E-Pub Articles Ahead of Print ::: Letters in Drug Design & Discovery

ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)


Volume 12, 10 Issues, 2015


Download PDF Flyer




Letters in Drug Design & Discovery

Aims & ScopeAbstracted/Indexed in


Submit Abstracts Online Submit Manuscripts Online

Editor-in-Chief:
Atta-ur-Rahman, FRS
Honorary Life Fellow
Kings College
University of Cambridge
Cambridge
UK
Email: lddd@benthamscience.org

View Full Editorial Board

Subscribe Purchase Articles Order Reprints

Current: 0.770
5 - Year: 0.757

E-Pub Articles Ahead of Print

Design, Synthesis and Biological Evaluation of4-(Imidazolylmethyl)-2-Aryl-Quinoline Derivatives as Aromatase Inhibitors and Anti-Breast Cancer Agents
Razieh Ghodsi, Ebrahim Azizi, Maria Grazia Ferlin, Vincenzo Pezzi and Afshin Zarghi
View Abstract Purchase Online
Development of Energy-Based Pharmacophore Model and Stepwise Virtual Screening of LRRK2 Inhibitors Through Molecular Dynamics and Mechanics
Sagar S. Bhayye, Kunal Roy and Achintya Saha
View Abstract Purchase Online
Synthesis, Biological Evaluation and Molecular Docking Studies of 4H-Benzo-[h]Chromenes, 7H-Benzo[h]Chromeno[2,3-d]Pyrimidines as Antitumor Agents
Ahmed H. Halawa, Ahmed M. Fouda, Al-Anood M. Al-Dies and Ahmed M. El-Agrody
View Abstract Purchase Online
Evaluation of Serine Protease Inhibitors as Potent FVIIa-sTF Inhibitors in the Blood Coagulation Cascade
Andrea Roxanne J. Anas and Ken-ichi Harada
View Abstract Purchase Online
A Series of 2, 4(1H, 3H)-Quinazolinedione Derivatives: Synthesis and Biological Evaluation as Potential Anticancer Agents
Hulya Akgun, Demet Us Yilmaz, Rengul Cetin Atalay and Damla Gozen
View Abstract Purchase Online
Novel Derivatives of Benfluron and Dimefluron: Synthesis and Anticancer Activity
Lenka Sucha, Marek Kolenic, Jiri Kratochvil, Milan Pour, Milan Nobilis, Eva Cermakova, Martina Rezacova and Pavel Tomsik
View Abstract Purchase Online
Computational Docking Studies of Novel Heterocyclic Carboxamides as Potential PI3Kα Inhibitors
Kamal Sweidan, Dima A. Sabbah, Jorn Engelmann, Heba Abdel-Halim and Ghassan Abu Sheikha
View Abstract Purchase Online
Recent Developments in the Synthesis and Applications of Anticancer Amonafide Derivatives a Mini Review
Gary Gellerman
View Abstract Purchase Online
Effect of Acute Administration of 8-(Trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-amine Hydrochloride (TC-2153) on Biogenic Amines Metabolism in Mouse Brain
Elizabeth A. Kulikova, Ekaterina Y. Bazhenova, Nina K. Popova, Tatyana M. Khomenko, Konstantin P. Volcho, Nariman F. Salakhutdinov and Alexander V. Kulikov
View Abstract Purchase Online
Discovery of New Inhibitors of Urease Enzyme: A Study Using STD-NMR Spectroscopy
Jalaluddin A. J. Awllia, Ayesha Sara, Atia-tul- Wahab, Maryam AL-Ghamdi, Saima Rasheed, Etimad Huwait and M. Iqbal Choudhary
View Abstract Purchase Online
3D-QSAR and Molecular Docking Studies of Flavonoid Derivatives as Potent Acetylcholinesterase Inhibitors
An Zhou, Zeyu Wu, Ailing Hui, Bin Wang, Xianchun Duan, Haixiang Wang and Jian Pan
View Abstract Purchase Online
Syntheses and Activity of Carbohydrate-Containing Chitinase Inhibitors
Gangliang Huang, Xinya Mei, Xin Chen and Feng Xiao
View Abstract Purchase Online
Synthesis, Cytoprotective and Anti-Tumor Activities of Isatin Schiff Bases
Gang Chen, Mei Meng, Yu Zhang, Xiaojiang Hao, Ye Wang and Shuzhen Mu
