupilova, Roman Hrstka and Martin Bartosik.


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Discovery of Flexible Naphthyltriazolylmethane-based Thioacetic Acids as Highly Active Uric Acid Transporter 1 (URAT1) Inhibitors for the Treatment of Hyperuricemia of Gout


Xiansheng Zhang, Jingwei Wu, Wei Liu, Yuqiang Liu, Yafei Xie, Qian Shang, Zhixing Zhou, Weiren Xu, Lida Tang, Jianwu Wang and Guilong Zhao.


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6-benzothiazolyl Ureas, Thioureas and Guanidines are Potent Inhibitors of ABAD/17β-HSD10 and Potential Drugs for Alzheimer’s Disease Treatment: Design, Synthesis and in vitro Evaluation


Ondrej Benek, Lukas Hroch, Laura Aitken, Rafael Dolezal, Patrick Guest, Marketa Benkova, Ondrej Soukup, Karel Musil, Kamil Kuca, Terry K Smith, Frank Gunn-Moore and Kamil Musilek.


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Naphthyridines with Antiviral Activity - A Review


Inder Pal Singh, Sanjay Kumar and Shiv Gupta.


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Nitric Oxide Signaling and the Cross Talk with Prostanoids Pathways in Vascular System


Bruno R. Silva, Tiago D. Paula, Michele Paulo and Lusiane M Bendhack.


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Isolation of Chemical Constituents of Centaurea virgata Lam. and Xanthine Oxidase-Inhibitory Activity of the Plant Extract and Compounds


Burcu S Tuzun, Zsuzsanna Hajdu, Orsolya Orban-Gyapai, Zoltan P Zomborszki, Nikoletta Jedlinszki, Peter Forgo, Bijen Kıvcak and Judit Hohmann.


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Synthesis, Spectroscopic Characterization and Antimicrobial Activities of Benzoxazolone Derivatives


Nida Iqbal Siddiqui, Muhammad Ali Versiani, Khurshid Jawaid, Maryam Shafique, Abdul Hameed, Nida Ambreen, Aneela Karim and Khalid Mohammed Khan.


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Antimicrobial Evaluation of 5-Substituted Aryl 1H-Tetrazoles


Liana Feinn, Joshua Dudley, Adiel Coca and Elizabeth Lewis Roberts.


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Synthesis and Antiproliferative Activity of New pyrazolo[3,4-c]pyridines


Efthymios-Spyridon Gavriil, Nikolaos Lougiakis, Nicole Pouli, Panagiotis Marakos, Alexios-Leandros Skaltsounis, Sangkil Nam, Richard Jove, David Horne, Katerina Gioti, Harris Pratsinis, Dimitris Kletsas and Roxane Tenta.


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Synthesis of Some Steroidal Derivatives with Side Chain of 20- and 22- Hydrazone Aromatic Heterocycles and their Antiproliferative Acitivity


Chunfang Gan, Liang Liu, Jianguo Cui, Zhiping Liu, Haixin Shi, Qifu Lin, Haibing Sheng, Chunhui Yang and Yanmin Huang.


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Elucidation of Antiangiogenic Potential of Vitexin Obtained from Cucumis Sativus Targeting Hsp90 Protein: A Novel Multipathway Targeted Approach to Restrain Angiogenic Phenomena


Neha Sharma, Salman Akhtar, Qazi M. Sajid Jamal, Mohammad A. Kamal, M. Kalim A. Khan, M. Haris Siddiqui and Usman Sayeed.


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A Microwave-Promoted/Assisted Method for Rapid Prepararation of Biaryl Seven-membered Lactones


Chunqi Hu, Jun Li and Wenting Du.


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Molecular Docking and Pharmacophore Modeling Studies of Fluorinated Benzamides as Potential CETP Inhibitors


Reema Abu Khalaf, Sarah Al-Rawashdeh, Dima Sabbah and Ghassan Abu Sheikha.


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Synthesis and Biological Evaluation of Benzophenone Derivatives as Potential HIV-1 Inhibitors


Zhendong Song, Ping Wang, Shanshan Huang, Changyuan Wang, Ruirui Wang, Liumeng Yang, Yuhong Zhen, Kexin Liu, Yongtang Zheng and Xiaodong Ma.


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Synthesis, Antitubercular and Anticancer Activities of p-nitrophenylethylenediamine- Derived Schiff Bases


Raquel S. Amim, Cláudia Pessoa, Maria C. S. Lourenço, Marcus V. N. de Souza and Josane A Lessa.


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Anti-inflammatory and Hypolipidemic Effect of Novel Conjugates with Trolox and Other Antioxidant Acids


Panagiotis Theodosis-Nobelos, Panos N. Kourounakis and Eleni A Rekka.


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Antioxidant and Anticholinesterase Activities of Some Dialkylamino Substituted 3-hydroxyflavone Derivatives


Burcu Culhaoglu, Asli Capan, Mehmet Boga, Mehmet Ozturk, Turan Ozturk and Gulacti Topcu.


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Cytotoxic Phyllactone Analogs from the Marine Sponge Phyllospongia papyrecea


Huawei Zhang, Phillip Crews, Karen Tenney and Frederick A Valeriote.


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Gastrointestinal Motility and Acute Toxicity of Pistagremic acid Isolated from the Galls of Pistacia integerrima


Abdur Rauf, Tareq Abu-Izneid, Aneela Maalik, Saud Bawazeer, Ajmal Khan, Taibi Ben Hadda, Haroon Khan, Mohamed Fawzy Ramadan, Imran Khan, Mohammad S. Mubarak, Ghias Uddin, Alia Bahadar and Umar Farooq.


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Anti-inflammatory, analgesic and anti-ulcerogenic activities of novel bis-thiadiazoles, bis-thiazoles and bis-formazanes


Zeinab A. Muhammad, Ghada S. Masaret, Mohamed M. Amin, Magda A. Abdallah and Thoraya A Farghaly.


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Microwave-assisted Synthesis of 2-Styrylquinoline-4-carboxylic Acids as Antitubercular Agents


Gisela C. Muscia, Silvia E. Asis and Graciela Y Buldain.


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Tamoxifen and Fulvestrant Hybrids Showed Potency as Selective Estrogen Receptor Down-Regulators


Takuji Shoda, Masashi Kato, Takuma Fujisato, Yosuke Demizu, Hideshi Inoue, Mikihiko Naito and Masaaki Kurihara.


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Current medical treatment of early breast cancer


Franco Lumachi.





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