E-Pub Articles Ahead of Print ::: Letters in Drug Design & Discovery

ISSN: 1875-628X (Online)
ISSN: 1570-1808 (Print)


Volume 12, 10 Issues, 2015


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Letters in Drug Design & Discovery

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Editor-in-Chief:
Atta-ur-Rahman, FRS
Honorary Life Fellow
Kings College
University of Cambridge
Cambridge
UK
Email: lddd@benthamscience.org

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E-Pub Articles Ahead of Print

In Silico Modeling of Antimalarial Protein Kinase Inhibitors
Rahul Balasaheb Aher and Kunal Roy
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Accumulation Effects of 3-N-Benzyloxycarbonyl-β-Aminobutyric Salicylate on the Alkaloids in Catharanthusroseus Cells
Er-Bing Yang, Yong Wang, Hong-Jun Zang, Zheng-Ming Li and Xing-Hai Liu
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Prediction of Caco-2 Cell Permeability Using Bilinear Indices and Multiple Linear Regression
Huong Le-Thi-Thu, Yudith Canizares-Carmenate, Yovani Marrero-Ponce, Francisco Torrens and Juan A. Castillo-Garit
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Curcumin: the Yellow Molecule with Pleiotropic Biological Effects
Prabhakar Singh, Kanti Bhooshan Pandey and Syed Ibrahim Rizvi
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Application of Sustained-release Carrier of NanoAg-Epidermal Growth Factor in Promoting Refractory Diabetic Wound Healing
Ning-ning Tang, Feng Hu, Jin-yan Liu, Can Liu, Chao-qi Yin, Yong Chen and Jian-da Zhou
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Synthesis of 4-Phenylthieno[2,3-e][1,2,4]triazolo[4,3-a]pyrimidine-5(4H)-one Derivatives and Evaluation of Their Anti-inflammatory Activity
Fu-Jun Pan, Shi-Ben Wang, Da-Chuan Liu, Guo-Hua Gong and Zhe-Shan Quan
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Design and Synthesis of Novel Spiro-Piperidinyl Pyrazolone Derivatives and Their Potential Antiviral Activity
Rajagopalan Srinivasan, Badiadka Narayana, Balladka Kunhanna Sarojini, Veerakyathappa Bhanuprakash and Chenna Govindaraju Darshan Raj
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Molecular Simulation of HDAC1/3 Inhibitor: Insights into the Structural Basis of Selectivity
Lei Zhang and Lihui Zhang
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Novel Aminopeptidase N Inhibitors with Improved Antitumor Activities
Qiang Wang, Qiao Shi and Lu Huang
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Studies on the IC50 of Trisubstituted Thiazoles as Cdc7 Kinase Inhibitors
Huazhen Yang, Xun Liu, Zhiling Ye, Fucheng Song, Lianhua Cui, Zhuang Yu, Hongzong Si and Honglin Zhai
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Design, Synthesis and Biological Evaluation of4-(Imidazolylmethyl)-2-Aryl-Quinoline Derivatives as Aromatase Inhibitors and Anti-Breast Cancer Agents
Razieh Ghodsi, Ebrahim Azizi, Maria Grazia Ferlin, Vincenzo Pezzi and Afshin Zarghi
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Development of Energy-Based Pharmacophore Model and Stepwise Virtual Screening of LRRK2 Inhibitors Through Molecular Dynamics and Mechanics
Sagar S. Bhayye, Kunal Roy and Achintya Saha
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Synthesis, Biological Evaluation and Molecular Docking Studies of 4H-Benzo-[h]Chromenes, 7H-Benzo[h]Chromeno[2,3-d]Pyrimidines as Antitumor Agents
Ahmed H. Halawa, Ahmed M. Fouda, Al-Anood M. Al-Dies and Ahmed M. El-Agrody
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Evaluation of Serine Protease Inhibitors as Potent FVIIa-sTF Inhibitors in the Blood Coagulation Cascade
Andrea Roxanne J. Anas and Ken-ichi Harada
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A Series of 2, 4(1H, 3H)-Quinazolinedione Derivatives: Synthesis and Biological Evaluation as Potential Anticancer Agents
Hulya Akgun, Demet Us Yilmaz, Rengul Cetin Atalay and Damla Gozen