View Abstract Purchase Online
Design, Synthesis and Evaluation of Novel 9-substituted Carbazole Derivatives as Potential Anticancer Agents
Nitin Kumar and Devender Pathak
View Abstract Purchase Online
In Silico Molecular Interaction Studies of Chiral Heterocyclic Analogs of SAHA as Selective Histone Deacetylase 8 Inhibitors
Appavoo Umamaheswari, Navabshan Irfan and Ayarivan Puratchikody
View Abstract Purchase Online
An Insight into Patents of Fluoroquinolone Derivatives
Prabodh Chander Sharma, Mona Piplani and Harish Rajak
View Abstract Purchase Online
Psychoemotional Background of Temporomandibular Joint Dysfunction and Possible drug Therapy
Pihut Malgorzata, Gierowski Krzysztof, Ceranowicz Piotr and Ferendiuk Ewa
View Abstract Purchase Online
Synthesis and Cytotoxicities of 2-[4-Hydroxy-(3, 5-Bis-Aminomethyl)-Benzylidene]-Indan-1-ones
Mehtap Tugrak, Halise Inci Gul and Hiroshi Sakagami
View Abstract Purchase Online
A Review on Recent Robotic and Analytic Technologies in High Throughput Screening and Synthesis for Drug Discovery
Min Zhu
View Abstract Purchase Online
QSAR Studies on the Bioactivity of Plasmodium Falciparum Glucose-6-Phosphate Dehydrogenase Inhibitors
Xiaoli Hou, Yue Kong, Maolin Wang and Aixia Yan
View Abstract Purchase Online
HIF Inhibitors: New Hope for Cancer Therapy
Mayur Poddar, Tejraj M. Aminabhavi and Malleshappa N. Noolvi
View Abstract Purchase Online
Oxime Carbamates as Potential Insecticidal Agents: Design, Synthesis and Biological Evaluation
Shaoyong Ke, Ziwen Yang, Liqiao Shi, Manli Liu, Ying Liang, Kaimei Wang, Aibing Jiang and Zhigang Zhang
View Abstract Purchase Online
Application of Agents Against Interferon-Gamma-Dependent Chemokines in Immunotherapy
Poupak Fallahi, Silvia Martina Ferrari, Dilia Giuggioli, Clodoveo Ferri and Alessandro Antonelli
View Abstract Purchase Online
Exploring Structure-Based Drug Design for the Development of Multi-Target Antihypertensives
Estella G. da Mota, Elaine F. F. da Cunha and Matheus P. Freitas
View Abstract Purchase Online
Synthesis and Anticancer Activity of 1, 3, 5-Triaryl-1H-Pyrazole
Sajad Ghadbegi, Seyed Nasser Ostad, Abbas Shafiee and Mohsen Amini
View Abstract Purchase Online
Utilization of the DaT-SCAN SPECT in the Diagnosis of Parkinson's Disease in Older Subjects
Fulvio Lauretani, Livia Ruffini, Augusto Scaglioni, Carla Cidda, Chiara Guareschi, Anna Nardelli, Gian Paolo Ceda and Marcello Maggio
View Abstract Purchase Online
In Silicoanalysis of Plasmodium Falciparum Actinand Profilin Interaction at the Interface Region for Antimalarial Design
Asrar Alam, Zahid Kamal and Atiya Fatima
View Abstract Purchase Online
Structure, DNA Binding and Cytotoxicity Studies of [Cu(D-glu)(phen)(H2O)]•NO3•2H2O
Ling Liu, Jie Mou, Youguang Zheng, Tonghui Huang, Shuaishuai Wang and Yi Liu
View Abstract Purchase Online
Synthetic Naphthoflavonoids Showing Inhibitory Effects on Clonogenicity against Cisplatin-Resistant A2780/Cis Human Ovarian Cancer Cells
Yearam Jung, Soon Young Shin, Yeonjoong Yong, Hyuk Yoon, Seunghyun Ahn, Hyeryoung Jung, Dongsoo Koh, Young Han Lee and Yoongho Lim
View Abstract Purchase Online
Synthesis and Cytotoxic Activities of a Curcumin Analogue and Its Mannich Derivatives
Kadir Ozden Yerdelen, Halise Inci Gul, Hiroshi Sakagami, Naoki Umemura, Murat Sukuroglu and Halise Inci Gul
View Abstract Purchase Online
Substrate - Inositol Transporter Interactions: Molecular Docking Study