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Novel Derivatives of Benfluron and Dimefluron: Synthesis and Anticancer Activity
Lenka Sucha, Marek Kolenic, Jiri Kratochvil, Milan Pour, Milan Nobilis, Eva Cermakova, Martina Rezacova and Pavel Tomsik
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Computational Docking Studies of Novel Heterocyclic Carboxamides as Potential PI3Kα Inhibitors
Kamal Sweidan, Dima A. Sabbah, Jorn Engelmann, Heba Abdel-Halim and Ghassan Abu Sheikha
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Recent Developments in the Synthesis and Applications of Anticancer Amonafide Derivatives a Mini Review
Gary Gellerman
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Effect of Acute Administration of 8-(Trifluoromethyl)-1,2,3,4,5-benzopentathiepin-6-amine Hydrochloride (TC-2153) on Biogenic Amines Metabolism in Mouse Brain
Elizabeth A. Kulikova, Ekaterina Y. Bazhenova, Nina K. Popova, Tatyana M. Khomenko, Konstantin P. Volcho, Nariman F. Salakhutdinov and Alexander V. Kulikov
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Discovery of New Inhibitors of Urease Enzyme: A Study Using STD-NMR Spectroscopy
Jalaluddin A. J. Awllia, Ayesha Sara, Atia-tul- Wahab, Maryam AL-Ghamdi, Saima Rasheed, Etimad Huwait and M. Iqbal Choudhary
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3D-QSAR and Molecular Docking Studies of Flavonoid Derivatives as Potent Acetylcholinesterase Inhibitors
An Zhou, Zeyu Wu, Ailing Hui, Bin Wang, Xianchun Duan, Haixiang Wang and Jian Pan
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Syntheses and Activity of Carbohydrate-Containing Chitinase Inhibitors
Gangliang Huang, Xinya Mei, Xin Chen and Feng Xiao
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Synthesis, Cytoprotective and Anti-Tumor Activities of Isatin Schiff Bases
Gang Chen, Mei Meng, Yu Zhang, Xiaojiang Hao, Ye Wang and Shuzhen Mu
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Design, Synthesis and Evaluation of Novel 9-substituted Carbazole Derivatives as Potential Anticancer Agents
Nitin Kumar and Devender Pathak
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In Silico Molecular Interaction Studies of Chiral Heterocyclic Analogs of SAHA as Selective Histone Deacetylase 8 Inhibitors
Appavoo Umamaheswari, Navabshan Irfan and Ayarivan Puratchikody
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An Insight into Patents of Fluoroquinolone Derivatives
Prabodh Chander Sharma, Mona Piplani and Harish Rajak
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Psychoemotional Background of Temporomandibular Joint Dysfunction and Possible drug Therapy
Pihut Malgorzata, Gierowski Krzysztof, Ceranowicz Piotr and Ferendiuk Ewa
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Synthesis and Cytotoxicities of 2-[4-Hydroxy-(3, 5-Bis-Aminomethyl)-Benzylidene]-Indan-1-ones
Mehtap Tugrak, Halise Inci Gul and Hiroshi Sakagami
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A Review on Recent Robotic and Analytic Technologies in High Throughput Screening and Synthesis for Drug Discovery
Min Zhu
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QSAR Studies on the Bioactivity of Plasmodium Falciparum Glucose-6-Phosphate Dehydrogenase Inhibitors
Xiaoli Hou, Yue Kong, Maolin Wang and Aixia Yan
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HIF Inhibitors: New Hope for Cancer Therapy
Mayur Poddar, Tejraj M. Aminabhavi and Malleshappa N. Noolvi
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Oxime Carbamates as Potential Insecticidal Agents: Design, Synthesis and Biological Evaluation
Shaoyong Ke, Ziwen Yang, Liqiao Shi, Manli Liu, Ying Liang, Kaimei Wang, Aibing Jiang and Zhigang Zhang
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Application of Agents Against Interferon-Gamma-Dependent Chemokines in Immunotherapy
Poupak Fallahi, Silvia Martina Ferrari, Dilia Giuggioli, Clodoveo Ferri and Alessandro Antonelli