Mariyana Atanasova and Irini Doytchinova
View Abstract Purchase Online
Preparation and Characterization of CS/(β-CD)/PAA Composite Hydrogels for Controlled Drug Delivery
Jie Ren, Xiaoci Yang, Mengqi Yao, Jinfen Gu, Xiaohua Tang and Wu Yang
View Abstract Purchase Online
Synthesis, Antitumor of New Pyrimidineand Caffeine Derivatives
Ameen Ali Abu-Hashem and Hoda Abdel Raouf Hussein
View Abstract Purchase Online
Design, Synthesis and AntitumorActivities of Bis-arylureas and Bisarylamides Based on 1H-benzo[d]imidazole Moiety as Novel BRaf V600E/VEGFR2 Dual Inhibitors
Weimin Yang, Yadong Chen, Yanmin Zhang, Sanzhi Tang, Hongli Chen, Weifang Tang and Tao Lu
View Abstract Purchase Online
Synthesis and Biological Activity of Thiazole Dithiocarbamate Derivatives
Nalan Gundogdu-Karaburun
View Abstract Purchase Online
Synthesis and Anticancer Activity of Some 2-[3/4-(2-Substituted Phenyl-2- oxoethoxy)benzylidene]-6-substituted-2,3-dihydro-1H-inden-1-one Derivatives
Nalan Gundogdu-Karaburun, Ahmet Cagri Karaburun, Seref Demirayak, Ismail Kayagil and Leyla Yurttas
View Abstract Purchase Online
Synthesis and Biological Evaluation of New Tubulin Inhibitors: Shikonin Thio-glycoside Derivatives
Xiao-Ming Wang, Hong-Yan Lin, Jin-Liang Qi, Li-Fei Bai and Yong-Hua Yang
View Abstract Purchase Online
Fat-Soluble Vitamins Release Based on Clinoptilolite Zeolite as an Oral Drug Delivery System
Mehdi Rahimi, Hamid Mobedi, Aliasghar Behnamghader, Alireza Nateghi Baygi, Houri Mivehchi and Esmaeil Biazar
View Abstract Purchase Online
Synthesis and Biological Evaluations of 3-Benzothiazol-2-yl Coumarin Derivatives as MEK1 Inhibitors
Chao Wang, Fengrong Xu, Yan Niu, Yun Wu, Jing Sun, Yihong Peng, Lei Liang and Ping Xu
View Abstract Purchase Online
Synthesis and Biological Evaluation of Arylthiourea Derivatives with Antitubercular Activity
Rusong Luo, Tuomo Laitinen, Liyan Teng, Tapio Nevalainen, Maija Lahtela-Kakkonen, Baofu Zheng, Honghai Wang, Antti Poso and Xuelian Zhang
View Abstract Purchase Online
Synthesis and Antiproliferative Evaluation of Hybrids of Indolin-2-one and Quinazoline-4(3H)-one Linked via Imine Bond
Wei-Yao Wu, Sheng-Li Cao, Bei-Bei Mao, Ji Liao, Zhong-Feng Li, Hao-Bin Song and Xingzhi Xu
View Abstract Purchase Online
Construction and High Expression of a Recombinant Amino-Proximal HSV-2 Glycoprotein B Polypeptide with Immunogenicity in Escherichia coli
Xu Ning, Tu Jingjing, Wang Xian Yan and Xu Fang
View Abstract Purchase Online
Synthesis and Study of Antitumor Activity of Artimisinin Glucoside
Yanrong Ren and Guoping Chen
View Abstract Purchase Online
Synthesis and Biological Activity of New 2,3-dihydro-1H-cyclopenta[b]- quinoline Derivatives as Acetylcholinesterase Inhibitors
Pawel Szymanski, Magdalena Markowicz, Marek Bajda, Barbara Malawska and Elzbieta Mikiciuk-Olasik
View Abstract Purchase Online
Novel Aminoalcohol Derivatives Bearing 4-Phenylphenol as Antischistosomal Drugs
Li-Ping Duan, Jian Xue, Yi Tao and Hao-Bing Zhang
View Abstract Purchase Online
Deformable Surfactant Vesicles Loading Ammonium Glycyrrhizinate: Characterization and In Vitro Permeation Studies
Luisa Di Marzio, Carlotta Marianecci, Federica Rinaldi, Sara Esposito and Maria Carafa
View Abstract Purchase Online
Advertisement

Related Journals




Related eBooks




Webmaster Contact: urooj@benthamscience.org Copyright © 2015 Bentham Science