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Exploring Structure-Based Drug Design for the Development of Multi-Target Antihypertensives
Estella G. da Mota, Elaine F. F. da Cunha and Matheus P. Freitas
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Synthesis and Anticancer Activity of 1, 3, 5-Triaryl-1H-Pyrazole
Sajad Ghadbegi, Seyed Nasser Ostad, Abbas Shafiee and Mohsen Amini
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Preparation and Characterization of CS/(β-CD)/PAA Composite Hydrogels for Controlled Drug Delivery
Jie Ren, Xiaoci Yang, Mengqi Yao, Jinfen Gu, Xiaohua Tang and Wu Yang
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Synthesis, Antitumor of New Pyrimidineand Caffeine Derivatives
Ameen Ali Abu-Hashem and Hoda Abdel Raouf Hussein
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Design, Synthesis and AntitumorActivities of Bis-arylureas and Bisarylamides Based on 1H-benzo[d]imidazole Moiety as Novel BRaf V600E/VEGFR2 Dual Inhibitors
Weimin Yang, Yadong Chen, Yanmin Zhang, Sanzhi Tang, Hongli Chen, Weifang Tang and Tao Lu
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Synthesis and Biological Activity of Thiazole Dithiocarbamate Derivatives
Nalan Gundogdu-Karaburun
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Synthesis and Anticancer Activity of Some 2-[3/4-(2-Substituted Phenyl-2- oxoethoxy)benzylidene]-6-substituted-2,3-dihydro-1H-inden-1-one Derivatives
Nalan Gundogdu-Karaburun, Ahmet Cagri Karaburun, Seref Demirayak, Ismail Kayagil and Leyla Yurttas
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Synthesis and Biological Evaluation of New Tubulin Inhibitors: Shikonin Thio-glycoside Derivatives
Xiao-Ming Wang, Hong-Yan Lin, Jin-Liang Qi, Li-Fei Bai and Yong-Hua Yang
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Fat-Soluble Vitamins Release Based on Clinoptilolite Zeolite as an Oral Drug Delivery System
Mehdi Rahimi, Hamid Mobedi, Aliasghar Behnamghader, Alireza Nateghi Baygi, Houri Mivehchi and Esmaeil Biazar
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Synthesis and Biological Evaluations of 3-Benzothiazol-2-yl Coumarin Derivatives as MEK1 Inhibitors
Chao Wang, Fengrong Xu, Yan Niu, Yun Wu, Jing Sun, Yihong Peng, Lei Liang and Ping Xu
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Synthesis and Biological Evaluation of Arylthiourea Derivatives with Antitubercular Activity
Rusong Luo, Tuomo Laitinen, Liyan Teng, Tapio Nevalainen, Maija Lahtela-Kakkonen, Baofu Zheng, Honghai Wang, Antti Poso and Xuelian Zhang
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Synthesis and Antiproliferative Evaluation of Hybrids of Indolin-2-one and Quinazoline-4(3H)-one Linked via Imine Bond
Wei-Yao Wu, Sheng-Li Cao, Bei-Bei Mao, Ji Liao, Zhong-Feng Li, Hao-Bin Song and Xingzhi Xu
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Construction and High Expression of a Recombinant Amino-Proximal HSV-2 Glycoprotein B Polypeptide with Immunogenicity in Escherichia coli
Xu Ning, Tu Jingjing, Wang Xian Yan and Xu Fang
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Synthesis and Study of Antitumor Activity of Artimisinin Glucoside
Yanrong Ren and Guoping Chen
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Synthesis and Biological Activity of New 2,3-dihydro-1H-cyclopenta[b]- quinoline Derivatives as Acetylcholinesterase Inhibitors
Pawel Szymanski, Magdalena Markowicz, Marek Bajda, Barbara Malawska and Elzbieta Mikiciuk-Olasik
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Novel Aminoalcohol Derivatives Bearing 4-Phenylphenol as Antischistosomal Drugs
Li-Ping Duan, Jian Xue, Yi Tao and Hao-Bing Zhang
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Deformable Surfactant Vesicles Loading Ammonium Glycyrrhizinate: Characterization and In Vitro Permeation Studies
Luisa Di Marzio, Carlotta Marianecci, Federica Rinaldi, Sara Esposito and Maria Carafa
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